Reaction Details Report a problem with these data
Target
Receptor protein-tyrosine kinase
Ligand
BDBM532954
Substrate
n/a
Meas. Tech.
Human, Dog and Rat c-Fms Enzyme Assay (Fluorescence Immunoassay Format)
IC50
8.00±n/a nM
Citation
Chen, J; Donahue, M; Lim, H; Lin, R; Salter, R; Wu, J; Gong, Y Substituted pyridine derivatives useful as C-FMS kinase inhibitors US Patent US11214566 Publication Date 1/4/2022
More Info.:
Target
Name:
Receptor protein-tyrosine kinase
Synonyms:
A0A8C0LZB8_CANLF | CSF1R | Colony stimulating factor 1 receptor
Type:
Protein
Mol. Mass.:
110154.61
Organism:
Dog
Description:
A0A8C0LZB8
Residue:
1003
Sequence:
MGLGAPLVLLVATAWHVQGVPVIEPRGPELVVEPGTAVTLRCVGNGSVEWEGPISPHWNLDPDSPSSILSTNNATFLNTGTYRCTEPGSPLGGSATIHIYVKDPVRPWKVLTQEVTVLEGQDALLPCLLTDPALEAGVSLMRVRGRPVLRQTNYSFSPWYGFTIHKAQFTETQGYQCSARVGGRMVTSMGIWLKVQKVIPGPPTLTLKPAELVRIQGEAANIECSASNVDVNFDVFLQHEDTKLTIPQQSDFQGNQYQKVLTLELDHVGFQDAGNYTCVATNVRGISSTSMIFRVVESAYLNLTSEQSLLQEVTVGEKVDLQVKVEAYPSLEGYNWTYLGPFSDQQAKLKFVITKDTYRYTSTLSLPRLKPSEAGRYSFLARNTRGGDSLTFELTLRYPPEVRITWTTVNGSDALLCEASGYPQPNVTWLQCRGHTDRCDEAQALVLEDSYSEVLSQEPFHKVIVHSLLAMGTMEHNMTYECRALNSVGNSSQAFRPIPIGAHIQPPDEPLFTPVLVTCMSIMVLLLLLLLLLFYKYKQKPKYQVRWKIIESYEGNSYTFIDPTQLPYNEKWEFPRNNLQFGKTLGAGAFGKVVEATAFGLGKEDAVLKVAVKMLKSTAHADEKEALMSELKIMSHLGQHENIVNLLGACTHGGPVLVITEYCCYGDLLNFLRRKAEAMLGPSVSVGQDPGAGAGYKNIHLEKKYVRRDSGFSSQGVDTYVEMRPVSTSSSNDSFSEQDLDKEDGRPLELRDLLHFSSQVAQGMAFLASKNCIHRDVAARNVLLTSGRVAKIGDFGLARDIMNDSNYIVKGNARLPVKWMAPESIFDCVYTVQSDVWSYGILLWEIFSLDTASCRPAGPWSPPEDPPSSRSAPSSRSRPKQTGESQTTPICQAAAVAVAAVVSQRRRALASTWPAVNRGILPSPCCSPTTTSSAEETTGKHCFSLPPSFNSTVDGAPRRGAYGLCPWSFHSTARPSSESQECEIHRSLGRTLPGPGPSLPVRG