Reaction Details
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Target
Dual specificity tyrosine-phosphorylation-regulated kinase 4
Ligand
BDBM50172243
Substrate
n/a
Meas. Tech.
ChEMBL_1579513 (CHEMBL3810711)
IC50
40±n/a nM
Citation
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More Info.:
Target
Name:
Dual specificity tyrosine-phosphorylation-regulated kinase 4
Synonyms:
DYRK4 | DYRK4_HUMAN
Type:
PROTEIN
Mol. Mass.:
59629.96
Organism:
Homo sapiens (Human)
Description:
ChEMBL_1475744
Residue:
520
Sequence:
MPASELKASEIPFHPSIKTQDPKAEEKSPKKQKVTLTAAEALKLFKNQLSPYEQSEILGYAELWFLGLEAKKLDTAPEKFSKTSFDDEHGFYLKVLHDHIAYRYEVLETIGKGSFGQVAKCLDHKNNELVALKIIRNKKRFHQQALMELKILEALRKKDKDNTYNVVHMKDFFYFRNHFCITFELLGINLYELMKNNNFQGFSLSIVRRFTLSVLKCLQMLSVEKIIHCDLKPENIVLYQKGQASVKVIDFGSSCYEHQKVYTYIQSRFYRSPEVILGHPYDVAIDMWSLGCITAELYTGYPLFPGENEVEQLACIMEVLGLPPAGFIQTASRRQTFFDSKGFPKNITNNRGKKRYPDSKDLTMVLKTYDTSFLDFLRRCLVWEPSLRMTPDQALKHAWIHQSRNLKPQPRPQTLRKSNSFFPSETRKDKVQGCHHSSRKADEITKETTEKTKDSPTKHVQHSGDQQDCLQHGADTVQLPQLVDAPKKSEAAVGAEVSMTSPGQSKNFSLKNTNVLPPIV