Compile Data Set for Download or QSAR
Report error Found 240 Enz. Inhib. hit(s) with all data for entry = 7228
TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 181966BDBM181966(US9145380, 169)
Affinity DataIC50: 22nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 182037BDBM182037(US9145380, 240)
Affinity DataIC50: 31nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 181846BDBM181846(US9145380, 49)
Affinity DataIC50: 36nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 181802BDBM181802(US9145380, 5)
Affinity DataIC50: 40nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 182009BDBM182009(US9145380, 212)
Affinity DataIC50: 41nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 181815BDBM181815(US9145380, 18)
Affinity DataIC50: 44nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 182005BDBM182005(US9145380, 208)
Affinity DataIC50: 55nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 181833BDBM181833(US9145380, 36)
Affinity DataIC50: 57nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 181903BDBM181903(US9145380, 106)
Affinity DataIC50: 74nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 181803BDBM181803(US9145380, 6)
Affinity DataIC50: 74nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 182008BDBM182008(US9145380, 211)
Affinity DataIC50: 75nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 181822BDBM181822(US9145380, 25)
Affinity DataIC50: 77nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 181801BDBM181801(US9145380, 4)
Affinity DataIC50: 79nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 181980BDBM181980(US9145380, 183)
Affinity DataIC50: 81nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 181849BDBM181849(US9145380, 52)
Affinity DataIC50: 84nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 181889BDBM181889(US9145380, 92)
Affinity DataIC50: 91nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 182004BDBM182004(US9145380, 207)
Affinity DataIC50: 97nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 182021BDBM182021(US9145380, 224)
Affinity DataIC50: 100nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 182014BDBM182014(US9145380, 217)
Affinity DataIC50: 110nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 181840BDBM181840(US9145380, 43)
Affinity DataIC50: 110nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 181831BDBM181831(US9145380, 34)
Affinity DataIC50: 120nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 182013BDBM182013(US9145380, 216)
Affinity DataIC50: 130nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 182028BDBM182028(US9145380, 231)
Affinity DataIC50: 130nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 181847BDBM181847(US9145380, 50)
Affinity DataIC50: 130nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 181798BDBM181798(US9145380, 1)
Affinity DataIC50: 130nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 182025BDBM182025(US9145380, 228)
Affinity DataIC50: 130nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 181904BDBM181904(US9145380, 107)
Affinity DataIC50: 140nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 181800BDBM181800(US9145380, 3)
Affinity DataIC50: 140nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 182030BDBM182030(US9145380, 233)
Affinity DataIC50: 150nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 181834BDBM181834(US9145380, 37)
Affinity DataIC50: 160nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 181850BDBM181850(US9145380, 53)
Affinity DataIC50: 160nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 181832BDBM181832(US9145380, 35)
Affinity DataIC50: 170nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 182015BDBM182015(US9145380, 218)
Affinity DataIC50: 180nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 181813BDBM181813(US9145380, 16)
Affinity DataIC50: 190nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 181881BDBM181881(US9145380, 84)
Affinity DataIC50: 190nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 181961BDBM181961(US9145380, 164)
Affinity DataIC50: 190nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 181971BDBM181971(US9145380, 174)
Affinity DataIC50: 220nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 181918BDBM181918(US9145380, 121)
Affinity DataIC50: 220nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 181835BDBM181835(US9145380, 38)
Affinity DataIC50: 220nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 181867BDBM181867(US9145380, 70)
Affinity DataIC50: 220nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 182006BDBM182006(US9145380, 209)
Affinity DataIC50: 220nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 181983BDBM181983(US9145380, 186)
Affinity DataIC50: 250nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 181985BDBM181985(US9145380, 188)
Affinity DataIC50: 270nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 182017BDBM182017(US9145380, 220)
Affinity DataIC50: 270nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 181824BDBM181824(US9145380, 27)
Affinity DataIC50: 270nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 181851BDBM181851(US9145380, 54)
Affinity DataIC50: 270nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 181866BDBM181866(US9145380, 69)
Affinity DataIC50: 270nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 181820BDBM181820(US9145380, 23)
Affinity DataIC50: 270nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 181799BDBM181799(US9145380, 2)
Affinity DataIC50: 270nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

TargetProstaglandin E synthase 2(Human)
Astrazeneca

US Patent
LigandChemical structure of BindingDB Monomer ID 181826BDBM181826(US9145380, 29)
Affinity DataIC50: 280nMpH: 6.8Assay Description:A solution of test compound was added to a diluted microsome preparation containing human mPGES-1 and pre-incubated for 15 minutes in potassium phosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
US Patent

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