Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 6693
TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM147469(US8957219, II-2-67)
Affinity DataIC50: 29nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2015
Entry Details
US Patent

TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM147471(US8957219, II-2-144)
Affinity DataIC50: 29nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2015
Entry Details
US Patent

TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM147472(US8957219, II-2-211)
Affinity DataIC50: 32nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2015
Entry Details
US Patent

TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM147473(US8957219, II-2-291)
Affinity DataIC50: 56nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2015
Entry Details
US Patent

TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM147470(US8957219, II-2-131)
Affinity DataIC50: 92nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2015
Entry Details
US Patent

TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM47169(US8957219, II-2-1)
Affinity DataIC50: 110nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2015
Entry Details
US Patent

TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM47168(US8957219, II-1-1)
Affinity DataIC50: 230nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2015
Entry Details
US Patent

TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM147468(US8957219, II-1-246)
Affinity DataIC50: 280nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2015
Entry Details
US Patent

TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM147467(US8957219, II-1-202)
Affinity DataIC50: 290nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2015
Entry Details
US Patent

TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM147464(US8957219, II-1-11)
Affinity DataIC50: 560nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2015
Entry Details
US Patent

TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM147465(US8957219, II-1-17)
Affinity DataIC50: 1.30E+3nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2015
Entry Details
US Patent

TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM147466(US8957219, II-1-190)
Affinity DataIC50: 2.10E+3nMT: 2°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2015
Entry Details
US Patent