TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Hanyang University
Curated by ChEMBL
Hanyang University
Curated by ChEMBL
TargetProto-oncogene tyrosine-protein kinase ROS(Homo sapiens (Human))
Hanyang University
Curated by ChEMBL
Hanyang University
Curated by ChEMBL
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Hanyang University
Curated by ChEMBL
Hanyang University
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Inhibition of CDK1/Cyclin BMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Hanyang University
Curated by ChEMBL
Hanyang University
Curated by ChEMBL
Affinity DataIC50: 1.90nMAssay Description:Inhibition of CDK2/Cyclin EMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30nMAssay Description:Inhibition of Aurora-AMore data for this Ligand-Target Pair
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Hanyang University
Curated by ChEMBL
Hanyang University
Curated by ChEMBL
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hanyang University
Curated by ChEMBL
Hanyang University
Curated by ChEMBL
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Hanyang University
Curated by ChEMBL
Hanyang University
Curated by ChEMBL
Affinity DataIC50: 4.40nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Hanyang University
Curated by ChEMBL
Hanyang University
Curated by ChEMBL
Affinity DataIC50: 4.90nMAssay Description:Inhibition of human CRAF using [gamma-33P]ATP after 40 mins by scintillation countingMore data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Hanyang University
Curated by ChEMBL
Hanyang University
Curated by ChEMBL
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Hanyang University
Curated by ChEMBL
Hanyang University
Curated by ChEMBL
Affinity DataIC50: 9.20nMAssay Description:Inhibition of GSK3-betaMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Hanyang University
Curated by ChEMBL
Hanyang University
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Hanyang University
Curated by ChEMBL
Hanyang University
Curated by ChEMBL
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
Hanyang University
Curated by ChEMBL
Hanyang University
Curated by ChEMBL
TargetMacrophage-stimulating protein receptor(Homo sapiens (Human))
Hanyang University
Curated by ChEMBL
Hanyang University
Curated by ChEMBL
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Hanyang University
Curated by ChEMBL
Hanyang University
Curated by ChEMBL
Affinity DataIC50: 668nMAssay Description:Inhibition of human CRAF using [gamma-33P]ATP after 40 mins by scintillation countingMore data for this Ligand-Target Pair
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Hanyang University
Curated by ChEMBL
Hanyang University
Curated by ChEMBL
Affinity DataIC50: 961nMAssay Description:Inhibition of human CRAF using [gamma-33P]ATP after 40 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 1.75E+3nMAssay Description:Inhibition of JNK1More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Hanyang University
Curated by ChEMBL
Hanyang University
Curated by ChEMBL
Affinity DataIC50: 2.15E+3nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
Affinity DataIC50: 3.95E+3nMAssay Description:Inhibition of ERK2More data for this Ligand-Target Pair
Affinity DataIC50: 6.80E+3nMAssay Description:Inhibition of MTORMore data for this Ligand-Target Pair