Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50034188
TargetMelanocyte-stimulating hormone receptor(Human)
H. Lee Moffitt Cancer Center & Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358559BDBM50358559(CHEMBL1923662)
Affinity DataKi:  0.170nMAssay Description:Displacement of Eu-NDP-alphaMSH from human MC1 receptor expressed in human HCT116 cells after 1.5 hrs by time-resolved fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
H. Lee Moffitt Cancer Center & Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358561BDBM50358561(CHEMBL1923664)
Affinity DataKi:  0.240nMAssay Description:Displacement of Eu-NDP-alphaMSH from human MC1 receptor expressed in human HCT116 cells after 1.5 hrs by time-resolved fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
H. Lee Moffitt Cancer Center & Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358564BDBM50358564(CHEMBL1923667)
Affinity DataKi:  0.710nMAssay Description:Displacement of Eu-NDP-alphaMSH from human MC5 receptor expressed in human HEK293 cells after 1.5 hrs by time-resolved fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
H. Lee Moffitt Cancer Center & Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358562BDBM50358562(CHEMBL1923665)
Affinity DataKi:  0.75nMAssay Description:Displacement of Eu-NDP-alphaMSH from human MC4 receptor expressed in human HEK293 cells after 1.5 hrs by time-resolved fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
H. Lee Moffitt Cancer Center & Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358562BDBM50358562(CHEMBL1923665)
Affinity DataKi:  0.760nMAssay Description:Displacement of Eu-NDP-alphaMSH from human MC5 receptor expressed in human HEK293 cells after 1.5 hrs by time-resolved fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
H. Lee Moffitt Cancer Center & Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358564BDBM50358564(CHEMBL1923667)
Affinity DataKi:  0.770nMAssay Description:Displacement of Eu-NDP-alphaMSH from human MC4 receptor expressed in human HEK293 cells after 1.5 hrs by time-resolved fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
H. Lee Moffitt Cancer Center & Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358563BDBM50358563(CHEMBL1923666)
Affinity DataKi:  1.40nMAssay Description:Displacement of Eu-NDP-alphaMSH from human MC5 receptor expressed in human HEK293 cells after 1.5 hrs by time-resolved fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
H. Lee Moffitt Cancer Center & Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358563BDBM50358563(CHEMBL1923666)
Affinity DataKi:  1.70nMAssay Description:Displacement of Eu-NDP-alphaMSH from human MC4 receptor expressed in human HEK293 cells after 1.5 hrs by time-resolved fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
H. Lee Moffitt Cancer Center & Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121900BDBM50121900(Ac-Ser-Try-Ser-Nle-Glu-His-DPhe-Arg-Trp-Gly-Lys-Pr...)
Affinity DataKi:  1.80nMAssay Description:Displacement of Eu-NDP-alphaMSH from human MC1 receptor expressed in human HCT116 cells after 1.5 hrs by time-resolved fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
H. Lee Moffitt Cancer Center & Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358560BDBM50358560(CHEMBL1923663)
Affinity DataKi:  1.80nMAssay Description:Displacement of Eu-NDP-alphaMSH from human MC1 receptor expressed in human HCT116 cells after 1.5 hrs by time-resolved fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
H. Lee Moffitt Cancer Center & Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358562BDBM50358562(CHEMBL1923665)
Affinity DataKi:  2nMAssay Description:Displacement of Eu-NDP-alphaMSH from human MC1 receptor expressed in human HCT116 cells after 1.5 hrs by time-resolved fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
H. Lee Moffitt Cancer Center & Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358563BDBM50358563(CHEMBL1923666)
Affinity DataKi:  2.60nMAssay Description:Displacement of Eu-NDP-alphaMSH from human MC1 receptor expressed in human HCT116 cells after 1.5 hrs by time-resolved fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
H. Lee Moffitt Cancer Center & Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358565BDBM50358565(CHEMBL1923668)
Affinity DataKi:  3.90nMAssay Description:Displacement of Eu-NDP-alphaMSH from human MC5 receptor expressed in human HEK293 cells after 1.5 hrs by time-resolved fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
H. Lee Moffitt Cancer Center & Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358565BDBM50358565(CHEMBL1923668)
Affinity DataKi:  4.20nMAssay Description:Displacement of Eu-NDP-alphaMSH from human MC1 receptor expressed in human HCT116 cells after 1.5 hrs by time-resolved fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
H. Lee Moffitt Cancer Center & Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358565BDBM50358565(CHEMBL1923668)
Affinity DataKi:  4.40nMAssay Description:Displacement of Eu-NDP-alphaMSH from human MC4 receptor expressed in human HEK293 cells after 1.5 hrs by time-resolved fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
H. Lee Moffitt Cancer Center & Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358564BDBM50358564(CHEMBL1923667)
Affinity DataKi:  5.60nMAssay Description:Displacement of Eu-NDP-alphaMSH from human MC1 receptor expressed in human HCT116 cells after 1.5 hrs by time-resolved fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
H. Lee Moffitt Cancer Center & Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121900BDBM50121900(Ac-Ser-Try-Ser-Nle-Glu-His-DPhe-Arg-Trp-Gly-Lys-Pr...)
Affinity DataKi:  9.90nMAssay Description:Displacement of Eu-NDP-alphaMSH from human MC5 receptor expressed in human HEK293 cells after 1.5 hrs by time-resolved fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
H. Lee Moffitt Cancer Center & Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121900BDBM50121900(Ac-Ser-Try-Ser-Nle-Glu-His-DPhe-Arg-Trp-Gly-Lys-Pr...)
Affinity DataKi:  19nMAssay Description:Displacement of Eu-NDP-alphaMSH from human MC4 receptor expressed in human HEK293 cells after 1.5 hrs by time-resolved fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
H. Lee Moffitt Cancer Center & Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358559BDBM50358559(CHEMBL1923662)
Affinity DataKi:  27nMAssay Description:Displacement of Eu-NDP-alphaMSH from human MC5 receptor expressed in human HEK293 cells after 1.5 hrs by time-resolved fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
H. Lee Moffitt Cancer Center & Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358561BDBM50358561(CHEMBL1923664)
Affinity DataKi:  46nMAssay Description:Displacement of Eu-NDP-alphaMSH from human MC5 receptor expressed in human HEK293 cells after 1.5 hrs by time-resolved fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
H. Lee Moffitt Cancer Center & Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358560BDBM50358560(CHEMBL1923663)
Affinity DataKi:  58nMAssay Description:Displacement of Eu-NDP-alphaMSH from human MC5 receptor expressed in human HEK293 cells after 1.5 hrs by time-resolved fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
H. Lee Moffitt Cancer Center & Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358559BDBM50358559(CHEMBL1923662)
Affinity DataKi:  160nMAssay Description:Displacement of Eu-NDP-alphaMSH from human MC4 receptor expressed in human HEK293 cells after 1.5 hrs by time-resolved fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
H. Lee Moffitt Cancer Center & Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358561BDBM50358561(CHEMBL1923664)
Affinity DataKi:  254nMAssay Description:Displacement of Eu-NDP-alphaMSH from human MC4 receptor expressed in human HEK293 cells after 1.5 hrs by time-resolved fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
H. Lee Moffitt Cancer Center & Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358560BDBM50358560(CHEMBL1923663)
Affinity DataKi:  988nMAssay Description:Displacement of Eu-NDP-alphaMSH from human MC4 receptor expressed in human HEK293 cells after 1.5 hrs by time-resolved fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed