Compile Data Set for Download or QSAR
Report error Found 148 Enz. Inhib. hit(s) with all data for entry = 50012173
TargetProbable G-protein coupled receptor 88(Mouse)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50554975(CHEMBL4595209)
Affinity DataEC50:  25nMAssay Description:Agonist activity at GPR88 in mouse striatal membrane assessed as [35S]-GTPgammaS-binding by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50554975(CHEMBL4595209)
Affinity DataEC50:  47nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50554975(CHEMBL4595209)
Affinity DataEC50:  47nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50555038(CHEMBL4784623)
Affinity DataEC50:  59nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50555038(CHEMBL4784623)
Affinity DataEC50:  59nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50555041(CHEMBL4751633)
Affinity DataEC50:  71nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50555041(CHEMBL4751633)
Affinity DataEC50:  71nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50065915(CHEMBL3401461)
Affinity DataEC50:  72nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50065915(CHEMBL3401461)
Affinity DataEC50:  73nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50555044(CHEMBL4760182)
Affinity DataEC50:  74nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50555044(CHEMBL4760182)
Affinity DataEC50:  74nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50555043(CHEMBL4783876)
Affinity DataEC50:  78nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50555043(CHEMBL4783876)
Affinity DataEC50:  78nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50555036(CHEMBL4749371)
Affinity DataEC50:  112nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50555036(CHEMBL4749371)
Affinity DataEC50:  112nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50554994(CHEMBL4744793)
Affinity DataEC50:  120nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50554994(CHEMBL4744793)
Affinity DataEC50:  120nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50555045(CHEMBL4795623)
Affinity DataEC50:  138nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50555042(CHEMBL4789484)
Affinity DataEC50:  138nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50555045(CHEMBL4795623)
Affinity DataEC50:  138nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50555042(CHEMBL4789484)
Affinity DataEC50:  138nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50555037(CHEMBL4756228)
Affinity DataEC50:  148nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50555037(CHEMBL4756228)
Affinity DataEC50:  148nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50064644(CHEMBL3403767)
Affinity DataEC50:  174nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50064644(CHEMBL3403767)
Affinity DataEC50:  174nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50554996(CHEMBL4786591)
Affinity DataEC50:  182nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50554996(CHEMBL4786591)
Affinity DataEC50:  182nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50064645(CHEMBL3403768)
Affinity DataEC50:  195nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50064645(CHEMBL3403768)
Affinity DataEC50:  195nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50555004(CHEMBL4764798)
Affinity DataEC50:  209nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50555001(CHEMBL4763023)
Affinity DataEC50:  209nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50555004(CHEMBL4764798)
Affinity DataEC50:  209nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50555001(CHEMBL4763023)
Affinity DataEC50:  209nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50554999(CHEMBL4754332)
Affinity DataEC50:  214nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50554999(CHEMBL4754332)
Affinity DataEC50:  214nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50555018(CHEMBL4759273)
Affinity DataEC50:  219nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50555018(CHEMBL4759273)
Affinity DataEC50:  219nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50554982(CHEMBL4763920)
Affinity DataEC50:  234nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50555003(CHEMBL4760733)
Affinity DataEC50:  234nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50554982(CHEMBL4763920)
Affinity DataEC50:  234nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50555003(CHEMBL4760733)
Affinity DataEC50:  234nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50555000(CHEMBL4762227)
Affinity DataEC50:  240nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50555000(CHEMBL4762227)
Affinity DataEC50:  240nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50555017(CHEMBL4790074)
Affinity DataEC50:  245nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50554998(CHEMBL4787141)
Affinity DataEC50:  245nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50555017(CHEMBL4790074)
Affinity DataEC50:  245nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50554998(CHEMBL4787141)
Affinity DataEC50:  245nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50554979(CHEMBL4757666)
Affinity DataEC50:  251nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50554979(CHEMBL4757666)
Affinity DataEC50:  251nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 88(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50554980(CHEMBL4741911)
Affinity DataEC50:  257nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
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