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Report error Found 79 Enz. Inhib. hit(s) with all data for entry = 50009193 Sort by
TargetD(2) dopamine receptor(Human)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50001888([3-(2-Chloro-phenothiazin-10-yl)-propyl]-dimethyl-...)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]-raclopride from recombinant human D2 receptor expressed in HEK293 cells measured after 1 hr by microbeta scintillation counting ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50222218(CHEBI:51137 | Mianserin)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]-ketanserin from recombinant human 5HT2A receptor expressed in HEK293 cells measured after 1.5 hrs by microbeta scintillation cou...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM10755([3H]-5-HT | 5-Hydroxy Tryptamine | 2-imino-1-methy...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]-8-OH-DPAT from recombinant human 5HT1A receptor expressed in CHO cell membranes measured after 60 mins by microbeta scintillatio...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetD(2) dopamine receptor(Human)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  4.5nMAssay Description:Displacement of [3H]-raclopride from recombinant human D2 receptor expressed in HEK293 cells measured after 1 hr by microbeta scintillation counting ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM35254(CHEMBL715 | 2-methyl-4-(4-methylpiperazin-1-yl)-10...)
Affinity DataKi:  4.60nMAssay Description:Displacement of [3H]-ketanserin from recombinant human 5HT2A receptor expressed in HEK293 cells measured after 1.5 hrs by microbeta scintillation cou...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM35254(CHEMBL715 | 2-methyl-4-(4-methylpiperazin-1-yl)-10...)
Affinity DataKi:  7nMAssay Description:Displacement of [3H]-LSD from recombinant human 5HT6 receptor expressed in HEK293 cells measured after 1 hr by microbeta scintillation counting analy...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50526006(CHEMBL4515193)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]-citalopram from SERT in rat cortex tissue measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50001884(8-Chloro-11-(4-methyl-piperazin-1-yl)-5H-dibenzo[b...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]-5-CT from recombinant human 5HT7 receptor expressed in HEK293 cells measured after 1 hr by microbeta scintillation counting anal...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50526014(CHEMBL4469813)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]-ketanserin from recombinant human 5HT2A receptor expressed in HEK293 cells measured after 1.5 hrs by microbeta scintillation cou...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50526007(CHEMBL4451231)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]-8-OH-DPAT from recombinant human 5HT1A receptor expressed in CHO cell membranes measured after 60 mins by microbeta scintillatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50526025(CHEMBL4438147)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]-citalopram from SERT in rat cortex tissue measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50010859(CHEMBL11 | Imipramin | IMIPRAMINE HYDROCHLORIDE | ...)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]-citalopram from SERT in rat cortex tissue measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetSodium-dependent serotonin transporter(Rat)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50526021(CHEMBL4556098)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]-citalopram from SERT in rat cortex tissue measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50526014(CHEMBL4469813)
Affinity DataKi:  41nMAssay Description:Displacement of [3H]-citalopram from SERT in rat cortex tissue measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50526014(CHEMBL4469813)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]-8-OH-DPAT from recombinant human 5HT1A receptor expressed in CHO cell membranes measured after 60 mins by microbeta scintillatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(2) dopamine receptor(Human)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50001955(APOKYN | CHEMBL53 | (Apomorphine) 6-Methyl-5,6,6a,...)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]-raclopride from recombinant human D2 receptor expressed in HEK293 cells measured after 1 hr by microbeta scintillation counting ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50526008(CHEMBL4462139)
Affinity DataKi:  46nMAssay Description:Displacement of [3H]-8-OH-DPAT from recombinant human 5HT1A receptor expressed in CHO cell membranes measured after 60 mins by microbeta scintillatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50526008(CHEMBL4462139)
Affinity DataKi:  46nMAssay Description:Displacement of [3H]-citalopram from SERT in rat cortex tissue measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50526029(CHEMBL4587833)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]-8-OH-DPAT from recombinant human 5HT1A receptor expressed in CHO cell membranes measured after 60 mins by microbeta scintillatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50526030(CHEMBL4576769)
Affinity DataKi:  53nMAssay Description:Displacement of [3H]-8-OH-DPAT from recombinant human 5HT1A receptor expressed in CHO cell membranes measured after 60 mins by microbeta scintillatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50526015(CHEMBL4570209)
Affinity DataKi:  62nMAssay Description:Displacement of [3H]-8-OH-DPAT from recombinant human 5HT1A receptor expressed in CHO cell membranes measured after 60 mins by microbeta scintillatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50526027(CHEMBL4441125)
Affinity DataKi:  63nMAssay Description:Displacement of [3H]-8-OH-DPAT from recombinant human 5HT1A receptor expressed in CHO cell membranes measured after 60 mins by microbeta scintillatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50526007(CHEMBL4451231)
Affinity DataKi:  68nMAssay Description:Displacement of [3H]-citalopram from SERT in rat cortex tissue measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50526031(CHEMBL4470492)
Affinity DataKi:  69nMAssay Description:Displacement of [3H]-8-OH-DPAT from recombinant human 5HT1A receptor expressed in CHO cell membranes measured after 60 mins by microbeta scintillatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50526024(CHEMBL4459776)
Affinity DataKi:  76nMAssay Description:Displacement of [3H]-citalopram from SERT in rat cortex tissue measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50526012(CHEMBL4572860)
Affinity DataKi:  80nMAssay Description:Displacement of [3H]-8-OH-DPAT from recombinant human 5HT1A receptor expressed in CHO cell membranes measured after 60 mins by microbeta scintillatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50526013(CHEMBL4567376)
Affinity DataKi:  82nMAssay Description:Displacement of [3H]-citalopram from SERT in rat cortex tissue measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50526015(CHEMBL4570209)
Affinity DataKi:  86nMAssay Description:Displacement of [3H]-citalopram from SERT in rat cortex tissue measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50526026(CHEMBL4457041)
Affinity DataKi:  86nMAssay Description:Displacement of [3H]-citalopram from SERT in rat cortex tissue measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50526011(CHEMBL4466717)
Affinity DataKi:  87nMAssay Description:Displacement of [3H]-citalopram from SERT in rat cortex tissue measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50526024(CHEMBL4459776)
Affinity DataKi:  102nMAssay Description:Displacement of [3H]-8-OH-DPAT from recombinant human 5HT1A receptor expressed in CHO cell membranes measured after 60 mins by microbeta scintillatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50526029(CHEMBL4587833)
Affinity DataKi:  103nMAssay Description:Displacement of [3H]-citalopram from SERT in rat cortex tissue measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50526023(CHEMBL4439370)
Affinity DataKi:  115nMAssay Description:Displacement of [3H]-citalopram from SERT in rat cortex tissue measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50526012(CHEMBL4572860)
Affinity DataKi:  118nMAssay Description:Displacement of [3H]-citalopram from SERT in rat cortex tissue measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50526019(CHEMBL4441004)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]-8-OH-DPAT from recombinant human 5HT1A receptor expressed in CHO cell membranes measured after 60 mins by microbeta scintillatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50526028(CHEMBL4473888)
Affinity DataKi:  132nMAssay Description:Displacement of [3H]-8-OH-DPAT from recombinant human 5HT1A receptor expressed in CHO cell membranes measured after 60 mins by microbeta scintillatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50526020(CHEMBL4473005)
Affinity DataKi:  135nMAssay Description:Displacement of [3H]-citalopram from SERT in rat cortex tissue measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50526020(CHEMBL4473005)
Affinity DataKi:  136nMAssay Description:Displacement of [3H]-8-OH-DPAT from recombinant human 5HT1A receptor expressed in CHO cell membranes measured after 60 mins by microbeta scintillatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50526025(CHEMBL4438147)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]-8-OH-DPAT from recombinant human 5HT1A receptor expressed in CHO cell membranes measured after 60 mins by microbeta scintillatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50526021(CHEMBL4556098)
Affinity DataKi:  147nMAssay Description:Displacement of [3H]-8-OH-DPAT from recombinant human 5HT1A receptor expressed in CHO cell membranes measured after 60 mins by microbeta scintillatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50526026(CHEMBL4457041)
Affinity DataKi:  155nMAssay Description:Displacement of [3H]-8-OH-DPAT from recombinant human 5HT1A receptor expressed in CHO cell membranes measured after 60 mins by microbeta scintillatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50526016(CHEMBL4518119)
Affinity DataKi:  173nMAssay Description:Displacement of [3H]-citalopram from SERT in rat cortex tissue measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50526009(CHEMBL4563197)
Affinity DataKi:  176nMAssay Description:Displacement of [3H]-8-OH-DPAT from recombinant human 5HT1A receptor expressed in CHO cell membranes measured after 60 mins by microbeta scintillatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50526017(CHEMBL4570910)
Affinity DataKi:  192nMAssay Description:Displacement of [3H]-citalopram from SERT in rat cortex tissue measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50526027(CHEMBL4441125)
Affinity DataKi:  207nMAssay Description:Displacement of [3H]-citalopram from SERT in rat cortex tissue measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50526006(CHEMBL4515193)
Affinity DataKi:  209nMAssay Description:Displacement of [3H]-8-OH-DPAT from recombinant human 5HT1A receptor expressed in CHO cell membranes measured after 60 mins by microbeta scintillatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50526023(CHEMBL4439370)
Affinity DataKi:  218nMAssay Description:Displacement of [3H]-8-OH-DPAT from recombinant human 5HT1A receptor expressed in CHO cell membranes measured after 60 mins by microbeta scintillatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50526030(CHEMBL4576769)
Affinity DataKi:  240nMAssay Description:Displacement of [3H]-citalopram from SERT in rat cortex tissue measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50526005(CHEMBL4475065)
Affinity DataKi:  248nMAssay Description:Displacement of [3H]-citalopram from SERT in rat cortex tissue measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50526010(CHEMBL4451382)
Affinity DataKi:  255nMAssay Description:Displacement of [3H]-citalopram from SERT in rat cortex tissue measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
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