Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50009982
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 23971BDBM23971(CHEMBL29292 | (2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-...)
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 23971BDBM23971(CHEMBL29292 | (2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-...)
Affinity DataIC50: 1.12E+4nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 10 hrs measured every 6 mins by fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534075BDBM50534075(CHEMBL4483393)
Affinity DataIC50: 1.65E+4nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534075BDBM50534075(CHEMBL4483393)
Affinity DataIC50: 3.36E+4nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 10 hrs measured every 6 mins by fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534077BDBM50534077(CHEMBL4464704)
Affinity DataIC50: 6.36E+4nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534070BDBM50534070(CHEMBL4454667)
Affinity DataIC50: 6.83E+4nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534074BDBM50534074(CHEMBL4468968)
Affinity DataIC50: 6.93E+4nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534069BDBM50534069(CHEMBL4473220)
Affinity DataIC50: 7.68E+4nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534072BDBM50534072(CHEMBL4455383)
Affinity DataIC50: 1.11E+5nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534078BDBM50534078(CHEMBL4557950)
Affinity DataIC50: 1.38E+5nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534081BDBM50534081(CHEMBL4460083)
Affinity DataIC50: 1.63E+5nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534071BDBM50534071(CHEMBL4563759)
Affinity DataIC50: 3.79E+5nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534080BDBM50534080(CHEMBL4576374)
Affinity DataIC50: 4.09E+5nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534073BDBM50534073(CHEMBL4537106)
Affinity DataIC50: 7.81E+5nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534076BDBM50534076(CHEMBL4435767)
Affinity DataIC50: 1.05E+6nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534079BDBM50534079(CHEMBL4456116)
Affinity DataIC50: 1.11E+6nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed