Compile Data Set for Download or QSAR
Report error Found 33 Enz. Inhib. hit(s) with all data for entry = 50003414
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470598BDBM50470598(CHEMBL126050)
Affinity DataKi:  1nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470590BDBM50470590(CHEMBL341357)
Affinity DataKi:  1.30nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470591BDBM50470591(CHEMBL124208)
Affinity DataKi:  1.30nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470604BDBM50470604(CHEMBL338825)
Affinity DataKi:  1.30nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470596BDBM50470596(CHEMBL125310)
Affinity DataKi:  1.60nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470583BDBM50470583(CHEMBL125696)
Affinity DataKi:  1.60nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470587BDBM50470587(CHEMBL124648)
Affinity DataKi:  2.5nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470591BDBM50470591(CHEMBL124208)
Affinity DataKi:  2.5nMAssay Description:The compound was tested for binding affinity against Tachykinin receptor 2 from guinea pig tracheaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470603BDBM50470603(CHEMBL124013)
Affinity DataKi:  4nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470605BDBM50470605(CHEMBL122169)
Affinity DataKi:  4nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470582BDBM50470582(CHEMBL126043)
Affinity DataKi:  5nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470595BDBM50470595(CHEMBL122019)
Affinity DataKi:  6.30nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470599BDBM50470599(CHEMBL330766)
Affinity DataKi:  6.30nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470591BDBM50470591(CHEMBL124208)
Affinity DataKi:  7.90nMAssay Description:The compound was tested for binding affinity against Tachykinin receptor 2 from human expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470592BDBM50470592(CHEMBL339311)
Affinity DataKi:  7.90nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470606BDBM50470606(CHEMBL446099)
Affinity DataKi:  10nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470581BDBM50470581(CHEMBL341008)
Affinity DataKi:  10nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470597BDBM50470597(CHEMBL330826)
Affinity DataKi:  10nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470584BDBM50470584(CHEMBL125001)
Affinity DataKi:  13nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470585BDBM50470585(CHEMBL415518)
Affinity DataKi:  16nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470607BDBM50470607(CHEMBL124624)
Affinity DataKi:  20nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470608BDBM50470608(CHEMBL338030)
Affinity DataKi:  20nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470601BDBM50470601(CHEMBL123731)
Affinity DataKi:  20nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470589BDBM50470589(CHEMBL331011)
Affinity DataKi:  79nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470594BDBM50470594(CHEMBL340405)
Affinity DataKi:  100nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470602BDBM50470602(CHEMBL340747)
Affinity DataKi:  100nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470600BDBM50470600(CHEMBL435619)
Affinity DataKi:  100nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470586BDBM50470586(CHEMBL435610)
Affinity DataKi:  126nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470593BDBM50470593(CHEMBL126158)
Affinity DataKi:  200nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470588BDBM50470588(CHEMBL340548)
Affinity DataKi:  1.59E+3nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470591BDBM50470591(CHEMBL124208)
Affinity DataKi:  7.94E+3nMAssay Description:The compound was tested for binding affinity against Tachykinin receptor 1 from rabbit cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470591BDBM50470591(CHEMBL124208)
Affinity DataKi: <1.00E+4nMAssay Description:The compound was tested for binding affinity against Tachykinin receptor 1 from guinea pig tracheaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Guinea pig)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470591BDBM50470591(CHEMBL124208)
Affinity DataKi:  7.94E+4nMAssay Description:The compound was tested for binding affinity against Tachykinin receptor 3 from guinea pig cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed