Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 8288
TargetCannabinoid receptor 2(Human)
Cairo University

LigandChemical structure of BindingDB Monomer ID 239146BDBM239146((E)-Ethyl 2-(6-(3,4-dimethoxyphenyl)-4-oxohex-5-en...)
Affinity DataKi: >1.00E+4nM IC50: 1.00E+4nMAssay Description:Membranes from HEK-293 cells transfected with the human recombinant CB1 receptor(Bmax=2.5pmol/mg protein) and human recombinant CB2 receptor (B max=4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Cairo University

LigandChemical structure of BindingDB Monomer ID 239147BDBM239147((E)-6-(3,4-Dimethoxyphenyl)-N-(2-hydroxybutan-2-yl...)
Affinity DataKi: >1.00E+4nM IC50: 1.00E+4nMAssay Description:Membranes from HEK-293 cells transfected with the human recombinant CB1 receptor(Bmax=2.5pmol/mg protein) and human recombinant CB2 receptor (B max=4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Cairo University

LigandChemical structure of BindingDB Monomer ID 239144BDBM239144((E)-N-(4-Hydroxyphenyl)-4-oxo-6-p-tolylhex-5-enami...)
Affinity DataKi: >1.00E+4nM IC50: 1.00E+4nMAssay Description:Membranes from HEK-293 cells transfected with the human recombinant CB1 receptor(Bmax=2.5pmol/mg protein) and human recombinant CB2 receptor (B max=4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Cairo University

LigandChemical structure of BindingDB Monomer ID 239145BDBM239145((E)-6-[4-(Dimethylamino)phenyl]-N-(2-hydroxybutan-...)
Affinity DataKi: >1.00E+4nM IC50: 1.00E+4nMAssay Description:Membranes from HEK-293 cells transfected with the human recombinant CB1 receptor(Bmax=2.5pmol/mg protein) and human recombinant CB2 receptor (B max=4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Cairo University

LigandChemical structure of BindingDB Monomer ID 239142BDBM239142((E)-N-(2-Hydroxybutan-2-yl)-4-oxo-6-p-tolylhex-5-e...)
Affinity DataKi: >1.00E+4nM IC50: 1.00E+4nMAssay Description:Membranes from HEK-293 cells transfected with the human recombinant CB1 receptor(Bmax=2.5pmol/mg protein) and human recombinant CB2 receptor (B max=4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Cairo University

LigandChemical structure of BindingDB Monomer ID 239143BDBM239143((E)-N-(1,3-Dihydroxy-2-(hydroxymethylpropan-2-yl)-...)
Affinity DataKi: >1.00E+4nM IC50: 1.00E+4nMAssay Description:Membranes from HEK-293 cells transfected with the human recombinant CB1 receptor(Bmax=2.5pmol/mg protein) and human recombinant CB2 receptor (B max=4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Cairo University

LigandChemical structure of BindingDB Monomer ID 239140BDBM239140((E)-N-(1,3-Dihydroxy-2-(hydroxymethyl)propan-2-yl)...)
Affinity DataKi: >1.00E+4nM IC50: 1.00E+4nMAssay Description:Membranes from HEK-293 cells transfected with the human recombinant CB1 receptor(Bmax=2.5pmol/mg protein) and human recombinant CB2 receptor (B max=4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Cairo University

LigandChemical structure of BindingDB Monomer ID 239141BDBM239141((E) Ethyl [2-(4-oxo-6-phenylhex)-5-enamido]acetate...)
Affinity DataKi: >1.00E+4nM IC50: 1.00E+4nMAssay Description:Membranes from HEK-293 cells transfected with the human recombinant CB1 receptor(Bmax=2.5pmol/mg protein) and human recombinant CB2 receptor (B max=4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Cairo University

LigandChemical structure of BindingDB Monomer ID 239154BDBM239154(4-Acetamidophenyl 4-(naphthalen-1-ylamino)-4-oxobu...)
Affinity DataKi: >1.00E+4nM IC50: 1.00E+4nMAssay Description:Membranes from HEK-293 cells transfected with the human recombinant CB1 receptor(Bmax=2.5pmol/mg protein) and human recombinant CB2 receptor (B max=4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Cairo University

LigandChemical structure of BindingDB Monomer ID 239152BDBM239152(N-(2-Hydroxybutan-2-yl)-2-(4-naphthalen-1-ylamino)...)
Affinity DataKi: >1.00E+4nM IC50: 1.00E+4nMAssay Description:Membranes from HEK-293 cells transfected with the human recombinant CB1 receptor(Bmax=2.5pmol/mg protein) and human recombinant CB2 receptor (B max=4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Cairo University

LigandChemical structure of BindingDB Monomer ID 239153BDBM239153(Ethyl 2-(4-(naphthalen-1-ylamino)-4-oxobutanamido)...)
Affinity DataKi: >1.00E+4nM IC50: 1.00E+4nMAssay Description:Membranes from HEK-293 cells transfected with the human recombinant CB1 receptor(Bmax=2.5pmol/mg protein) and human recombinant CB2 receptor (B max=4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Cairo University

LigandChemical structure of BindingDB Monomer ID 239150BDBM239150((E)-4-Acetamidophenyl 4-oxo-6-phenylhex-5-enoate (...)
Affinity DataKi: >1.00E+4nM IC50: 1.00E+4nMAssay Description:Membranes from HEK-293 cells transfected with the human recombinant CB1 receptor(Bmax=2.5pmol/mg protein) and human recombinant CB2 receptor (B max=4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Cairo University

LigandChemical structure of BindingDB Monomer ID 239151BDBM239151((E)-6-(Biphenyl-4-yl)-N-(2-hydroxybutan-2-yl)-4-ox...)
Affinity DataKi: >1.00E+4nM IC50: 1.00E+4nMAssay Description:Membranes from HEK-293 cells transfected with the human recombinant CB1 receptor(Bmax=2.5pmol/mg protein) and human recombinant CB2 receptor (B max=4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Cairo University

LigandChemical structure of BindingDB Monomer ID 239148BDBM239148((E)-6-(4-(Benzyloxy)phenyl)-N-(2-hydroxybutan-2-yl...)
Affinity DataKi: >1.00E+4nM IC50: 1.00E+4nMAssay Description:Membranes from HEK-293 cells transfected with the human recombinant CB1 receptor(Bmax=2.5pmol/mg protein) and human recombinant CB2 receptor (B max=4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Cairo University

LigandChemical structure of BindingDB Monomer ID 239149BDBM239149((E)-Ethyl 2-(6-(4-(benzyloxy)phenyl)-4-oxohex-5-en...)
Affinity DataKi: >1.00E+4nM IC50: 1.00E+4nMAssay Description:Membranes from HEK-293 cells transfected with the human recombinant CB1 receptor(Bmax=2.5pmol/mg protein) and human recombinant CB2 receptor (B max=4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Cairo University

LigandChemical structure of BindingDB Monomer ID 239139BDBM239139((E)-N-(2-Hydroxybutan-2-yl)-4-oxo-6-phenylhex-5-en...)
Affinity DataKi: >1.00E+4nM IC50: 1.00E+4nMAssay Description:Membranes from HEK-293 cells transfected with the human recombinant CB1 receptor(Bmax=2.5pmol/mg protein) and human recombinant CB2 receptor (B max=4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Cairo University

LigandChemical structure of BindingDB Monomer ID 239146BDBM239146((E)-Ethyl 2-(6-(3,4-dimethoxyphenyl)-4-oxohex-5-en...)
Affinity DataKi: >1.00E+4nM IC50: 1.00E+4nMAssay Description:Membranes from HEK-293 cells transfected with the human recombinant CB1 receptor(Bmax=2.5pmol/mg protein) and human recombinant CB2 receptor (B max=4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Cairo University

LigandChemical structure of BindingDB Monomer ID 239147BDBM239147((E)-6-(3,4-Dimethoxyphenyl)-N-(2-hydroxybutan-2-yl...)
Affinity DataKi: >1.00E+4nM IC50: 1.00E+4nMAssay Description:Membranes from HEK-293 cells transfected with the human recombinant CB1 receptor(Bmax=2.5pmol/mg protein) and human recombinant CB2 receptor (B max=4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Cairo University

LigandChemical structure of BindingDB Monomer ID 239144BDBM239144((E)-N-(4-Hydroxyphenyl)-4-oxo-6-p-tolylhex-5-enami...)
Affinity DataKi: >1.00E+4nM IC50: 1.00E+4nMAssay Description:Membranes from HEK-293 cells transfected with the human recombinant CB1 receptor(Bmax=2.5pmol/mg protein) and human recombinant CB2 receptor (B max=4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Cairo University

LigandChemical structure of BindingDB Monomer ID 239145BDBM239145((E)-6-[4-(Dimethylamino)phenyl]-N-(2-hydroxybutan-...)
Affinity DataKi: >1.00E+4nM IC50: 1.00E+4nMAssay Description:Membranes from HEK-293 cells transfected with the human recombinant CB1 receptor(Bmax=2.5pmol/mg protein) and human recombinant CB2 receptor (B max=4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Cairo University

LigandChemical structure of BindingDB Monomer ID 239142BDBM239142((E)-N-(2-Hydroxybutan-2-yl)-4-oxo-6-p-tolylhex-5-e...)
Affinity DataKi: >1.00E+4nM IC50: 1.00E+4nMAssay Description:Membranes from HEK-293 cells transfected with the human recombinant CB1 receptor(Bmax=2.5pmol/mg protein) and human recombinant CB2 receptor (B max=4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Cairo University

LigandChemical structure of BindingDB Monomer ID 239143BDBM239143((E)-N-(1,3-Dihydroxy-2-(hydroxymethylpropan-2-yl)-...)
Affinity DataKi: >1.00E+4nM IC50: 1.00E+4nMAssay Description:Membranes from HEK-293 cells transfected with the human recombinant CB1 receptor(Bmax=2.5pmol/mg protein) and human recombinant CB2 receptor (B max=4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Cairo University

LigandChemical structure of BindingDB Monomer ID 239140BDBM239140((E)-N-(1,3-Dihydroxy-2-(hydroxymethyl)propan-2-yl)...)
Affinity DataKi: >1.00E+4nM IC50: 1.00E+4nMAssay Description:Membranes from HEK-293 cells transfected with the human recombinant CB1 receptor(Bmax=2.5pmol/mg protein) and human recombinant CB2 receptor (B max=4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Cairo University

LigandChemical structure of BindingDB Monomer ID 239141BDBM239141((E) Ethyl [2-(4-oxo-6-phenylhex)-5-enamido]acetate...)
Affinity DataKi: >1.00E+4nM IC50: 1.00E+4nMAssay Description:Membranes from HEK-293 cells transfected with the human recombinant CB1 receptor(Bmax=2.5pmol/mg protein) and human recombinant CB2 receptor (B max=4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Cairo University

LigandChemical structure of BindingDB Monomer ID 239154BDBM239154(4-Acetamidophenyl 4-(naphthalen-1-ylamino)-4-oxobu...)
Affinity DataKi: >1.00E+4nM IC50: 1.00E+4nMAssay Description:Membranes from HEK-293 cells transfected with the human recombinant CB1 receptor(Bmax=2.5pmol/mg protein) and human recombinant CB2 receptor (B max=4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Cairo University

LigandChemical structure of BindingDB Monomer ID 239139BDBM239139((E)-N-(2-Hydroxybutan-2-yl)-4-oxo-6-phenylhex-5-en...)
Affinity DataKi: >1.00E+4nM IC50: 1.00E+4nMAssay Description:Membranes from HEK-293 cells transfected with the human recombinant CB1 receptor(Bmax=2.5pmol/mg protein) and human recombinant CB2 receptor (B max=4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Cairo University

LigandChemical structure of BindingDB Monomer ID 239152BDBM239152(N-(2-Hydroxybutan-2-yl)-2-(4-naphthalen-1-ylamino)...)
Affinity DataKi: >1.00E+4nM IC50: 1.00E+4nMAssay Description:Membranes from HEK-293 cells transfected with the human recombinant CB1 receptor(Bmax=2.5pmol/mg protein) and human recombinant CB2 receptor (B max=4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Cairo University

LigandChemical structure of BindingDB Monomer ID 239153BDBM239153(Ethyl 2-(4-(naphthalen-1-ylamino)-4-oxobutanamido)...)
Affinity DataKi: >1.00E+4nM IC50: 1.00E+4nMAssay Description:Membranes from HEK-293 cells transfected with the human recombinant CB1 receptor(Bmax=2.5pmol/mg protein) and human recombinant CB2 receptor (B max=4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Cairo University

LigandChemical structure of BindingDB Monomer ID 239150BDBM239150((E)-4-Acetamidophenyl 4-oxo-6-phenylhex-5-enoate (...)
Affinity DataKi: >1.00E+4nM IC50: 1.00E+4nMAssay Description:Membranes from HEK-293 cells transfected with the human recombinant CB1 receptor(Bmax=2.5pmol/mg protein) and human recombinant CB2 receptor (B max=4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Cairo University

LigandChemical structure of BindingDB Monomer ID 239151BDBM239151((E)-6-(Biphenyl-4-yl)-N-(2-hydroxybutan-2-yl)-4-ox...)
Affinity DataKi: >1.00E+4nM IC50: 1.00E+4nMAssay Description:Membranes from HEK-293 cells transfected with the human recombinant CB1 receptor(Bmax=2.5pmol/mg protein) and human recombinant CB2 receptor (B max=4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Cairo University

LigandChemical structure of BindingDB Monomer ID 239148BDBM239148((E)-6-(4-(Benzyloxy)phenyl)-N-(2-hydroxybutan-2-yl...)
Affinity DataKi: >1.00E+4nM IC50: 1.00E+4nMAssay Description:Membranes from HEK-293 cells transfected with the human recombinant CB1 receptor(Bmax=2.5pmol/mg protein) and human recombinant CB2 receptor (B max=4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Cairo University

LigandChemical structure of BindingDB Monomer ID 239149BDBM239149((E)-Ethyl 2-(6-(4-(benzyloxy)phenyl)-4-oxohex-5-en...)
Affinity DataKi: >1.00E+4nM IC50: 1.00E+4nMAssay Description:Membranes from HEK-293 cells transfected with the human recombinant CB1 receptor(Bmax=2.5pmol/mg protein) and human recombinant CB2 receptor (B max=4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2017
Entry Details Article
PubMed