Compile Data Set for Download or QSAR
Report error Found 102 Enz. Inhib. hit(s) with all data for entry = 50017573
TargetTau-tubulin kinase 1(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602886BDBM50602886(CHEMBL5182036)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of GST-tagged TTBK1 (1 to 421) (unknown origin) using DNA Topoisomerase 2-alpha-Thr1342 as substrate incubated for 15 mins followed by ATP...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetTau-tubulin kinase 2(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602886BDBM50602886(CHEMBL5182036)
Affinity DataIC50: 2.70nMAssay Description:Inhibition of TTBK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetTau-tubulin kinase 1(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602885BDBM50602885(CHEMBL5193906)
Affinity DataIC50: 120nMAssay Description:Inhibition of TTBK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetTau-tubulin kinase 2(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602885BDBM50602885(CHEMBL5193906)
Affinity DataIC50: 170nMAssay Description:Inhibition of TTBK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetTau-tubulin kinase 1(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 4622BDBM4622(CHEMBL127907 | 3-[(6,7-dimethoxyquinazolin-4-yl)am...)
Affinity DataKd:  240nMAssay Description:Binding affinity to CM5 sensor chip immobilized C-terminal His6/TEV fused-GST-tagged human TTBK1 (14 to 313 residues) expressed in baculovirus infect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetTau-tubulin kinase 1(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602904BDBM50602904(CHEMBL5204869 | US20250051335, Compound 2)
Affinity DataIC50: 240nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetTau-tubulin kinase 1(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602917BDBM50602917(CHEMBL5200069 | US20250051335, Compound 14)
Affinity DataIC50: 330nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetTau-tubulin kinase 1(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602907BDBM50602907(CHEMBL5193488 | US20250051335, Compound 5)
Affinity DataIC50: 340nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetTau-tubulin kinase 1(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602930BDBM50602930(CHEMBL5181249)
Affinity DataIC50: 360nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetTau-tubulin kinase 1(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602922BDBM50602922(CHEMBL5184336 | US20250051335, Compound 21)
Affinity DataIC50: 370nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetTau-tubulin kinase 1(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602921BDBM50602921(CHEMBL5180098 | US20250051335, Compound 18)
Affinity DataIC50: 380nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetTau-tubulin kinase 1(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602932BDBM50602932(CHEMBL5178965)
Affinity DataIC50: 390nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetTau-tubulin kinase 1(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602903BDBM50602903(CHEMBL5198544 | US20250051335, Compound 1)
Affinity DataIC50: 390nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetTau-tubulin kinase 1(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602910BDBM50602910(CHEMBL5209196 | US20250051335, Compound 8)
Affinity DataIC50: 420nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetTau-tubulin kinase 1(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602906BDBM50602906(CHEMBL5187459 | US20250051335, Compound 4)
Affinity DataIC50: 440nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetTau-tubulin kinase 1(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602920BDBM50602920(CHEMBL5187125 | US20250051335, Compound 20)
Affinity DataIC50: 450nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetTau-tubulin kinase 1(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602931BDBM50602931(CHEMBL5197012)
Affinity DataIC50: 480nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetTau-tubulin kinase 2(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602917BDBM50602917(CHEMBL5200069 | US20250051335, Compound 14)
Affinity DataIC50: 490nMAssay Description:Inhibition of recombinant human TTBK2 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetTau-tubulin kinase 1(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602900BDBM50602900(CHEMBL5185704 | US11814388, Compound 3)
Affinity DataIC50: 520nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetTau-tubulin kinase 1(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602911BDBM50602911(CHEMBL5171328 | US20250051335, Compound 9)
Affinity DataIC50: 520nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetTau-tubulin kinase 1(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602929BDBM50602929(CHEMBL5193034)
Affinity DataIC50: 610nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetTau-tubulin kinase 1(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602925BDBM50602925(CHEMBL5188513 | US20250051335, Compound 23)
Affinity DataIC50: 650nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetTau-tubulin kinase 1(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602934BDBM50602934(CHEMBL5206548)
Affinity DataIC50: 750nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetTau-tubulin kinase 1(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602909BDBM50602909(CHEMBL5197789 | US20250051335, Compound 7)
Affinity DataIC50: 750nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetTau-tubulin kinase 1(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602926BDBM50602926(CHEMBL5200160 | US11814388, Compound 9 | US2025005...)
Affinity DataIC50: 750nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetTau-tubulin kinase 1(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602905BDBM50602905(CHEMBL5208565 | US20250051335, Compound 3)
Affinity DataIC50: 770nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetTau-tubulin kinase 1(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602899BDBM50602899(CHEMBL5207783)
Affinity DataIC50: 790nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetTau-tubulin kinase 1(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602916BDBM50602916(CHEMBL5196033 | US20250051335, Compound 17)
Affinity DataIC50: 840nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetTau-tubulin kinase 2(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602903BDBM50602903(CHEMBL5198544 | US20250051335, Compound 1)
Affinity DataIC50: 850nMAssay Description:Inhibition of recombinant human TTBK2 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetTau-tubulin kinase 2(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602907BDBM50602907(CHEMBL5193488 | US20250051335, Compound 5)
Affinity DataIC50: 970nMAssay Description:Inhibition of recombinant human TTBK2 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetTau-tubulin kinase 1(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602933BDBM50602933(CHEMBL5178462)
Affinity DataIC50: 990nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetTau-tubulin kinase 1(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50328192BDBM50328192(N-(4-(Trifluoromethoxy)phenyl)-7H-pyrrolo[2,3-d]py...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetTau-tubulin kinase 1(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602912BDBM50602912(CHEMBL5179559 | US20250051335, Compound 10)
Affinity DataIC50: 1.02E+3nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetTau-tubulin kinase 2(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602909BDBM50602909(CHEMBL5197789 | US20250051335, Compound 7)
Affinity DataIC50: 1.21E+3nMAssay Description:Inhibition of recombinant human TTBK2 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetTau-tubulin kinase 2(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602926BDBM50602926(CHEMBL5200160 | US11814388, Compound 9 | US2025005...)
Affinity DataIC50: 1.21E+3nMAssay Description:Inhibition of recombinant human TTBK2 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetTau-tubulin kinase 2(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602910BDBM50602910(CHEMBL5209196 | US20250051335, Compound 8)
Affinity DataIC50: 1.24E+3nMAssay Description:Inhibition of recombinant human TTBK2 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetTau-tubulin kinase 2(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602900BDBM50602900(CHEMBL5185704 | US11814388, Compound 3)
Affinity DataIC50: 1.32E+3nMAssay Description:Inhibition of recombinant human TTBK2 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetTau-tubulin kinase 1(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602923BDBM50602923(CHEMBL5178871 | US20250051335, Compound 19)
Affinity DataIC50: 1.32E+3nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetTau-tubulin kinase 1(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602928BDBM50602928(CHEMBL5209161 | US20250051335, Compound 26)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetTau-tubulin kinase 1(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602901BDBM50602901(CHEMBL5202436)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetTau-tubulin kinase 1(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602914BDBM50602914(CHEMBL5192144 | US20250051335, Compound 12)
Affinity DataIC50: 1.55E+3nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetTau-tubulin kinase 1(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602896BDBM50602896(CHEMBL5182006)
Affinity DataIC50: 1.58E+3nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetTau-tubulin kinase 2(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602899BDBM50602899(CHEMBL5207783)
Affinity DataIC50: 1.68E+3nMAssay Description:Inhibition of recombinant human TTBK2 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetTau-tubulin kinase 1(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602927BDBM50602927(CHEMBL5193908 | US20250051335, Compound 25)
Affinity DataIC50: 1.71E+3nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetTau-tubulin kinase 2(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602933BDBM50602933(CHEMBL5178462)
Affinity DataIC50: 1.75E+3nMAssay Description:Inhibition of recombinant human TTBK2 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetTau-tubulin kinase 2(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602931BDBM50602931(CHEMBL5197012)
Affinity DataIC50: 2.03E+3nMAssay Description:Inhibition of recombinant human TTBK2 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetTau-tubulin kinase 2(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602906BDBM50602906(CHEMBL5187459 | US20250051335, Compound 4)
Affinity DataIC50: 2.14E+3nMAssay Description:Inhibition of recombinant human TTBK2 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetTau-tubulin kinase 1(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602913BDBM50602913(CHEMBL5207918 | US20250051335, Compound 11)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetTau-tubulin kinase 1(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50506661BDBM50506661(CHEMBL4517951)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetTau-tubulin kinase 1(Human)
Csic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602919BDBM50602919(CHEMBL5169390)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
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