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Report error Found 59 Enz. Inhib. hit(s) with all data for entry = 50040813 Sort by
TargetAminopeptidase N(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50400532(CHEMBL2204959)
Affinity DataIC50: 50nMAssay Description:Inhibition of APN in porcine kidney microsome assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50400529(CHEMBL2204943)
Affinity DataIC50: 99nMAssay Description:Inhibition of APN in porcine kidney microsome assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50400541(CHEMBL2204950)
Affinity DataIC50: 290nMAssay Description:Inhibition of APN in porcine kidney microsome assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50400544(CHEMBL2204947)
Affinity DataIC50: 330nMAssay Description:Inhibition of APN in porcine kidney microsome assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50400538(CHEMBL2204953)
Affinity DataIC50: 410nMAssay Description:Inhibition of APN in porcine kidney microsome assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400532(CHEMBL2204959)
Affinity DataIC50: 420nMAssay Description:Inhibition of APN in human ES2 cell surface assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substrate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400529(CHEMBL2204943)
Affinity DataIC50: 480nMAssay Description:Inhibition of APN in human ES2 cell surface assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substrate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50400546(CHEMBL2204945)
Affinity DataIC50: 570nMAssay Description:Inhibition of APN in porcine kidney microsome assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50400542(CHEMBL2204949)
Affinity DataIC50: 570nMAssay Description:Inhibition of APN in porcine kidney microsome assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50400543(CHEMBL2204948)
Affinity DataIC50: 660nMAssay Description:Inhibition of APN in porcine kidney microsome assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50400540(CHEMBL2204951)
Affinity DataIC50: 690nMAssay Description:Inhibition of APN in porcine kidney microsome assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50400537(CHEMBL2204954)
Affinity DataIC50: 730nMAssay Description:Inhibition of APN in porcine kidney microsome assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400541(CHEMBL2204950)
Affinity DataIC50: 790nMAssay Description:Inhibition of APN in human ES2 cell surface assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substrate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50400539(CHEMBL2204952)
Affinity DataIC50: 830nMAssay Description:Inhibition of APN in porcine kidney microsome assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400537(CHEMBL2204954)
Affinity DataIC50: 910nMAssay Description:Inhibition of APN in human ES2 cell surface assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substrate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400544(CHEMBL2204947)
Affinity DataIC50: 940nMAssay Description:Inhibition of APN in human ES2 cell surface assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substrate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50400551(CHEMBL2205650)
Affinity DataIC50: 980nMAssay Description:Inhibition of APN in porcine kidney microsome assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50400535(CHEMBL2204956)
Affinity DataIC50: 1.03E+3nMAssay Description:Inhibition of APN in porcine kidney microsome assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400542(CHEMBL2204949)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of APN in human ES2 cell surface assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substrate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400538(CHEMBL2204953)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of APN in human ES2 cell surface assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substrate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50400536(CHEMBL2204955)
Affinity DataIC50: 1.64E+3nMAssay Description:Inhibition of APN in porcine kidney microsome assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50400532(CHEMBL2204959)
Affinity DataIC50: 1.82E+3nMAssay Description:Inhibition of mouse APNMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50400550(CHEMBL2205651)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of APN in porcine kidney microsome assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50400547(CHEMBL2204944)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of APN in porcine kidney microsome assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50400556(CHEMBL2204965)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of APN in porcine kidney microsome assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50400529(CHEMBL2204943)
Affinity DataIC50: 2.26E+3nMAssay Description:Inhibition of mouse APNMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50400548(CHEMBL2205653)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of APN in porcine kidney microsome assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50400555(CHEMBL2204966)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of APN in porcine kidney microsome assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50400545(CHEMBL2204946)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of APN in porcine kidney microsome assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50400549(CHEMBL2205652)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of APN in porcine kidney microsome assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50400553(CHEMBL2205648)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of APN in porcine kidney microsome assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400540(CHEMBL2204951)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of APN in human ES2 cell surface assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substrate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50400559(CHEMBL2204962)
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of APN in porcine kidney microsome assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50400558(CHEMBL2204963)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of APN in porcine kidney microsome assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50400552(CHEMBL2205649)
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of APN in porcine kidney microsome assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50400541(CHEMBL2204950)
Affinity DataIC50: 5.61E+3nMAssay Description:Inhibition of mouse APNMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50400533(CHEMBL2204958)
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of APN in porcine kidney microsome assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400546(CHEMBL2204945)
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibition of APN in human ES2 cell surface assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substrate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400539(CHEMBL2204952)
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of APN in human ES2 cell surface assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substrate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50400557(CHEMBL2204964)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of APN in porcine kidney microsome assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM23971(CHEMBL29292 | (2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-...)
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of APN in porcine kidney microsome assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50400534(CHEMBL2204957)
Affinity DataIC50: 9.90E+3nMAssay Description:Inhibition of APN in porcine kidney microsome assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50400554(CHEMBL2205647)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of APN in porcine kidney microsome assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50400531(CHEMBL2204960)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of APN in porcine kidney microsome assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50400530(CHEMBL2204961)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of APN in porcine kidney microsome assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM23971(CHEMBL29292 | (2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of APN in human ES2 cell surface assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substrate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM23971(CHEMBL29292 | (2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-...)
Affinity DataIC50: 2.32E+4nMAssay Description:Inhibition of mouse APNMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target72 kDa type IV collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM23971(CHEMBL29292 | (2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-...)
Affinity DataIC50: 2.76E+5nMAssay Description:Inhibition of recombinant MMP-2 using succinylated gelatin as substrate incubated for 10 mins before addition of substrate measured after 60 mins by ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target72 kDa type IV collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400532(CHEMBL2204959)
Affinity DataIC50: 5.45E+5nMAssay Description:Inhibition of recombinant MMP-2 using succinylated gelatin as substrate incubated for 10 mins before addition of substrate measured after 60 mins by ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target72 kDa type IV collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400544(CHEMBL2204947)
Affinity DataIC50: 5.73E+5nMAssay Description:Inhibition of recombinant MMP-2 using succinylated gelatin as substrate incubated for 10 mins before addition of substrate measured after 60 mins by ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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