Compile Data Set for Download or QSAR
Report error Found 114 Enz. Inhib. hit(s) with all data for entry = 50033272
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342582BDBM50342582((E)-4-chloro-3-(2-(4-chlorophenyl)-2-oxoethylidene...)
Affinity DataIC50: 90nMAssay Description:Inhibition of human transglutaminase 2 using ZGBC as a substrate after 30 to 60 mins by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342570BDBM50342570((E)-4-bromo-3-(2-oxo-2-(pyridin-3-yl)ethylidene)in...)
Affinity DataKi:  250nMAssay Description:Inhibition of human transglutaminase 2 using ZGBC as a substrate after 30 to 60 mins by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342568BDBM50342568((E)-1-benzyl-4-chloro-3-(2-oxo-2-(pyridin-3-yl)eth...)
Affinity DataIC50: 360nMAssay Description:Inhibition of human transglutaminase 2 using ZGBC as a substrate after 30 to 60 mins by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342554BDBM50342554((E)-6-bromo-3-(2-oxo-2-(pyridin-3-yl)ethylidene)in...)
Affinity DataIC50: 360nMAssay Description:Inhibition of human transglutaminase 2 using ZGBC as a substrate after 30 to 60 mins by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342570BDBM50342570((E)-4-bromo-3-(2-oxo-2-(pyridin-3-yl)ethylidene)in...)
Affinity DataKi:  400nMAssay Description:Inhibition of human transglutaminase 2 using Cbz-Gln-Gly as a substrate by GDH-coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342568BDBM50342568((E)-1-benzyl-4-chloro-3-(2-oxo-2-(pyridin-3-yl)eth...)
Affinity DataKi:  410nMAssay Description:Inhibition of human transglutaminase 2 using Cbz-Gln-Gly as a substrate by GDH-coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342571BDBM50342571((E)-5-bromo-3-(2-oxo-2-(pyridin-3-yl)ethylidene)in...)
Affinity DataIC50: 560nMAssay Description:Inhibition of human transglutaminase 2 using ZGBC as a substrate after 30 to 60 mins by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342590BDBM50342590((E)-4-chloro-3-(2-oxo-2-(pyridin-3-yl)ethylidene)-...)
Affinity DataIC50: 570nMAssay Description:Inhibition of human transglutaminase 2 using ZGBC as a substrate after 30 to 60 mins by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342597BDBM50342597((E)-methyl 4-((4-chloro-2-oxo-3-(2-oxo-2-(pyridin-...)
Affinity DataIC50: 660nMAssay Description:Inhibition of human transglutaminase 2 using ZGBC as a substrate after 30 to 60 mins by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342571BDBM50342571((E)-5-bromo-3-(2-oxo-2-(pyridin-3-yl)ethylidene)in...)
Affinity DataKi:  680nMAssay Description:Inhibition of human transglutaminase 2 using ZGBC as a substrate after 30 to 60 mins by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342562BDBM50342562((E)-4-chloro-3-(2-oxopropylidene)indolin-2-one | C...)
Affinity DataKi:  700nMAssay Description:Inhibition of human transglutaminase 2 using Cbz-Gln-Gly as a substrate by GDH-coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342581BDBM50342581((E)-4-chloro-3-(2-(3-chlorophenyl)-2-oxoethylidene...)
Affinity DataIC50: 700nMAssay Description:Inhibition of human transglutaminase 2 using Cbz-Gln-Gly as a substrate by GDH-coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342583BDBM50342583((E)-4-chloro-3-(2-(2-methoxyphenyl)-2-oxoethyliden...)
Affinity DataIC50: 740nMAssay Description:Inhibition of human transglutaminase 2 using ZGBC as a substrate after 30 to 60 mins by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342590BDBM50342590((E)-4-chloro-3-(2-oxo-2-(pyridin-3-yl)ethylidene)-...)
Affinity DataIC50: 800nMAssay Description:Inhibition of human transglutaminase 2 using Cbz-Gln-Gly as a substrate by GDH-coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342582BDBM50342582((E)-4-chloro-3-(2-(4-chlorophenyl)-2-oxoethylidene...)
Affinity DataIC50: 800nMAssay Description:Inhibition of human transglutaminase 2 using Cbz-Gln-Gly as a substrate by GDH-coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342577BDBM50342577((E)-4-chloro-3-(2-oxo-2-(pyridin-2-yl)ethylidene)i...)
Affinity DataIC50: 890nMAssay Description:Inhibition of human transglutaminase 2 using ZGBC as a substrate after 30 to 60 mins by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342563BDBM50342563((E)-5-chloro-3-(2-oxopropylidene)indolin-2-one | C...)
Affinity DataKi:  900nMAssay Description:Inhibition of human transglutaminase 2 using Cbz-Gln-Gly as a substrate by GDH-coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342565BDBM50342565((E)-4-chloro-3-(2-oxo-2-(pyridin-3-yl)ethylidene)i...)
Affinity DataIC50: 900nMAssay Description:Inhibition of human transglutaminase 2 using Cbz-Gln-Gly as a substrate by GDH-coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342570BDBM50342570((E)-4-bromo-3-(2-oxo-2-(pyridin-3-yl)ethylidene)in...)
Affinity DataIC50: 900nMAssay Description:Inhibition of human transglutaminase 2 using Cbz-Gln-Gly as a substrate by GDH-coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342583BDBM50342583((E)-4-chloro-3-(2-(2-methoxyphenyl)-2-oxoethyliden...)
Affinity DataIC50: 900nMAssay Description:Inhibition of human transglutaminase 2 using Cbz-Gln-Gly as a substrate by GDH-coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342580BDBM50342580((E)-4-chloro-3-(2-(6-methoxypyridin-3-yl)-2-oxoeth...)
Affinity DataIC50: 950nMAssay Description:Inhibition of human transglutaminase 2 using ZGBC as a substrate after 30 to 60 mins by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342579BDBM50342579((E)-3-(2-(5-bromopyridin-3-yl)-2-oxoethylidene)-4-...)
Affinity DataIC50: 970nMAssay Description:Inhibition of human transglutaminase 2 using ZGBC as a substrate after 30 to 60 mins by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342570BDBM50342570((E)-4-bromo-3-(2-oxo-2-(pyridin-3-yl)ethylidene)in...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human transglutaminase 2 using ZGBC as a substrate after 30 to 60 mins by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342589BDBM50342589((E)-4-chloro-1-isobutyl-3-(2-oxo-2-(pyridin-3-yl)e...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human transglutaminase 2 using Cbz-Gln-Gly as a substrate by GDH-coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342568BDBM50342568((E)-1-benzyl-4-chloro-3-(2-oxo-2-(pyridin-3-yl)eth...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of human transglutaminase 2 using ZGBC as a substrate after 30 to 60 mins by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342578BDBM50342578((E)-4-chloro-3-(2-oxo-2-(pyridin-4-yl)ethylidene)i...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human transglutaminase 2 using ZGBC as a substrate after 30 to 60 mins by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342593BDBM50342593((E)-4-chloro-3-(2-oxo-2-(pyridin-3-yl)ethylidene)-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human transglutaminase 2 using ZGBC as a substrate after 30 to 60 mins by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342584BDBM50342584((E)-4-chloro-3-(2-(3-methoxyphenyl)-2-oxoethyliden...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human transglutaminase 2 using Cbz-Gln-Gly as a substrate by GDH-coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342577BDBM50342577((E)-4-chloro-3-(2-oxo-2-(pyridin-2-yl)ethylidene)i...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human transglutaminase 2 using Cbz-Gln-Gly as a substrate by GDH-coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342584BDBM50342584((E)-4-chloro-3-(2-(3-methoxyphenyl)-2-oxoethyliden...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human transglutaminase 2 using ZGBC as a substrate after 30 to 60 mins by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342585BDBM50342585((E)-4-chloro-3-(2-(4-methoxyphenyl)-2-oxoethyliden...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human transglutaminase 2 using Cbz-Gln-Gly as a substrate by GDH-coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342587BDBM50342587((E)-3-(2-(4-aminophenyl)-2-oxoethylidene)-4-chloro...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human transglutaminase 2 using Cbz-Gln-Gly as a substrate by GDH-coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342596BDBM50342596((E)-methyl 3-((4-chloro-2-oxo-3-(2-oxo-2-(pyridin-...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human transglutaminase 2 using Cbz-Gln-Gly as a substrate by GDH-coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342578BDBM50342578((E)-4-chloro-3-(2-oxo-2-(pyridin-4-yl)ethylidene)i...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human transglutaminase 2 using Cbz-Gln-Gly as a substrate by GDH-coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342598BDBM50342598((E)-5-chloro-3-(2-oxo-2-(pyridin-3-yl)ethylidene)i...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human transglutaminase 2 using ZGBC as a substrate after 30 to 60 mins by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342597BDBM50342597((E)-methyl 4-((4-chloro-2-oxo-3-(2-oxo-2-(pyridin-...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human transglutaminase 2 using Cbz-Gln-Gly as a substrate by GDH-coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342585BDBM50342585((E)-4-chloro-3-(2-(4-methoxyphenyl)-2-oxoethyliden...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human transglutaminase 2 using ZGBC as a substrate after 30 to 60 mins by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342565BDBM50342565((E)-4-chloro-3-(2-oxo-2-(pyridin-3-yl)ethylidene)i...)
Affinity DataKi:  1.30E+3nMAssay Description:Inhibition of human transglutaminase 2 using Cbz-Gln-Gly as a substrate by GDH-coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342593BDBM50342593((E)-4-chloro-3-(2-oxo-2-(pyridin-3-yl)ethylidene)-...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human transglutaminase 2 using Cbz-Gln-Gly as a substrate by GDH-coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342579BDBM50342579((E)-3-(2-(5-bromopyridin-3-yl)-2-oxoethylidene)-4-...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human transglutaminase 2 using Cbz-Gln-Gly as a substrate by GDH-coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342580BDBM50342580((E)-4-chloro-3-(2-(6-methoxypyridin-3-yl)-2-oxoeth...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human transglutaminase 2 using Cbz-Gln-Gly as a substrate by GDH-coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342588BDBM50342588((E)-4-chloro-1-isopropyl-3-(2-oxo-2-(pyridin-3-yl)...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human transglutaminase 2 using Cbz-Gln-Gly as a substrate by GDH-coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342586BDBM50342586((E)-3-(2-(3-aminophenyl)-2-oxoethylidene)-4-chloro...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human transglutaminase 2 using Cbz-Gln-Gly as a substrate by GDH-coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342568BDBM50342568((E)-1-benzyl-4-chloro-3-(2-oxo-2-(pyridin-3-yl)eth...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human transglutaminase 2 using Cbz-Gln-Gly as a substrate by GDH-coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342592BDBM50342592((E)-4-chloro-3-(2-oxo-2-(pyridin-3-yl)ethylidene)-...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human transglutaminase 2 using Cbz-Gln-Gly as a substrate by GDH-coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342554BDBM50342554((E)-6-bromo-3-(2-oxo-2-(pyridin-3-yl)ethylidene)in...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human transglutaminase 2 using Cbz-Gln-Gly as a substrate by GDH-coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342562BDBM50342562((E)-4-chloro-3-(2-oxopropylidene)indolin-2-one | C...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human transglutaminase 2 using Cbz-Gln-Gly as a substrate by GDH-coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342588BDBM50342588((E)-4-chloro-1-isopropyl-3-(2-oxo-2-(pyridin-3-yl)...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human transglutaminase 2 using ZGBC as a substrate after 30 to 60 mins by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342555BDBM50342555((E)-7-chloro-3-(2-oxo-2-(pyridin-3-yl)ethylidene)i...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human transglutaminase 2 using ZGBC as a substrate after 30 to 60 mins by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Stanford University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342552BDBM50342552((E)-5-nitro-3-(2-oxo-2-(pyridin-3-yl)ethylidene)in...)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of human transglutaminase 2 using ZGBC as a substrate after 30 to 60 mins by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
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