Compile Data Set for Download or QSAR
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Found 25 Enz. Inhib. hit(s) with all data for entry = 50040828
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400772(CHEMBL2204985)
Affinity DataKi:  9.30nMAssay Description:Binding affinity to human GPR119More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400773(CHEMBL2204984)
Affinity DataKi:  15nMAssay Description:Binding affinity to human GPR119More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400774(CHEMBL2204983)
Affinity DataKi:  30nMAssay Description:Binding affinity to human GPR119More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400776(CHEMBL2204986)
Affinity DataKi:  37nMAssay Description:Binding affinity to human GPR119More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400775(CHEMBL2204982)
Affinity DataKi:  99nMAssay Description:Binding affinity to human GPR119More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400776(CHEMBL2204986)
Affinity DataEC50:  19nMAssay Description:Agonist activity at GPR119 in human HEK293 cells assessed as cAMP level by beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400764(CHEMBL2204981)
Affinity DataEC50:  28nMAssay Description:Agonist activity at GPR119 expressed in CHO-K1 cells assessed as cAMP level after 1 hr by homogenous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400765(CHEMBL2203304)
Affinity DataEC50:  27nMAssay Description:Agonist activity at GPR119 expressed in CHO-K1 cells assessed as cAMP level after 1 hr by homogenous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400766(CHEMBL2204980)
Affinity DataEC50:  23nMAssay Description:Agonist activity at GPR119 expressed in CHO-K1 cells assessed as cAMP level after 1 hr by homogenous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400767(CHEMBL2204979)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human GPR119 expressed in MIN6 cells assessed as intracellular cAMP concentration after 45 mins by Alphascreen analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400768(CHEMBL2204978)
Affinity DataEC50:  3nMAssay Description:Agonist activity at human GPR119 expressed in MIN6 cells assessed as intracellular cAMP concentration after 45 mins by Alphascreen analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400769(CHEMBL2204977)
Affinity DataEC50:  3nMAssay Description:Agonist activity at human GPR119 expressed in MIN6 cells assessed as intracellular cAMP concentration after 45 mins by Alphascreen analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400770(CHEMBL2204976)
Affinity DataEC50:  228nMAssay Description:Agonist activity at human GPR119 expressed in MIN6 cells assessed as intracellular cAMP concentration after 45 mins by Alphascreen analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400771(CHEMBL2204975)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human GPR119 expressed in MIN6 cells assessed as intracellular cAMP concentration after 45 mins by Alphascreen analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400772(CHEMBL2204985)
Affinity DataEC50:  2.80nMAssay Description:Agonist activity at GPR119 in human HEK293 cells assessed as cAMP level by beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400773(CHEMBL2204984)
Affinity DataEC50:  11nMAssay Description:Agonist activity at GPR119 in human HEK293 cells assessed as cAMP level by beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400774(CHEMBL2204983)
Affinity DataEC50:  22nMAssay Description:Agonist activity at GPR119 in human HEK293 cells assessed as cAMP level by beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400775(CHEMBL2204982)
Affinity DataEC50:  44nMAssay Description:Agonist activity at GPR119 in human HEK293 cells assessed as cAMP level by beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400777(CHEMBL2204974)
Affinity DataEC50:  1.00E+8nMAssay Description:Agonist activity at GPR119 expressed in CHO-K1 cells assessed as cAMP level after 1 hr by homogenous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400776(CHEMBL2204986)
Affinity DataEC50:  30nMAssay Description:Agonist activity at GPR119 in human U20S cells assessed as binding to beta-arrestin by chemilumiscence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400773(CHEMBL2204984)
Affinity DataEC50:  5.30nMAssay Description:Agonist activity at GPR119 in human U20S cells assessed as binding to beta-arrestin by chemilumiscence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400772(CHEMBL2204985)
Affinity DataEC50:  5.40nMAssay Description:Agonist activity at GPR119 in human U20S cells assessed as binding to beta-arrestin by chemilumiscence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400775(CHEMBL2204982)
Affinity DataEC50:  63nMAssay Description:Agonist activity at GPR119 in human U20S cells assessed as binding to beta-arrestin by chemilumiscence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400775(CHEMBL2204982)
Affinity DataEC50:  141nMAssay Description:Agonist activity at GPR119 in human HEK293 cells by beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400774(CHEMBL2204983)
Affinity DataEC50:  15nMAssay Description:Agonist activity at GPR119 in human U20S cells assessed as binding to beta-arrestin by chemilumiscence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed