Compile Data Set for Download or QSAR
Report error Found 89 Enz. Inhib. hit(s) with all data for entry = 50035801
Target5-hydroxytryptamine receptor 1A(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016966BDBM50016966(CHEMBL543967 | 1,1-Dioxo-2-[4-(4-thieno[3,2-c]pyri...)
Affinity DataIC50: 0.680nMAssay Description:Ability to bind at serotonin 5-hydroxytryptamine 1A receptors of rat hippocampus by displacing [3H]8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016963BDBM50016963(CHEMBL554473 | 2-[4-(4-Thieno[3,2-c]pyridin-4-yl-p...)
Affinity DataIC50: 0.690nMAssay Description:Ability to bind at alpha-1 adrenergic receptor by displacing [3H]WB-4101More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016955BDBM50016955(CHEMBL278876 | 4-[4-(4-Thieno[3,2-c]pyridin-4-yl-p...)
Affinity DataIC50: 1.10nMAssay Description:Ability to bind at alpha-1 adrenergic receptor by displacing [3H]WB-4101More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016966BDBM50016966(CHEMBL543967 | 1,1-Dioxo-2-[4-(4-thieno[3,2-c]pyri...)
Affinity DataIC50: 1.20nMAssay Description:Ability to bind at alpha-1 adrenergic receptor by displacing [3H]WB-4101More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016955BDBM50016955(CHEMBL278876 | 4-[4-(4-Thieno[3,2-c]pyridin-4-yl-p...)
Affinity DataIC50: 1.20nMAssay Description:Ability to bind at serotonin 5-hydroxytryptamine 1A receptors of rat hippocampus by displacing [3H]8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016959BDBM50016959(CHEMBL537924 | 4-Methyl-1-[4-(4-thieno[3,2-c]pyrid...)
Affinity DataIC50: 1.30nMAssay Description:Ability to bind at serotonin 5-hydroxytryptamine 1A receptors of rat hippocampus by displacing [3H]8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016971BDBM50016971(CHEMBL536797 | 3-{4-[4-(2-Methyl-furo[3,2-c]pyridi...)
Affinity DataIC50: 2.20nMAssay Description:Ability to bind at 5-hydroxytryptamine 1A receptor of rat hippocampus by displacing [3H]8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A/1B/1D/1F(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016966BDBM50016966(CHEMBL543967 | 1,1-Dioxo-2-[4-(4-thieno[3,2-c]pyri...)
Affinity DataIC50: 2.30nMAssay Description:Ability to bind at 5-hydroxytryptamine 1 receptor of rat hippocampus by displacing [3H]5-HTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016969BDBM50016969(CHEMBL543018 | 1-[4-(4-Thieno[3,2-c]pyridin-4-yl-p...)
Affinity DataIC50: 2.5nMAssay Description:Ability to bind at serotonin 5-hydroxytryptamine 1A receptors of rat hippocampus by displacing [3H]8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016963BDBM50016963(CHEMBL554473 | 2-[4-(4-Thieno[3,2-c]pyridin-4-yl-p...)
Affinity DataIC50: 2.70nMAssay Description:Ability to bind at serotonin 5-hydroxytryptamine 1A receptors of rat hippocampus by displacing [3H]8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016963BDBM50016963(CHEMBL554473 | 2-[4-(4-Thieno[3,2-c]pyridin-4-yl-p...)
Affinity DataIC50: 2.80nMAssay Description:Ability to bind at serotonin 5-hydroxytryptamine 2 receptors of rat hippocampus by displacing [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016960BDBM50016960(CHEMBL537702 | 4,4-Dimethyl-1-[4-(4-thieno[3,2-c]p...)
Affinity DataIC50: 3nMAssay Description:Ability to bind at serotonin 5-hydroxytryptamine 2 receptors of rat hippocampus by displacing [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A/1B/1D/1F(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016967BDBM50016967(CHEMBL544203 | 3-{4-[4-(2-Methyl-thieno[3,2-c]pyri...)
Affinity DataIC50: 3.60nMAssay Description:Ability to bind at 5-hydroxytryptamine 1 receptor of rat hippocampus by displacing [3H]5-HTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A/1B/1D/1F(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016956BDBM50016956(CHEMBL552616 | 1-{4-[4-(2-Bromo-thieno[3,2-c]pyrid...)
Affinity DataIC50: 3.70nMAssay Description:Ability to bind at 5-hydroxytryptamine 1 receptor of rat hippocampus by displacing [3H]5-HTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A/1B/1D/1F(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016957BDBM50016957(CHEMBL558026 | 3-[4-(4-Thieno[2,3-c]pyridin-7-yl-p...)
Affinity DataIC50: 3.70nMAssay Description:Ability to bind at 5-hydroxytryptamine 1 receptor of rat hippocampus by displacing [3H]5-HTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A/1B/1D/1F(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016958BDBM50016958(CHEMBL15560 | 1-(4-Fluoro-phenyl)-4-(4-thieno[3,2-...)
Affinity DataIC50: 3.80nMAssay Description:Ability to bind at 5-hydroxytryptamine 1 receptor of rat hippocampus by displacing [3H]5-HTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016964BDBM50016964(CHEMBL537707 | 3-[4-(4-Thieno[3,2-c]pyridin-4-yl-p...)
Affinity DataIC50: 3.90nMAssay Description:Ability to bind at 5-hydroxytryptamine 2 receptor of rat hippocampus by displacing [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016959BDBM50016959(CHEMBL537924 | 4-Methyl-1-[4-(4-thieno[3,2-c]pyrid...)
Affinity DataIC50: 4.20nMAssay Description:Ability to bind at serotonin 5-hydroxytryptamine 2 receptors of rat hippocampus by displacing [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016965BDBM50016965(CHEMBL544202 | 4,4-Dimethyl-1-{4-[4-(2-methyl-furo...)
Affinity DataIC50: 4.90nMAssay Description:Ability to bind at serotonin 5-hydroxytryptamine 1A receptors of rat hippocampus by displacing [3H]8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A/1B/1D/1F(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016963BDBM50016963(CHEMBL554473 | 2-[4-(4-Thieno[3,2-c]pyridin-4-yl-p...)
Affinity DataIC50: 5.30nMAssay Description:Ability to bind at 5-hydroxytryptamine 1 receptor of rat hippocampus by displacing [3H]5-HTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A/1B/1D/1F(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016960BDBM50016960(CHEMBL537702 | 4,4-Dimethyl-1-[4-(4-thieno[3,2-c]p...)
Affinity DataIC50: 5.70nMAssay Description:Ability to bind at 5-hydroxytryptamine 1 receptor of rat hippocampus by displacing [3H]5-HTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016966BDBM50016966(CHEMBL543967 | 1,1-Dioxo-2-[4-(4-thieno[3,2-c]pyri...)
Affinity DataIC50: 5.70nMAssay Description:Ability to bind at serotonin 5-hydroxytryptamine 2 receptors of rat hippocampus by displacing [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016958BDBM50016958(CHEMBL15560 | 1-(4-Fluoro-phenyl)-4-(4-thieno[3,2-...)
Affinity DataIC50: 5.80nMAssay Description:Ability to bind at serotonin 5-hydroxytryptamine 2 receptors of rat hippocampus by displacing [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016968BDBM50016968(CHEMBL557995 | 1-(4-Fluoro-phenyl)-4-[4-(2-methyl-...)
Affinity DataIC50: 6.20nMAssay Description:Ability to bind at serotonin 5-hydroxytryptamine 1A receptors of rat hippocampus by displacing [3H]8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016955BDBM50016955(CHEMBL278876 | 4-[4-(4-Thieno[3,2-c]pyridin-4-yl-p...)
Affinity DataIC50: 6.70nMAssay Description:Ability to bind at serotonin 5-hydroxytryptamine 2 receptors of rat hippocampus by displacing [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A/1B/1D/1F(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016964BDBM50016964(CHEMBL537707 | 3-[4-(4-Thieno[3,2-c]pyridin-4-yl-p...)
Affinity DataIC50: 8.10nMAssay Description:Ability to bind at 5-hydroxytryptamine 1 receptor of rat hippocampus by displacing [3H]5-HTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016975BDBM50016975(CHEMBL554419 | 1-[4-(4-Furo[3,2-c]pyridin-4-yl-pip...)
Affinity DataIC50: 8.60nMAssay Description:Ability to bind at 5-hydroxytryptamine 1A receptor of rat hippocampus by displacing [3H]8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A/1B/1D/1F(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016959BDBM50016959(CHEMBL537924 | 4-Methyl-1-[4-(4-thieno[3,2-c]pyrid...)
Affinity DataIC50: 8.80nMAssay Description:Ability to bind at 5-hydroxytryptamine 1 receptor of rat hippocampus by displacing [3H]5-HTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50001888BDBM50001888([3-(2-Chloro-phenothiazin-10-yl)-propyl]-dimethyl-...)
Affinity DataIC50: 8.80nMAssay Description:Ability to bind at 5-hydroxytryptamine 2 receptor of rat hippocampus by displacing [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016974BDBM50016974(CHEMBL542789 | 1-(4-Fluoro-phenyl)-4-(4-furo[3,2-c...)
Affinity DataIC50: 12nMAssay Description:Ability to bind at serotonin 5-hydroxytryptamine 1A receptors of rat hippocampus by displacing [3H]8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016960BDBM50016960(CHEMBL537702 | 4,4-Dimethyl-1-[4-(4-thieno[3,2-c]p...)
Affinity DataIC50: 19nMAssay Description:Ability to bind at alpha-1 adrenergic receptor by displacing [3H]WB-4101More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016969BDBM50016969(CHEMBL543018 | 1-[4-(4-Thieno[3,2-c]pyridin-4-yl-p...)
Affinity DataIC50: 19nMAssay Description:Ability to bind at serotonin 5-hydroxytryptamine 2 receptors of rat hippocampus by displacing [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016957BDBM50016957(CHEMBL558026 | 3-[4-(4-Thieno[2,3-c]pyridin-7-yl-p...)
Affinity DataIC50: 20nMAssay Description:Ability to bind at 5-hydroxytryptamine 2 receptor of rat hippocampus by displacing [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50001884BDBM50001884(8-Chloro-11-(4-methyl-piperazin-1-yl)-5H-dibenzo[b...)
Affinity DataIC50: 21nMAssay Description:Ability to bind at 5-hydroxytryptamine 2 receptor of rat hippocampus by displacing [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016958BDBM50016958(CHEMBL15560 | 1-(4-Fluoro-phenyl)-4-(4-thieno[3,2-...)
Affinity DataIC50: 23nMAssay Description:Ability to bind at alpha-1 adrenergic receptor by displacing [3H]WB-4101More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016977BDBM50016977(CHEMBL553758 | 3-[4-(4-Furo[3,2-c]pyridin-4-yl-pip...)
Affinity DataIC50: 24nMAssay Description:Ability to bind at Alpha-1 adrenergic receptor by displacing [3H]WB-4101More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016974BDBM50016974(CHEMBL542789 | 1-(4-Fluoro-phenyl)-4-(4-furo[3,2-c...)
Affinity DataIC50: 24nMAssay Description:Ability to bind at alpha-1 adrenergic receptor by displacing [3H]WB-4101More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A/1B/1D/1F(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016973BDBM50016973(CHEMBL543253 | 3-{4-[4-(2-Bromo-thieno[3,2-c]pyrid...)
Affinity DataIC50: 25nMAssay Description:Ability to bind at 5-hydroxytryptamine 1 receptor of rat hippocampus by displacing [3H]5-HTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016956BDBM50016956(CHEMBL552616 | 1-{4-[4-(2-Bromo-thieno[3,2-c]pyrid...)
Affinity DataIC50: 27nMAssay Description:Ability to bind at alpha-1 adrenergic receptor by displacing [3H]WB-4101More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016971BDBM50016971(CHEMBL536797 | 3-{4-[4-(2-Methyl-furo[3,2-c]pyridi...)
Affinity DataIC50: 28nMAssay Description:Ability to bind at Alpha-1 adrenergic receptor by displacing [3H]WB-4101More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50001888BDBM50001888([3-(2-Chloro-phenothiazin-10-yl)-propyl]-dimethyl-...)
Affinity DataIC50: 31nMAssay Description:Ability to bind at Alpha-1 adrenergic receptor by displacing [3H]WB-4101More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016964BDBM50016964(CHEMBL537707 | 3-[4-(4-Thieno[3,2-c]pyridin-4-yl-p...)
Affinity DataIC50: 31nMAssay Description:Ability to bind at Alpha-1 adrenergic receptor by displacing [3H]WB-4101More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A/1B/1D/1F(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016961BDBM50016961(CHEMBL16072 | 4-[4-(4-Furo[3,2-c]pyridin-4-yl-pipe...)
Affinity DataIC50: 34nMAssay Description:Ability to bind at 5-hydroxytryptamine 1 receptor of rat hippocampus by displacing [3H]5-HTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016957BDBM50016957(CHEMBL558026 | 3-[4-(4-Thieno[2,3-c]pyridin-7-yl-p...)
Affinity DataIC50: 37nMAssay Description:Ability to bind at Alpha-1 adrenergic receptor by displacing [3H]WB-4101More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50001888BDBM50001888([3-(2-Chloro-phenothiazin-10-yl)-propyl]-dimethyl-...)
Affinity DataIC50: 40nMAssay Description:Ability to bind at dopamine receptor D2 of rat corpus striatum by displacing [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016961BDBM50016961(CHEMBL16072 | 4-[4-(4-Furo[3,2-c]pyridin-4-yl-pipe...)
Affinity DataIC50: 41nMAssay Description:Ability to bind at alpha-1 adrenergic receptor by displacing [3H]WB-4101More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016967BDBM50016967(CHEMBL544203 | 3-{4-[4-(2-Methyl-thieno[3,2-c]pyri...)
Affinity DataIC50: 43nMAssay Description:Ability to bind at 5-hydroxytryptamine 2 receptor of rat hippocampus by displacing [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016975BDBM50016975(CHEMBL554419 | 1-[4-(4-Furo[3,2-c]pyridin-4-yl-pip...)
Affinity DataIC50: 47nMAssay Description:Ability to bind at Alpha-1 adrenergic receptor by displacing [3H]WB-4101More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016974BDBM50016974(CHEMBL542789 | 1-(4-Fluoro-phenyl)-4-(4-furo[3,2-c...)
Affinity DataIC50: 55nMAssay Description:Ability to bind at serotonin 5-hydroxytryptamine 2 receptors of rat hippocampus by displacing [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Bristol-Myers

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50016961BDBM50016961(CHEMBL16072 | 4-[4-(4-Furo[3,2-c]pyridin-4-yl-pipe...)
Affinity DataIC50: 55nMAssay Description:Ability to bind at serotonin 5-hydroxytryptamine 2 receptors of rat hippocampus by displacing [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
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