Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50043036
TargetHistamine H1 receptor(Guinea pig)
Huazhong University of Science and Technology
Curated by ChEMBL
Huazhong University of Science and Technology
Curated by ChEMBL
Affinity DataKi: 3.80nMAssay Description:Displacement of [3H]mepyramine from histamine H1 receptor in guinea pig cerebellum after 60 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding affinity to dopamine D2 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Binding affinity to dopamine D2 receptor (unknown origin)More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Guinea pig)
Huazhong University of Science and Technology
Curated by ChEMBL
Huazhong University of Science and Technology
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Displacement of [3H]mepyramine from histamine H1 receptor in guinea pig cerebellum after 60 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Guinea pig)
Huazhong University of Science and Technology
Curated by ChEMBL
Huazhong University of Science and Technology
Curated by ChEMBL
Affinity DataKi: 21nMAssay Description:Displacement of [3H]mepyramine from histamine H1 receptor in guinea pig cerebellum after 60 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Guinea pig)
Huazhong University of Science and Technology
Curated by ChEMBL
Huazhong University of Science and Technology
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Displacement of [3H]mepyramine from histamine H1 receptor in guinea pig cerebellum after 60 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Guinea pig)
Huazhong University of Science and Technology
Curated by ChEMBL
Huazhong University of Science and Technology
Curated by ChEMBL
Affinity DataKi: 38nMAssay Description:Displacement of [3H]mepyramine from histamine H1 receptor in guinea pig cerebellum after 60 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Guinea pig)
Huazhong University of Science and Technology
Curated by ChEMBL
Huazhong University of Science and Technology
Curated by ChEMBL
Affinity DataKi: 550nMAssay Description:Displacement of [3H]mepyramine from histamine H1 receptor in guinea pig cerebellum after 60 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Guinea pig)
Huazhong University of Science and Technology
Curated by ChEMBL
Huazhong University of Science and Technology
Curated by ChEMBL
Affinity DataKi: 1.13E+3nMAssay Description:Displacement of [3H]mepyramine from histamine H1 receptor in guinea pig cerebellum after 60 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Guinea pig)
Huazhong University of Science and Technology
Curated by ChEMBL
Huazhong University of Science and Technology
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]mepyramine from histamine H1 receptor in guinea pig cerebellum after 60 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMT: 25°CAssay Description:Antagonist activity at dopamine D2 receptor (unknown origin) expressed in CHOK1 cells coexpressing Galpha15 assessed as inhibition of agonist-induced...More data for this Ligand-Target Pair
Affinity DataIC50: 26nMT: 25°CAssay Description:Antagonist activity at dopamine D2 receptor (unknown origin) expressed in CHOK1 cells coexpressing Galpha15 assessed as inhibition of agonist-induced...More data for this Ligand-Target Pair
Affinity DataEC50: 6.70nMAssay Description:Agonist activity at dopamine D2 receptor (unknown origin) expressed in CHOK1 cells coexpressing Galpha15 by FLIPR assayMore data for this Ligand-Target Pair
3D Structure (crystal)