Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50021673
TargetP2X purinoceptor 7(Rat)
Nanchang University

Curated by ChEMBL
LigandPNGBDBM50234965(A-740003 | N-(1-{[(Cyanoimino)(5-quinolinylamino)m...)
Affinity DataIC50: 18nMAssay Description:Antagonist activity at rat P2X7 receptor by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetP2X purinoceptor 7(Human)
Nanchang University

Curated by ChEMBL
LigandPNGBDBM50234965(A-740003 | N-(1-{[(Cyanoimino)(5-quinolinylamino)m...)
Affinity DataIC50: 40nMAssay Description:Antagonist activity at human P2X7 receptor expressed in U-251 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetP2X purinoceptor 7(Human)
Nanchang University

Curated by ChEMBL
LigandPNGBDBM50414283(CHEMBL562308)
Affinity DataEC50:  1.00E+5nMAssay Description:Antagonist activity at human P2X7 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMedPDB3D3D Structure (crystal)