Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50008913 Sort by
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50523489(CHEMBL4518093)
Affinity DataIC50: 35nMAssay Description:Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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PubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50523489(CHEMBL4518093)
Affinity DataIC50: 158nMAssay Description:Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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PubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50523491(CHEMBL4475410)
Affinity DataIC50: 414nMAssay Description:Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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PubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50523490(CHEMBL4575245)
Affinity DataIC50: 485nMAssay Description:Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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PubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50523488(CHEMBL4468450)
Affinity DataIC50: 810nMAssay Description:Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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PubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50523492(CHEMBL4453066)
Affinity DataIC50: 940nMAssay Description:Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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PubMed
TargetAdenosylhomocysteinase(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50523489(CHEMBL4518093)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of SAHH (unknown origin) using SAH as substrate preincubated for 10 mins followed by substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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PubMed
TargetProtein arginine N-methyltransferase 1(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50523489(CHEMBL4518093)
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of rat His6-tagged PRMT1 expressed in Escherichia coli BL21(DE3) using H4-21 peptide as substrate preincubated for 10 mins in presence of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetHistone-lysine N-methyltransferase EHMT2(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50523489(CHEMBL4518093)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human His-tagged G9a (913 to 1193 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL using H3-21 peptide as substrate prei...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetNicotinamide N-methyltransferase(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50523489(CHEMBL4518093)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human His-tagged NNMT (1 to 264 residues) expressed in Escherichia coli BL21(DE3) using 1-quinoline as substrate preincubated for 10 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetHistone-lysine N-methyltransferase SETD7(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50523489(CHEMBL4518093)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human His-tagged SETD7 (1 to 366 residues) expressed in Escherichia coli using H3-21 peptide as substrate preincubated for 10 mins in p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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PubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50523489(CHEMBL4518093)
Affinity DataKi:  39nMAssay Description:Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50523491(CHEMBL4475410)
Affinity DataKi:  103nMAssay Description:Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50523490(CHEMBL4575245)
Affinity DataKi:  121nMAssay Description:Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed