Compile Data Set for Download or QSAR
Report error Found 33 Enz. Inhib. hit(s) with all data for entry = 50021134
TargetSerine/threonine-protein kinase PLK4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50591934(CHEMBL5209160)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of PLK4 (unknown origin) by discoverX kinome scan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50591939(CHEMBL5185225)
Affinity DataKi:  0.160nMAssay Description:Binding affinity to PLK4 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50591932(CHEMBL5171469)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of PLK4 (unknown origin) by discoverX kinome scan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetAurora kinase A(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50004205(MK-0457 | MK-045 | VX-680 | VX-68 | TOZASERTIB | U...)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of Aurora-A (unknown origin) by kinase-glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50637358(CHEMBL5556344)
Affinity DataKi:  0.600nMAssay Description:Binding affinity to PLK4 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataKi:  2.60nMAssay Description:Binding affinity to full length PLK4 (unknown origin) using (TPSDSLIYDDGLS) biotinylated peptide as substrate assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM3033(Indolocarbazole deriv. | 3-{23-methyl-14-oxo-3,13,...)
Affinity DataKi:  3.40nMAssay Description:Binding affinity to full length PLK4 (unknown origin) using (TPSDSLIYDDGLS) biotinylated peptide as substrate assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM25117(AG-013736 | N-methyl-2-({3-[(E)-2-(pyridin-2-yl)et...)
Affinity DataIC50: 4.20nMAssay Description:Inhibition of PLK4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetAurora kinase C(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50004205(MK-0457 | MK-045 | VX-680 | VX-68 | TOZASERTIB | U...)
Affinity DataIC50: 4.60nMAssay Description:Inhibition of Aurora-C (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PAK 4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50591962(CHEMBL5175418)
Affinity DataIC50: 5.90nMAssay Description:Inhibition of PAK4 (unknown origin) incubated for 60 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50004205(MK-0457 | MK-045 | VX-680 | VX-68 | TOZASERTIB | U...)
Affinity DataKi:  7.70nMAssay Description:Binding affinity to PLK4 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50637354(CHEMBL5565760)
Affinity DataIC50: 11nMAssay Description:Inhibition of PLK4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50637357(CHEMBL5559612)
Affinity DataKi:  15nMAssay Description:Binding affinity to PLK4 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetAurora kinase B(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50004205(MK-0457 | MK-045 | VX-680 | VX-68 | TOZASERTIB | U...)
Affinity DataIC50: 18nMAssay Description:Inhibition of Aurora-B (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50591924(CHEMBL5179518)
Affinity DataIC50: 21nMAssay Description:Inhibition of PLK4 (unknown origin) by discoverX kinome scan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50591963(CHEMBL5173724)
Affinity DataIC50: 22nMAssay Description:Inhibition of PLK4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50437870(CHEMBL2407901)
Affinity DataIC50: 25nMAssay Description:Inhibition of PLK4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50637356(CHEMBL5558254)
Affinity DataIC50: 27nMAssay Description:Inhibition of PLK4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50355496(CHEMBL1908397)
Affinity DataIC50: 53nMAssay Description:Inhibition of PLK4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PAK 4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50591934(CHEMBL5209160)
Affinity DataIC50: 96nMAssay Description:Inhibition of PAK4 (unknown origin) incubated for 60 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50437869(CHEMBL2407902)
Affinity DataIC50: 100nMAssay Description:Inhibition of PLK4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 150nMAssay Description:Inhibition of full length PLK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PAK 4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50591920(CHEMBL5186873)
Affinity DataIC50: 273nMAssay Description:Inhibition of PAK4 (unknown origin) incubated for 60 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50591962(CHEMBL5175418)
Affinity DataIC50: 352nMAssay Description:Inhibition of PLK4 (unknown origin) by discoverX kinome scan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50591920(CHEMBL5186873)
Affinity DataIC50: 484nMAssay Description:Inhibition of PLK4 (unknown origin) by discoverX kinome scan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PAK 4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50591932(CHEMBL5171469)
Affinity DataIC50: 515nMAssay Description:Inhibition of PAK4 (unknown origin) incubated for 60 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 790nMAssay Description:Inhibition of full length PLK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK3(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of full length PLK3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PAK 4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50591924(CHEMBL5179518)
Affinity DataIC50: 1.96E+3nMAssay Description:Inhibition of PAK4 (unknown origin) incubated for 60 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50637355(CHEMBL5559158)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of PLK4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM3033(Indolocarbazole deriv. | 3-{23-methyl-14-oxo-3,13,...)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of full length PLK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK3(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM3033(Indolocarbazole deriv. | 3-{23-methyl-14-oxo-3,13,...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of full length PLK3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM3033(Indolocarbazole deriv. | 3-{23-methyl-14-oxo-3,13,...)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of full length PLK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed