Compile Data Set for Download or QSAR
maximum 50k data
Found 22 Enz. Inhib. hit(s) with all data for entry = 50018052
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50104413(CHEMBL87796 | Glutamyl-gamma-boronate analogue)
Affinity DataKi:  5.40nMAssay Description:Inhibition of human GGT1 transpeptidation in Pichia pastoris using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50104413(CHEMBL87796 | Glutamyl-gamma-boronate analogue)
Affinity DataKi:  25nMAssay Description:Inhibition of human GGT1 expressed in Pichia pastoris assessed as inhibition of GSH hydrolysis measured by L-glutamate release assayMore data for this Ligand-Target Pair
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50607251(CHEMBL5219012)
Affinity DataKi:  45nMAssay Description:Inhibition of human GGT1 transpeptidation in Pichia pastoris using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50607251(CHEMBL5219012)
Affinity DataKi:  77nMAssay Description:Inhibition of human GGT1 expressed in Pichia pastoris assessed as inhibition of GSH hydrolysis measured by L-glutamate release assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50607252(CHEMBL5219273)
Affinity DataKi:  2.60E+4nMAssay Description:Inhibition of human GGT1 transpeptidation in Pichia pastoris using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50607253(CHEMBL5220603)
Affinity DataKi:  4.60E+4nMAssay Description:Inhibition of human GGT1 transpeptidation in Pichia pastoris using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50607257(CHEMBL5219724)
Affinity DataKi:  4.90E+4nMAssay Description:Inhibition of human GGT1 transpeptidation in Pichia pastoris using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50607262(CHEMBL5218792)
Affinity DataKi:  6.10E+4nMAssay Description:Inhibition of human GGT1 transpeptidation in Pichia pastoris using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50607252(CHEMBL5219273)
Affinity DataKi:  8.70E+4nMAssay Description:Inhibition of human GGT1 expressed in Pichia pastoris assessed as inhibition of GSH hydrolysis measured by L-glutamate release assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50607258(CHEMBL5218962)
Affinity DataKi:  8.80E+4nMAssay Description:Inhibition of human GGT1 transpeptidation in Pichia pastoris using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50607257(CHEMBL5219724)
Affinity DataKi:  1.08E+5nMAssay Description:Inhibition of human GGT1 expressed in Pichia pastoris assessed as inhibition of GSH hydrolysis measured by L-glutamate release assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50607261(CHEMBL5218489)
Affinity DataKi:  1.73E+5nMAssay Description:Inhibition of human GGT1 transpeptidation in Pichia pastoris using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50607255(CHEMBL5219778)
Affinity DataKi:  2.02E+5nMAssay Description:Inhibition of human GGT1 transpeptidation in Pichia pastoris using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50607256(CHEMBL5220724)
Affinity DataKi:  2.20E+5nMAssay Description:Inhibition of human GGT1 transpeptidation in Pichia pastoris using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50607254(CHEMBL5219218)
Affinity DataKi:  2.54E+5nMAssay Description:Inhibition of human GGT1 transpeptidation in Pichia pastoris using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50607253(CHEMBL5220603)
Affinity DataKi:  2.60E+5nMAssay Description:Inhibition of human GGT1 expressed in Pichia pastoris assessed as inhibition of GSH hydrolysis measured by L-glutamate release assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50607259(CHEMBL5220006)
Affinity DataKi:  3.43E+5nMAssay Description:Inhibition of human GGT1 transpeptidation in Pichia pastoris using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50607256(CHEMBL5220724)
Affinity DataKi:  3.56E+5nMAssay Description:Inhibition of human GGT1 expressed in Pichia pastoris assessed as inhibition of GSH hydrolysis measured by L-glutamate release assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50607258(CHEMBL5218962)
Affinity DataKi:  5.08E+5nMAssay Description:Inhibition of human GGT1 expressed in Pichia pastoris assessed as inhibition of GSH hydrolysis measured by L-glutamate release assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50607260(CHEMBL5218520)
Affinity DataKi:  5.89E+5nMAssay Description:Inhibition of human GGT1 transpeptidation in Pichia pastoris using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50607254(CHEMBL5219218)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of human GGT1 expressed in Pichia pastoris assessed as inhibition of GSH hydrolysis measured by L-glutamate release assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50607255(CHEMBL5219778)
Affinity DataKi:  2.15E+6nMAssay Description:Inhibition of human GGT1 expressed in Pichia pastoris assessed as inhibition of GSH hydrolysis measured by L-glutamate release assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed