Compile Data Set for Download or QSAR
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Found 90 Enz. Inhib. hit(s) with all data for entry = 50000736
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50259839(CHEMBL4100677)
Affinity DataIC50:  8.60nMAssay Description:Agonist activity at TEV protease cleavage site linked GAL4-VP16-fused GPR35 in human Tango GPR35-bla U2OS cells assessed as induction of TEV protease...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50259842(CHEMBL4079816)
Affinity DataIC50:  13nMAssay Description:Agonist activity at GPR35 in human HT-29 cells by DMR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50259853(CHEMBL4092954)
Affinity DataIC50:  23nMAssay Description:Agonist activity at GPR35 in human HT-29 cells by DMR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50259845(CHEMBL4082281)
Affinity DataIC50:  31nMAssay Description:Agonist activity at GPR35 in human HT-29 cells by DMR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50259843(CHEMBL4081238)
Affinity DataIC50:  56nMAssay Description:Agonist activity at GPR35 in human HT-29 cells assessed as induction of cell desensitization to 1 uM zaprinast preincubated for 1 hr followed by zapr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50259841(CHEMBL4085211)
Affinity DataIC50:  330nMAssay Description:Agonist activity at GPR35 in human HT-29 cells assessed as induction of cell desensitization to 1 uM zaprinast preincubated for 1 hr followed by zapr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50259852(CHEMBL4065291)
Affinity DataIC50:  380nMAssay Description:Agonist activity at GPR35 in human HT-29 cells assessed as induction of cell desensitization to 1 uM zaprinast preincubated for 1 hr followed by zapr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50259854(CHEMBL4103143)
Affinity DataIC50:  460nMAssay Description:Agonist activity at GPR35 in human HT-29 cells assessed as induction of cell desensitization to 1 uM zaprinast preincubated for 1 hr followed by zapr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50259878(CHEMBL4073902)
Affinity DataIC50:  483nMAssay Description:Agonist activity at GPR35 in human HT-29 cells assessed as induction of cell desensitization to 1 uM zaprinast preincubated for 1 hr followed by zapr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50259864(CHEMBL4093683)
Affinity DataIC50:  590nMAssay Description:Agonist activity at GPR35 in human HT-29 cells by DMR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50259865(CHEMBL4066109)
Affinity DataIC50:  650nMAssay Description:Agonist activity at GPR35 in human HT-29 cells assessed as induction of cell desensitization to 1 uM zaprinast preincubated for 1 hr followed by zapr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50259844(CHEMBL4105535)
Affinity DataIC50:  750nMAssay Description:Agonist activity at GPR35 in human HT-29 cells by DMR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50259859(CHEMBL1830823)
Affinity DataIC50:  1.08E+3nMAssay Description:Agonist activity at human GPR35 expressed in CHO-K1 cells after 90 mins by beta-arrestin 2 recruitment assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50259866(CHEMBL4081445)
Affinity DataIC50:  1.69E+3nMAssay Description:Agonist activity at GPR35 in human HT-29 cells assessed as induction of cell desensitization to 1 uM zaprinast preincubated for 1 hr followed by zapr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50259856(CHEMBL1600989)
Affinity DataIC50:  2.30E+3nMAssay Description:Agonist activity at GPR35 in human HT-29 cells assessed as induction of cell desensitization to 1 uM zaprinast preincubated for 1 hr followed by zapr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50259888(CHEMBL4084237)
Affinity DataIC50:  2.82E+3nMAssay Description:Agonist activity at GPR35 in human HT-29 cells assessed as induction of cell desensitization to 1 uM zaprinast preincubated for 1 hr followed by zapr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50259846(CHEMBL4103860)
Affinity DataIC50:  2.89E+3nMAssay Description:Agonist activity at GPR35 in human HT-29 cells assessed as induction of cell desensitization to 1 uM zaprinast preincubated for 1 hr followed by zapr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50259860(CHEMBL4096323)
Affinity DataIC50:  3.75E+3nMAssay Description:Agonist activity at GPR35 in human HT-29 cells by DMR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50259858(CHEMBL4077503)
Affinity DataIC50:  3.76E+3nMAssay Description:Agonist activity at GPR35 in human HT-29 cells assessed as induction of cell desensitization to 1 uM zaprinast preincubated for 1 hr followed by zapr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50259884(CHEMBL1765162)
Affinity DataIC50:  5.08E+3nMAssay Description:Agonist activity at GPR35 in human HT-29 cells assessed as induction of cell desensitization to 1 uM zaprinast preincubated for 1 hr followed by zapr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50259840(CHEMBL4078055)
Affinity DataIC50:  8.61E+3nMAssay Description:Agonist activity at GPR35 in human HT-29 cells assessed as induction of cell desensitization to 1 uM zaprinast preincubated for 1 hr followed by zapr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50259863(CHEMBL4085935)
Affinity DataIC50:  9.33E+3nMAssay Description:Agonist activity at GPR35 in human HT-29 cells assessed as induction of cell desensitization to 1 uM zaprinast preincubated for 1 hr followed by zapr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50259886(CHEMBL2333943)
Affinity DataIC50:  1.13E+4nMAssay Description:Agonist activity at GPR35 in human HT-29 cells assessed as induction of cell desensitization to 1 uM zaprinast preincubated for 1 hr followed by zapr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50259855(CHEMBL1414071)
Affinity DataIC50:  1.32E+4nMAssay Description:Agonist activity at GPR35 in human HT-29 cells assessed as induction of cell desensitization to 1 uM zaprinast preincubated for 1 hr followed by zapr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50259879(CHEMBL4062531)
Affinity DataIC50:  1.41E+4nMAssay Description:Agonist activity at GPR35 in human HT-29 cells assessed as induction of cell desensitization to 1 uM zaprinast preincubated for 1 hr followed by zapr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50259861(CHEMBL4096105)
Affinity DataIC50:  1.49E+4nMAssay Description:Agonist activity at GPR35 in human HT-29 cells assessed as induction of cell desensitization to 1 uM zaprinast preincubated for 1 hr followed by zapr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50259885(CHEMBL4088382)
Affinity DataIC50:  2.14E+4nMAssay Description:Agonist activity at GPR35 in human HT-29 cells assessed as induction of cell desensitization to 1 uM zaprinast preincubated for 1 hr followed by zapr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50131066(2-Oxo-2H-chromene-3-carboxylic acid | CHEMBL83294)
Affinity DataIC50:  1.00E+5nMAssay Description:Agonist activity at GPR35 in human HT-29 cells assessed as induction of cell desensitization to 1 uM zaprinast preincubated for 1 hr followed by zapr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50233945(CHEBI:18344 | Kynurenic Acid | TRANSTORINE)
Affinity DataEC50:  1.52E+5nMAssay Description:Agonist activity at human GPR35 expressed in CHO-K1 cells by DMR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50259843(CHEMBL4081238)
Affinity DataEC50:  150nMAssay Description:Agonist activity at GPR35 in human HT-29 cells by DMR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50259845(CHEMBL4082281)
Affinity DataEC50:  51nMAssay Description:Agonist activity at GPR35 in human HT-29 cells by DMR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50259853(CHEMBL4092954)
Affinity DataEC50:  67nMAssay Description:Agonist activity at GPR35 in human HT-29 cells by DMR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50259854(CHEMBL4103143)
Affinity DataEC50:  1.41E+3nMAssay Description:Agonist activity at GPR35 in human HT-29 cells by DMR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM14363(3-(2-propoxyphenyl)-2,4,7,8,9-pentazabicyclo[4.3.0...)
Affinity DataEC50:  3.52E+3nMAssay Description:Agonist activity at TEV protease cleavage site linked GAL4-VP16-fused GPR35 in human Tango GPR35-bla U2OS cells assessed as induction of TEV protease...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50259839(CHEMBL4100677)
Affinity DataEC50:  197nMAssay Description:Agonist activity at TEV protease cleavage site linked GAL4-VP16-fused GPR35 in human Tango GPR35-bla U2OS cells assessed as induction of TEV protease...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50259846(CHEMBL4103860)
Affinity DataEC50:  2.33E+3nMAssay Description:Agonist activity at GPR35 in human HT-29 cells by DMR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50259840(CHEMBL4078055)
Affinity DataEC50:  8.61E+3nMAssay Description:Agonist activity at GPR35 in human HT-29 cells by DMR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50259885(CHEMBL4088382)
Affinity DataEC50:  2.14E+4nMAssay Description:Agonist activity at GPR35 in human HT-29 cells by DMR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50259844(CHEMBL4105535)
Affinity DataEC50:  887nMAssay Description:Agonist activity at GPR35 in human HT-29 cells by DMR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50259859(CHEMBL1830823)
Affinity DataEC50:  1.75E+3nMAssay Description:Agonist activity at GPR35 in human HT-29 cells by DMR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50259856(CHEMBL1600989)
Affinity DataEC50:  2.02E+3nMAssay Description:Agonist activity at GPR35 in human HT-29 cells by DMR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50436001(CHEMBL2392174 | CHEMBL2425818)
Affinity DataEC50:  12nMAssay Description:Agonist activity at human GPR35 expressed in CHO-K1 cells after 90 mins by beta-arrestin 2 recruitment assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM38549(2-[2-[4-[(4-chlorophenyl)-phenyl-methyl]piperazino...)
Affinity DataEC50:  500nMAssay Description:Agonist activity at human GPR35 expressed in CHO-K1 cells after 90 mins by beta-arrestin 2 recruitment assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50259887(CHEMBL3277775)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human GPR35 expressed in CHO-K1 cells after 90 mins by beta-arrestin 2 recruitment assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM35525(3,3''''-methylenebis(4-hydroxy-coumarin | 3,3''''-...)
Affinity DataEC50:  1.30E+3nMAssay Description:Agonist activity at human GPR35 expressed in CHO-K1 cells after 90 mins by beta-arrestin 2 recruitment assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM357857(Aphthasol | US10214536, Amlexanox)
Affinity DataEC50:  4.00E+3nMAssay Description:Agonist activity at human GPR35 expressed in CHO-K1 cells after 90 mins by beta-arrestin 2 recruitment assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50440033(CROMOLYN | Crolom | Cromoglicic Acid)
Affinity DataEC50:  7.00E+3nMAssay Description:Agonist activity at human GPR35 expressed in CHO-K1 cells after 90 mins by beta-arrestin 2 recruitment assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50259842(CHEMBL4079816)
Affinity DataEC50:  288nMAssay Description:Agonist activity at TEV protease cleavage site linked GAL4-VP16-fused GPR35 in human Tango GPR35-bla U2OS cells assessed as induction of TEV protease...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50259864(CHEMBL4093683)
Affinity DataEC50:  8.22E+3nMAssay Description:Agonist activity at GPR35 in human HT-29 cells by DMR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))
Dalian Institute of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50259860(CHEMBL4096323)
Affinity DataEC50:  4.27E+3nMAssay Description:Agonist activity at GPR35 in human HT-29 cells by DMR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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