Compile Data Set for Download or QSAR
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Report error Found 90 Enz. Inhib. hit(s) with all data for entry = 5649
TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92441(RXP470, 1 | RXP470, Compound 4)
Affinity DataKi:  0.200nM ΔG°:  -55.4kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92443(MMP Inhibitor, 3 | Thiophene derivative, compound ...)
Affinity DataKi:  1.90nM ΔG°:  -49.8kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92446(Inhibitor, 16)
Affinity DataKi:  2.5nM ΔG°:  -49.1kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92449(Inhibitor, 19)
Affinity DataKi:  2.90nM ΔG°:  -48.7kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92447(Inhibitor, 17)
Affinity DataKi:  3.30nM ΔG°:  -48.4kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92448(Inhibitor, 18)
Affinity DataKi:  3.30nM ΔG°:  -48.4kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92445(Inhibitor, 10 | US8691753, 105)
Affinity DataKi:  3.60nM ΔG°:  -48.2kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeutrophil collagenase(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92447(Inhibitor, 17)
Affinity DataKi:  5.30nM ΔG°:  -47.2kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetStromelysin-2(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92441(RXP470, 1 | RXP470, Compound 4)
Affinity DataKi:  8nM ΔG°:  -46.2kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCollagenase 3(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92448(Inhibitor, 18)
Affinity DataKi:  18nM ΔG°:  -44.2kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetStromelysin-1(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92441(RXP470, 1 | RXP470, Compound 4)
Affinity DataKi:  40nM ΔG°:  -42.2kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target72 kDa type IV collagenase(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92448(Inhibitor, 18)
Affinity DataKi:  47nM ΔG°:  -41.8kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCollagenase 3(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92441(RXP470, 1 | RXP470, Compound 4)
Affinity DataKi:  49nM ΔG°:  -41.7kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetStromelysin-2(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92448(Inhibitor, 18)
Affinity DataKi:  54nM ΔG°:  -41.5kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target72 kDa type IV collagenase(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92447(Inhibitor, 17)
Affinity DataKi:  57nM ΔG°:  -41.3kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMatrix metalloproteinase-9(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92447(Inhibitor, 17)
Affinity DataKi:  91nM ΔG°:  -40.2kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetA disintegrin and metalloproteinase with thrombospondin motifs 4(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92449(Inhibitor, 19)
Affinity DataKi:  92nM ΔG°:  -40.2kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMatrix metalloproteinase-14(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92441(RXP470, 1 | RXP470, Compound 4)
Affinity DataKi: >100nM ΔG°: >-40.0kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target72 kDa type IV collagenase(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92441(RXP470, 1 | RXP470, Compound 4)
Affinity DataKi: >100nM ΔG°: >-40.0kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeutrophil collagenase(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92441(RXP470, 1 | RXP470, Compound 4)
Affinity DataKi: >100nM ΔG°: >-40.0kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMatrix metalloproteinase-9(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92441(RXP470, 1 | RXP470, Compound 4)
Affinity DataKi: >100nM ΔG°: >-40.0kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetStromelysin-1(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92448(Inhibitor, 18)
Affinity DataKi:  103nM ΔG°:  -39.9kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetA disintegrin and metalloproteinase with thrombospondin motifs 4(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92445(Inhibitor, 10 | US8691753, 105)
Affinity DataKi:  113nM ΔG°:  -39.7kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target72 kDa type IV collagenase(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92446(Inhibitor, 16)
Affinity DataKi:  127nM ΔG°:  -39.4kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeutrophil collagenase(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92445(Inhibitor, 10 | US8691753, 105)
Affinity DataKi:  203nM ΔG°:  -38.2kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeutrophil collagenase(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92448(Inhibitor, 18)
Affinity DataKi:  205nM ΔG°:  -38.2kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetStromelysin-2(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92446(Inhibitor, 16)
Affinity DataKi:  299nM ΔG°:  -37.2kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetStromelysin-1(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92449(Inhibitor, 19)
Affinity DataKi:  329nM ΔG°:  -37.0kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCollagenase 3(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92447(Inhibitor, 17)
Affinity DataKi:  338nM ΔG°:  -36.9kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeutrophil collagenase(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92449(Inhibitor, 19)
Affinity DataKi:  338nM ΔG°:  -36.9kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetStromelysin-2(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92449(Inhibitor, 19)
Affinity DataKi:  352nM ΔG°:  -36.8kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target72 kDa type IV collagenase(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92445(Inhibitor, 10 | US8691753, 105)
Affinity DataKi:  377nM ΔG°:  -36.7kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetStromelysin-2(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92447(Inhibitor, 17)
Affinity DataKi:  390nM ΔG°:  -36.6kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetA disintegrin and metalloproteinase with thrombospondin motifs 4(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92448(Inhibitor, 18)
Affinity DataKi:  406nM ΔG°:  -36.5kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeutrophil collagenase(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92443(MMP Inhibitor, 3 | Thiophene derivative, compound ...)
Affinity DataKi:  410nM ΔG°:  -36.5kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCollagenase 3(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92449(Inhibitor, 19)
Affinity DataKi:  468nM ΔG°:  -36.1kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCollagenase 3(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92446(Inhibitor, 16)
Affinity DataKi:  501nM ΔG°:  -36.0kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target72 kDa type IV collagenase(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92449(Inhibitor, 19)
Affinity DataKi:  583nM ΔG°:  -35.6kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetA disintegrin and metalloproteinase with thrombospondin motifs 5(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92449(Inhibitor, 19)
Affinity DataKi:  585nM ΔG°:  -37.0kJ/molepH: 6.8 T: 37°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCollagenase 3(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92445(Inhibitor, 10 | US8691753, 105)
Affinity DataKi:  603nM ΔG°:  -35.5kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeutrophil collagenase(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92446(Inhibitor, 16)
Affinity DataKi:  671nM ΔG°:  -35.2kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCollagenase 3(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92443(MMP Inhibitor, 3 | Thiophene derivative, compound ...)
Affinity DataKi:  684nM ΔG°:  -35.2kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetStromelysin-2(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92443(MMP Inhibitor, 3 | Thiophene derivative, compound ...)
Affinity DataKi:  872nM ΔG°:  -34.6kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetA disintegrin and metalloproteinase with thrombospondin motifs 5(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92446(Inhibitor, 16)
Affinity DataKi:  874nM ΔG°:  -36.0kJ/molepH: 6.8 T: 37°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMatrix metalloproteinase-14(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92446(Inhibitor, 16)
Affinity DataKi:  968nM ΔG°:  -34.3kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMatrix metalloproteinase-14(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92443(MMP Inhibitor, 3 | Thiophene derivative, compound ...)
Affinity DataKi: >1.00E+3nM ΔG°: >-34.2kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMatrilysin(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92443(MMP Inhibitor, 3 | Thiophene derivative, compound ...)
Affinity DataKi: >1.00E+3nM ΔG°: >-34.2kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetStromelysin-1(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92443(MMP Inhibitor, 3 | Thiophene derivative, compound ...)
Affinity DataKi: >1.00E+3nM ΔG°: >-34.2kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target72 kDa type IV collagenase(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92443(MMP Inhibitor, 3 | Thiophene derivative, compound ...)
Affinity DataKi: >1.00E+3nM ΔG°: >-34.2kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetInterstitial collagenase(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92441(RXP470, 1 | RXP470, Compound 4)
Affinity DataKi: >1.00E+3nM ΔG°: >-34.2kJ/molepH: 6.8 T: 25°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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