Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50001330 Sort by
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
The Noguchi Institute

Curated by ChEMBL
LigandPNGBDBM50276373(CHEMBL4125713)
Affinity DataIC50: 800nMAssay Description:Inhibition of nigericin-induced NLRP3 inflammasome activation in C57BL/6 mouse bone marrow derived macrophages assessed as reduction in LPS-stimulate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
The Noguchi Institute

Curated by ChEMBL
LigandPNGBDBM50276377(CHEMBL4129636)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of nigericin-induced NLRP3 inflammasome activation in C57BL/6 mouse bone marrow derived macrophages assessed as reduction in LPS-stimulate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
The Noguchi Institute

Curated by ChEMBL
LigandPNGBDBM50276378(CHEMBL4126941)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of nigericin-induced NLRP3 inflammasome activation in C57BL/6 mouse bone marrow derived macrophages assessed as reduction in LPS-stimulate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
The Noguchi Institute

Curated by ChEMBL
LigandPNGBDBM50276376(CHEMBL4126909)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of nigericin-induced NLRP3 inflammasome activation in C57BL/6 mouse bone marrow derived macrophages assessed as reduction in LPS-stimulate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
The Noguchi Institute

Curated by ChEMBL
LigandPNGBDBM50276381(CHEMBL4128029)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of nigericin-induced NLRP3 inflammasome activation in PMA-differentiated human THP1 cells assessed as reduction in LPS-stimulated IL-1beta...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
The Noguchi Institute

Curated by ChEMBL
LigandPNGBDBM50276381(CHEMBL4128029)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of nigericin-induced NLRP3 inflammasome activation in C57BL/6 mouse bone marrow derived macrophages assessed as reduction in LPS-stimulate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
The Noguchi Institute

Curated by ChEMBL
LigandPNGBDBM50276377(CHEMBL4129636)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of nigericin-induced NLRP3 inflammasome activation in PMA-differentiated human THP1 cells assessed as reduction in LPS-stimulated IL-1beta...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
The Noguchi Institute

Curated by ChEMBL
LigandPNGBDBM50276376(CHEMBL4126909)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of nigericin-induced NLRP3 inflammasome activation in PMA-differentiated human THP1 cells assessed as reduction in LPS-stimulated IL-1beta...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
The Noguchi Institute

Curated by ChEMBL
LigandPNGBDBM50276372(CHEMBL4128176)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of nigericin-induced NLRP3 inflammasome activation in PMA-differentiated human THP1 cells assessed as reduction in LPS-stimulated IL-1beta...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
The Noguchi Institute

Curated by ChEMBL
LigandPNGBDBM50276373(CHEMBL4125713)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of nigericin-induced NLRP3 inflammasome activation in PMA-differentiated human THP1 cells assessed as reduction in LPS-stimulated IL-1beta...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
The Noguchi Institute

Curated by ChEMBL
LigandPNGBDBM50276375(CHEMBL4129407)
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of nigericin-induced NLRP3 inflammasome activation in PMA-differentiated human THP1 cells assessed as reduction in LPS-stimulated IL-1beta...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
The Noguchi Institute

Curated by ChEMBL
LigandPNGBDBM50276372(CHEMBL4128176)
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of nigericin-induced NLRP3 inflammasome activation in C57BL/6 mouse bone marrow derived macrophages assessed as reduction in LPS-stimulate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
The Noguchi Institute

Curated by ChEMBL
LigandPNGBDBM50276378(CHEMBL4126941)
Affinity DataIC50: 6.60E+3nMAssay Description:Inhibition of nigericin-induced NLRP3 inflammasome activation in PMA-differentiated human THP1 cells assessed as reduction in LPS-stimulated IL-1beta...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
The Noguchi Institute

Curated by ChEMBL
LigandPNGBDBM50276375(CHEMBL4129407)
Affinity DataIC50: 8.40E+3nMAssay Description:Inhibition of nigericin-induced NLRP3 inflammasome activation in C57BL/6 mouse bone marrow derived macrophages assessed as reduction in LPS-stimulate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
The Noguchi Institute

Curated by ChEMBL
LigandPNGBDBM50276380(CHEMBL4127699)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of nigericin-induced NLRP3 inflammasome activation in C57BL/6 mouse bone marrow derived macrophages assessed as reduction in LPS-stimulate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
The Noguchi Institute

Curated by ChEMBL
LigandPNGBDBM50276380(CHEMBL4127699)
Affinity DataIC50: 4.20E+4nMAssay Description:Inhibition of nigericin-induced NLRP3 inflammasome activation in PMA-differentiated human THP1 cells assessed as reduction in LPS-stimulated IL-1beta...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
The Noguchi Institute

Curated by ChEMBL
LigandPNGBDBM50276379(CHEMBL1234723 | CHEBI:16715)
Affinity DataIC50: 2.90E+7nMAssay Description:Inhibition of nigericin-induced NLRP3 inflammasome activation in C57BL/6 mouse bone marrow derived macrophages assessed as reduction in LPS-stimulate...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
The Noguchi Institute

Curated by ChEMBL
LigandPNGBDBM50276374(CHEMBL4126946)
Affinity DataIC50: 1.60E+6nMAssay Description:Inhibition of nigericin-induced NLRP3 inflammasome activation in C57BL/6 mouse bone marrow derived macrophages assessed as reduction in LPS-stimulate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
The Noguchi Institute

Curated by ChEMBL
LigandPNGBDBM50276374(CHEMBL4126946)
Affinity DataIC50: 2.30E+6nMAssay Description:Inhibition of nigericin-induced NLRP3 inflammasome activation in PMA-differentiated human THP1 cells assessed as reduction in LPS-stimulated IL-1beta...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed