Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50009195 Sort by
LigandPNGBDBM96504(4-chloranyl-2-(2-naphthalen-1-yloxyethanoylamino)b...)
Affinity DataIC50: 400nMAssay Description:Inhibition of Flag-tagged TRPM4 (unknown origin) expressed in HEK293 cells assessed as reduction in intracellular Na+ influx after 45 mins by ANG2 dy...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50526037(CHEMBL4439848)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of Flag-tagged TRPM4 (unknown origin) expressed in HEK293 cells assessed as reduction in intracellular Na+ influx after 45 mins by ANG2 dy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
LigandPNGBDBM50526038(CHEMBL4525597)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of Flag-tagged TRPM4 (unknown origin) expressed in HEK293 cells assessed as reduction in intracellular Na+ influx after 45 mins by ANG2 dy...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50526034(CHEMBL4540384)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of Flag-tagged TRPM4 (unknown origin) expressed in HEK293 cells assessed as reduction in intracellular Na+ influx after 45 mins by ANG2 dy...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50526040(CHEMBL4447880)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of Flag-tagged TRPM4 (unknown origin) expressed in HEK293 cells assessed as reduction in intracellular Na+ influx after 45 mins by ANG2 dy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
LigandPNGBDBM50526032(CHEMBL4574460)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of Flag-tagged TRPM4 (unknown origin) expressed in HEK293 cells assessed as reduction in intracellular Na+ influx after 45 mins by ANG2 dy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
LigandPNGBDBM50526035(CHEMBL4472038)
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of Flag-tagged TRPM4 (unknown origin) expressed in HEK293 cells assessed as reduction in intracellular Na+ influx after 45 mins by ANG2 dy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
LigandPNGBDBM50526036(CHEMBL4554529)
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of Flag-tagged TRPM4 (unknown origin) expressed in HEK293 cells assessed as reduction in intracellular Na+ influx after 45 mins by ANG2 dy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
LigandPNGBDBM50526039(CHEMBL4465106)
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of Flag-tagged TRPM4 (unknown origin) expressed in HEK293 cells assessed as reduction in intracellular Na+ influx after 45 mins by ANG2 dy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
LigandPNGBDBM50526033(CHEMBL2407182 | CHEBI:28820)
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibition of TRPM4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed