Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50040737
TargetMonoglyceride lipase(Human)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50399285(CHEMBL2180820 | US9102622, 14.3)
Affinity DataIC50: 56.1nMAssay Description:Inhibition of recombinant human hexahistidine-tagged MGL expressed in Escherichia coli using AHMMCE as substrate after 15 mins by medium throughput f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM60536(BDBM50399283 | US9102622, 13.2)
Affinity DataKi:  99nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50399279(CHEMBL2180822)
Affinity DataKi:  104nMAssay Description:Displacement of [3H]CP-55,940 from CB1 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50399287(CHEMBL2180557)
Affinity DataIC50: 116nMAssay Description:Inhibition of recombinant human hexahistidine-tagged MGL expressed in Escherichia coli using AHMMCE as substrate after 15 mins by medium throughput f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50399282(CHEMBL2180817 | US9102622, 13.4)
Affinity DataKi:  118nMAssay Description:Displacement of [3H]CP-55,940 from CB1 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50399279(CHEMBL2180822)
Affinity DataIC50: 156nMAssay Description:Inhibition of recombinant human hexahistidine-tagged MGL expressed in Escherichia coli using AHMMCE as substrate after 15 mins by medium throughput f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50399281(CHEMBL2180818 | US9102622, 14.1)
Affinity DataKi:  163nMAssay Description:Displacement of [3H]CP-55,940 from CB1 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50399286(CHEMBL2180819 | US9102622, 14.2)
Affinity DataIC50: 190nMAssay Description:Inhibition of recombinant human hexahistidine-tagged MGL expressed in Escherichia coli using AHMMCE as substrate after 15 mins by medium throughput f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50399280(CHEMBL2180821 | US9102622, 14.4)
Affinity DataKi:  192nMAssay Description:Displacement of [3H]CP-55,940 from CB1 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50399282(CHEMBL2180817 | US9102622, 13.4)
Affinity DataKi:  194nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50399282(CHEMBL2180817 | US9102622, 13.4)
Affinity DataIC50: 201nMAssay Description:Inhibition of recombinant human hexahistidine-tagged MGL expressed in Escherichia coli using AHMMCE as substrate after 15 mins by medium throughput f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50399279(CHEMBL2180822)
Affinity DataKi:  203nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50399288(CHEMBL2180830 | US9102622, 13.1)
Affinity DataIC50: 249nMAssay Description:Inhibition of recombinant human hexahistidine-tagged MGL expressed in Escherichia coli using AHMMCE as substrate after 15 mins by medium throughput f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM60536(BDBM50399283 | US9102622, 13.2)
Affinity DataKi:  335nMAssay Description:Displacement of [3H]CP-55,940 from CB1 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50399280(CHEMBL2180821 | US9102622, 14.4)
Affinity DataIC50: 383nMAssay Description:Inhibition of recombinant human hexahistidine-tagged MGL expressed in Escherichia coli using AHMMCE as substrate after 15 mins by medium throughput f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50399281(CHEMBL2180818 | US9102622, 14.1)
Affinity DataIC50: 427nMAssay Description:Inhibition of recombinant human hexahistidine-tagged MGL expressed in Escherichia coli using AHMMCE as substrate after 15 mins by medium throughput f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50399280(CHEMBL2180821 | US9102622, 14.4)
Affinity DataKi:  577nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50399281(CHEMBL2180818 | US9102622, 14.1)
Affinity DataKi:  698nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM60536(BDBM50399283 | US9102622, 13.2)
Affinity DataIC50: 752nMAssay Description:Inhibition of recombinant human hexahistidine-tagged MGL expressed in Escherichia coli using AHMMCE as substrate after 15 mins by medium throughput f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50399284(CHEMBL2180823)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant human hexahistidine-tagged MGL expressed in Escherichia coli using AHMMCE as substrate after 15 mins by medium throughput f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed