Compile Data Set for Download or QSAR
Report error Found 171 Enz. Inhib. hit(s) with all data for entry = 8249
TargetBromodomain-containing protein 3 [1-435](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237471BDBM237471(US9393232, 2.46)
Affinity DataIC50: 5.30nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 2 [1-473](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237471BDBM237471(US9393232, 2.46)
Affinity DataIC50: 6.60nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 4 [1-477](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 50156344BDBM50156344(CHEMBL3787210)
Affinity DataIC50: 8nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 2 [1-473](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237443BDBM237443(US9393232, 2.16)
Affinity DataIC50: 9.60nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 3 [1-435](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237443BDBM237443(US9393232, 2.16)
Affinity DataIC50: 9.90nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 4 [1-477](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237471BDBM237471(US9393232, 2.46)
Affinity DataIC50: 11nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 3 [1-435](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237494BDBM237494(US9393232, 4.1b | US9393232, 4.1a | US9393232, 4.1)
Affinity DataIC50: 14nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain testis-specific protein [1-397](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237471BDBM237471(US9393232, 2.46)
Affinity DataIC50: 14nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 2 [1-473](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237494BDBM237494(US9393232, 4.1b | US9393232, 4.1a | US9393232, 4.1)
Affinity DataIC50: 18nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 4 [1-477](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237443BDBM237443(US9393232, 2.16)
Affinity DataIC50: 19nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 4 [1-477](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237501BDBM237501(US9393232, 4.10a | BDBM237502)
Affinity DataIC50: 19nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain testis-specific protein [1-397](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237443BDBM237443(US9393232, 2.16)
Affinity DataIC50: 23nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 3 [1-435](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237521BDBM237521(US9393232, 2.22)
Affinity DataIC50: 23nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 3 [1-435](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237509BDBM237509(US9393232, 2.10b | US9393232, 2.10a)
Affinity DataIC50: 23nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 4 [1-477](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237428BDBM237428(US9393232, 2.2 | US9393232, 2.2b | US9393232, 2.2a)
Affinity DataIC50: 24nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 2 [1-473](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237509BDBM237509(US9393232, 2.10b | US9393232, 2.10a)
Affinity DataIC50: 24nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 4 [1-477](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237499BDBM237499(US9393232, 4.8)
Affinity DataIC50: 24nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 4 [1-477](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237533BDBM237533(US9393232, 4.6b | US9393232, 4.6a)
Affinity DataIC50: 24nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 4 [1-477](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 50156344BDBM50156344(CHEMBL3787210)
Affinity DataIC50: 24nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 4 [1-477](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237498BDBM237498(US9393232, 4.5)
Affinity DataIC50: 25nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 4 [1-477](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237437BDBM237437(US9393232, 2.9a | US9393232, 2.9b)
Affinity DataIC50: 25nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 4 [1-477](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237500BDBM237500(US9393232, 4.9a)
Affinity DataIC50: 25nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 3 [1-435](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237422BDBM237422(US9393232, 1.30a | US9393232, 1.30b)
Affinity DataIC50: 25nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 4 [1-477](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237470BDBM237470(US9393232, 2.45)
Affinity DataIC50: 26nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 4 [1-477](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237516BDBM237516(US9393232, 2.17a | US9393232, 2.17b | US9393232, 2...)
Affinity DataIC50: 26nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 4 [1-477](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237501BDBM237501(US9393232, 4.10a | BDBM237502)
Affinity DataIC50: 26nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 4 [1-477](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237516BDBM237516(US9393232, 2.17a | US9393232, 2.17b | US9393232, 2...)
Affinity DataIC50: 27nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 4 [1-477](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237467BDBM237467(US9393232, 2.42)
Affinity DataIC50: 27nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 4 [1-477](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237533BDBM237533(US9393232, 4.6b | US9393232, 4.6a)
Affinity DataIC50: 30nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain testis-specific protein [1-397](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237494BDBM237494(US9393232, 4.1b | US9393232, 4.1a | US9393232, 4.1)
Affinity DataIC50: 31nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 2 [1-473](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237521BDBM237521(US9393232, 2.22)
Affinity DataIC50: 32nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 4 [1-477](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237494BDBM237494(US9393232, 4.1b | US9393232, 4.1a | US9393232, 4.1)
Affinity DataIC50: 34nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 4 [1-477](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237391BDBM237391(US9393232, 1.1 | US9393232, 1.1a | US9393232, 1.1b)
Affinity DataIC50: 35nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 3 [1-435](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237428BDBM237428(US9393232, 2.2 | US9393232, 2.2b | US9393232, 2.2a)
Affinity DataIC50: 35nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 4 [1-477](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237482BDBM237482(US9393232, 2.59a | US9393232, 2.59b | US9393232, 2...)
Affinity DataIC50: 36nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 4 [1-477](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237432BDBM237432(US9393232, 2.4)
Affinity DataIC50: 36nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 4 [1-477](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237455BDBM237455(US9393232, 2.31)
Affinity DataIC50: 37nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 4 [1-477](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237535BDBM237535(US9393232, 4.9b)
Affinity DataIC50: 38nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 4 [1-477](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237516BDBM237516(US9393232, 2.17a | US9393232, 2.17b | US9393232, 2...)
Affinity DataIC50: 40nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 4 [1-477](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237479BDBM237479(US9393232, 2.57b | US9393232, 2.57a)
Affinity DataIC50: 41nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain testis-specific protein [1-397](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237521BDBM237521(US9393232, 2.22)
Affinity DataIC50: 42nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 4 [1-477](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237442BDBM237442(US9393232, 2.15)
Affinity DataIC50: 44nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 4 [1-477](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237496BDBM237496(US9393232, 4.3)
Affinity DataIC50: 49nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 4 [1-477](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237391BDBM237391(US9393232, 1.1 | US9393232, 1.1a | US9393232, 1.1b)
Affinity DataIC50: 51nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 4 [1-477](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237491BDBM237491(US9393232, 3.8)
Affinity DataIC50: 51nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 4 [1-477](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237485BDBM237485(US9393232, 3.2)
Affinity DataIC50: 52nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 2 [1-473](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237422BDBM237422(US9393232, 1.30a | US9393232, 1.30b)
Affinity DataIC50: 52nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 4 [1-477](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237490BDBM237490(US9393232, 3.7)
Affinity DataIC50: 53nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 4 [1-477](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237472BDBM237472(US9393232, 2.47)
Affinity DataIC50: 54nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

TargetBromodomain-containing protein 4 [1-477](Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 237461BDBM237461(US9393232, 2.37a | US9393232, 2.37b | US9393232, 2...)
Affinity DataIC50: 54nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
US Patent

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