TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Vanderbilt Medical Center
Curated by ChEMBL
Vanderbilt Medical Center
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:Antagonist activity against mGlu5 receptor assessed as inhibition of calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Vanderbilt Medical Center
Curated by ChEMBL
Vanderbilt Medical Center
Curated by ChEMBL
Affinity DataIC50: 660nMAssay Description:Antagonist activity against mGlu5 receptor assessed as inhibition of calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Vanderbilt Medical Center
Curated by ChEMBL
Vanderbilt Medical Center
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulation of mGlu5 receptor assessed as calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Vanderbilt Medical Center
Curated by ChEMBL
Vanderbilt Medical Center
Curated by ChEMBL
Affinity DataEC50: 470nMAssay Description:Positive allosteric modulation of mGlu5 receptor assessed as calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Vanderbilt Medical Center
Curated by ChEMBL
Vanderbilt Medical Center
Curated by ChEMBL
Affinity DataEC50: 850nMAssay Description:Positive allosteric modulation of mGlu5 receptor assessed as calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Vanderbilt Medical Center
Curated by ChEMBL
Vanderbilt Medical Center
Curated by ChEMBL
Affinity DataEC50: 290nMAssay Description:Positive allosteric modulation of mGlu5 receptor assessed as calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Vanderbilt Medical Center
Curated by ChEMBL
Vanderbilt Medical Center
Curated by ChEMBL
Affinity DataEC50: 54nMAssay Description:Positive allosteric modulation of mGlu5 receptor assessed as calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Vanderbilt Medical Center
Curated by ChEMBL
Vanderbilt Medical Center
Curated by ChEMBL
Affinity DataEC50: 56nMAssay Description:Positive allosteric modulation of mGlu5 receptor assessed as calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Vanderbilt Medical Center
Curated by ChEMBL
Vanderbilt Medical Center
Curated by ChEMBL
Affinity DataEC50: 130nMAssay Description:Positive allosteric modulation of mGlu5 receptor assessed as calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Vanderbilt Medical Center
Curated by ChEMBL
Vanderbilt Medical Center
Curated by ChEMBL
Affinity DataEC50: 5.90nMAssay Description:Positive allosteric modulation of mGlu5 receptor assessed as calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Vanderbilt Medical Center
Curated by ChEMBL
Vanderbilt Medical Center
Curated by ChEMBL
Affinity DataEC50: 870nMAssay Description:Positive allosteric modulation of mGlu5 receptor assessed as calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Vanderbilt Medical Center
Curated by ChEMBL
Vanderbilt Medical Center
Curated by ChEMBL
Affinity DataEC50: 900nMAssay Description:Positive allosteric modulation of mGlu5 receptor assessed as calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Vanderbilt Medical Center
Curated by ChEMBL
Vanderbilt Medical Center
Curated by ChEMBL
Affinity DataEC50: 5.70E+3nMAssay Description:Positive allosteric modulation of mGlu5 receptor assessed as calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Vanderbilt Medical Center
Curated by ChEMBL
Vanderbilt Medical Center
Curated by ChEMBL
Affinity DataEC50: 35nMAssay Description:Positive allosteric modulation of mGlu5 receptor assessed as calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Vanderbilt Medical Center
Curated by ChEMBL
Vanderbilt Medical Center
Curated by ChEMBL
Affinity DataEC50: 170nMAssay Description:Positive allosteric modulation of mGlu5 receptor assessed as calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Vanderbilt Medical Center
Curated by ChEMBL
Vanderbilt Medical Center
Curated by ChEMBL
Affinity DataEC50: 160nMAssay Description:Positive allosteric modulation of mGlu5 receptor assessed as calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Vanderbilt Medical Center
Curated by ChEMBL
Vanderbilt Medical Center
Curated by ChEMBL
Affinity DataEC50: 12nMAssay Description:Positive allosteric modulation of mGlu5 receptor assessed as calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Vanderbilt Medical Center
Curated by ChEMBL
Vanderbilt Medical Center
Curated by ChEMBL
Affinity DataEC50: 51nMAssay Description:Positive allosteric modulation of mGlu5 receptor assessed as calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Vanderbilt Medical Center
Curated by ChEMBL
Vanderbilt Medical Center
Curated by ChEMBL
Affinity DataEC50: 200nMAssay Description:Positive allosteric modulation of mGlu5 receptor assessed as calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Vanderbilt Medical Center
Curated by ChEMBL
Vanderbilt Medical Center
Curated by ChEMBL
Affinity DataEC50: 66nMAssay Description:Positive allosteric modulation of mGlu5 receptor assessed as calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Vanderbilt Medical Center
Curated by ChEMBL
Vanderbilt Medical Center
Curated by ChEMBL
Affinity DataEC50: 350nMAssay Description:Positive allosteric modulation of mGlu5 receptor assessed as calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Vanderbilt Medical Center
Curated by ChEMBL
Vanderbilt Medical Center
Curated by ChEMBL
Affinity DataEC50: 10nMAssay Description:Positive allosteric modulation of mGlu5 receptor assessed as calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Vanderbilt Medical Center
Curated by ChEMBL
Vanderbilt Medical Center
Curated by ChEMBL
Affinity DataEC50: 16nMAssay Description:Positive allosteric modulation of mGlu5 receptor assessed as calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Vanderbilt Medical Center
Curated by ChEMBL
Vanderbilt Medical Center
Curated by ChEMBL
Affinity DataEC50: 50nMAssay Description:Positive allosteric modulation of mGlu5 receptor assessed as calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Vanderbilt Medical Center
Curated by ChEMBL
Vanderbilt Medical Center
Curated by ChEMBL
Affinity DataEC50: 250nMAssay Description:Positive allosteric modulation of mGlu5 receptor assessed as calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Vanderbilt Medical Center
Curated by ChEMBL
Vanderbilt Medical Center
Curated by ChEMBL
Affinity DataEC50: 160nMAssay Description:Positive allosteric modulation of mGlu5 receptor assessed as calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Vanderbilt Medical Center
Curated by ChEMBL
Vanderbilt Medical Center
Curated by ChEMBL
Affinity DataEC50: 96nMAssay Description:Positive allosteric modulation of mGlu5 receptor assessed as calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Vanderbilt Medical Center
Curated by ChEMBL
Vanderbilt Medical Center
Curated by ChEMBL
Affinity DataEC50: 550nMAssay Description:Positive allosteric modulation of mGlu5 receptor assessed as calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Vanderbilt Medical Center
Curated by ChEMBL
Vanderbilt Medical Center
Curated by ChEMBL
Affinity DataEC50: 180nMAssay Description:Positive allosteric modulation of mGlu5 receptor assessed as calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Vanderbilt Medical Center
Curated by ChEMBL
Vanderbilt Medical Center
Curated by ChEMBL
Affinity DataEC50: 270nMAssay Description:Positive allosteric modulation of mGlu5 receptor assessed as calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Vanderbilt Medical Center
Curated by ChEMBL
Vanderbilt Medical Center
Curated by ChEMBL
Affinity DataEC50: 4.00E+3nMAssay Description:Positive allosteric modulation of mGlu5 receptor assessed as calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Vanderbilt Medical Center
Curated by ChEMBL
Vanderbilt Medical Center
Curated by ChEMBL
Affinity DataEC50: 3.60E+3nMAssay Description:Positive allosteric modulation of mGlu5 receptor assessed as calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Vanderbilt Medical Center
Curated by ChEMBL
Vanderbilt Medical Center
Curated by ChEMBL
Affinity DataEC50: 610nMAssay Description:Positive allosteric modulation of mGlu5 receptor assessed as calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Vanderbilt Medical Center
Curated by ChEMBL
Vanderbilt Medical Center
Curated by ChEMBL
Affinity DataEC50: 170nMAssay Description:Positive allosteric modulation of mGlu5 receptor assessed as calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Vanderbilt Medical Center
Curated by ChEMBL
Vanderbilt Medical Center
Curated by ChEMBL
Affinity DataEC50: 260nMAssay Description:Positive allosteric modulation of mGlu5 receptor assessed as calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Vanderbilt Medical Center
Curated by ChEMBL
Vanderbilt Medical Center
Curated by ChEMBL
Affinity DataEC50: 150nMAssay Description:Positive allosteric modulation of mGlu5 receptor assessed as calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Vanderbilt Medical Center
Curated by ChEMBL
Vanderbilt Medical Center
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulation of mGlu5 receptor assessed as calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Vanderbilt Medical Center
Curated by ChEMBL
Vanderbilt Medical Center
Curated by ChEMBL
Affinity DataEC50: 3.40E+3nMAssay Description:Positive allosteric modulation of mGlu5 receptor assessed as calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Vanderbilt Medical Center
Curated by ChEMBL
Vanderbilt Medical Center
Curated by ChEMBL
Affinity DataEC50: 4.90E+3nMAssay Description:Positive allosteric modulation of mGlu5 receptor assessed as calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Vanderbilt Medical Center
Curated by ChEMBL
Vanderbilt Medical Center
Curated by ChEMBL
Affinity DataEC50: 3.70E+3nMAssay Description:Positive allosteric modulation of mGlu5 receptor assessed as calcium mobilizationMore data for this Ligand-Target Pair