Compile Data Set for Download or QSAR
Report error Found 200 of affinity data for UniProtKB/TrEMBL: O00418
TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50343559BDBM50343559(1-(2-HYDROXYETHYL)-8-[[5-(4-METHYLPIPERAZIN-1-YL)-...)
Affinity DataIC50: 10nMAssay Description:Inhibition of EEF2K (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50442760BDBM50442760(CHEMBL2443044)
Affinity DataIC50: 10nMAssay Description:Inhibition of eEF2K (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50442759BDBM50442759(CHEMBL2443138)
Affinity DataIC50: 10nMAssay Description:Inhibition of eEF2K (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50442758BDBM50442758(CHEMBL2443139)
Affinity DataIC50: 10nMAssay Description:Inhibition of eEF2K (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50442757BDBM50442757(CHEMBL2443026)
Affinity DataIC50: 10nMAssay Description:Inhibition of eEF2K (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50600470BDBM50600470(CHEMBL5174034)
Affinity DataIC50: 32nMAssay Description:Inhibition of eEF2K (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50555899BDBM50555899(CHEMBL1683636)
Affinity DataIC50: 60nMAssay Description:Inhibition of eEF2K (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50284911BDBM50284911(CHEMBL4171806)
Affinity DataIC50: 60nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human eEF2K expressed in Escherichia coli using biotinylated myelin basic protein as substrate after ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50600471BDBM50600471(CHEMBL5204448)
Affinity DataIC50: 69nMAssay Description:Inhibition of eEF2K (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50314444BDBM50314444(2-(4-chlorophenyl)-10-thia-5,7,12-triazatetracyclo...)
Affinity DataIC50: 110nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50314436BDBM50314436(3-amino-4-(furan-2-yl)-6,7,8,9,10,11-hexahydro-5H-...)
Affinity DataIC50: 170nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50314406BDBM50314406(8-(morpholin-4-yl)-11-thia-9,14,16-triazatetracycl...)
Affinity DataIC50: 220nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50314406BDBM50314406(8-(morpholin-4-yl)-11-thia-9,14,16-triazatetracycl...)
Affinity DataIC50: 220nMAssay Description:Inhibition of eEF2K (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50600472BDBM50600472(CHEMBL5194579)
Affinity DataIC50: 230nMAssay Description:Inhibition of eEF2K (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50314427BDBM50314427(3-amino-4-(5-chlorofuran-2-yl)-5,6,7,8,9,10-hexahy...)
Affinity DataIC50: 280nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50053584BDBM50053584(CHEMBL1977874)
Affinity DataIC50: 280nMAssay Description:Inhibition of eEF2K (unknown origin) measured after 30 mins of incubationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50053584BDBM50053584(CHEMBL1977874)
Affinity DataIC50: 280nMAssay Description:ATP competitive inhibition of human eEF-2K using 5 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50053584BDBM50053584(CHEMBL1977874)
Affinity DataIC50: 280nMAssay Description:Inhibition of eEF2K (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50314428BDBM50314428(3-amino-4-(5-(trifluoromethyl)furan-2-yl)-5,6,7,8,...)
Affinity DataIC50: 300nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 293963BDBM293963(US10106552, Compound 38)
Affinity DataIC50: 300nMAssay Description:To determine the IC50 of compounds of the invention, recombinant eEF2K was diluted in an assay buffer in the presence of calmodulin, a calcium-bindin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2019
Entry Details
US Patent

TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50555900BDBM50555900(CHEMBL4776943)
Affinity DataIC50: 310nMAssay Description:Inhibition of eEF2K (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50314419BDBM50314419((E)-3-amino-4-(2-(furan-2-yl)vinyl)-5,6,7,8,9,10-h...)
Affinity DataIC50: 320nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50314429BDBM50314429(3-amino-4-(benzofuran-2-yl)-5,6,7,8,9,10-hexahydro...)
Affinity DataIC50: 330nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50646956BDBM50646956(CHEMBL5593199)
Affinity DataKd:  330nMAssay Description:Binding affinity to eEF2K (unknown origin) assessed as dissociation constant measured by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50314442BDBM50314442(2-(furan-2-yl)-10-thia-5,7,12-triazatetracyclo[11....)
Affinity DataIC50: 350nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 293960BDBM293960(US10106552, Compound 35)
Affinity DataIC50: 400nMAssay Description:To determine the IC50 of compounds of the invention, recombinant eEF2K was diluted in an assay buffer in the presence of calmodulin, a calcium-bindin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2019
Entry Details
US Patent

TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 293961BDBM293961(US10106552, Compound 36)
Affinity DataIC50: 400nMAssay Description:To determine the IC50 of compounds of the invention, recombinant eEF2K was diluted in an assay buffer in the presence of calmodulin, a calcium-bindin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2019
Entry Details
US Patent

TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 293965BDBM293965(US10106552, Compound 40)
Affinity DataIC50: 400nMAssay Description:To determine the IC50 of compounds of the invention, recombinant eEF2K was diluted in an assay buffer in the presence of calmodulin, a calcium-bindin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2019
Entry Details
US Patent

TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 293953BDBM293953(US10106552, Compound 28)
Affinity DataIC50: 400nMAssay Description:To determine the IC50 of compounds of the invention, recombinant eEF2K was diluted in an assay buffer in the presence of calmodulin, a calcium-bindin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2019
Entry Details
US Patent

TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50053584BDBM50053584(CHEMBL1977874)
Affinity DataIC50: 420nMAssay Description:Inhibition of human recombinant eEF-2K expressed in bacteria pre-incubated for 30 mins before adding peptide substrate and [gamma32P]ATP by scintilla...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50053584BDBM50053584(CHEMBL1977874)
Affinity DataIC50: 420nMAssay Description:Inhibition of eEF2K (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50646955BDBM50646955(CHEMBL5590973)
Affinity DataKd:  436nMAssay Description:Binding affinity to eEF2K (unknown origin) assessed as dissociation constant measured by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50375667BDBM50375667(TX-1918 | CHEMBL437612)
Affinity DataIC50: 440nMAssay Description:Inhibition of eEF2 kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50375667BDBM50375667(TX-1918 | CHEMBL437612)
Affinity DataIC50: 440nMAssay Description:Inhibition of eEF2K (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50375667BDBM50375667(TX-1918 | CHEMBL437612)
Affinity DataIC50: 440nMAssay Description:Inhibition of eEF2K in human A431 cells using eEF2 as substrate preincubated for 30 mins followed by ATP/[gamma-32P]-ATP addition measured after 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50314420BDBM50314420(3-amino-4-(3-methylthiophen-2-yl)-5,6,7,8,9,10-hex...)
Affinity DataIC50: 460nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50646957BDBM50646957(CHEMBL5592236)
Affinity DataKd:  492nMAssay Description:Binding affinity to eEF2K (unknown origin) assessed as dissociation constant measured by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 293966BDBM293966(US10106552, Compound 41)
Affinity DataIC50: 500nMAssay Description:To determine the IC50 of compounds of the invention, recombinant eEF2K was diluted in an assay buffer in the presence of calmodulin, a calcium-bindin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2019
Entry Details
US Patent

TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50053584BDBM50053584(CHEMBL1977874)
Affinity DataIC50: 510nMAssay Description:Inhibition of eEF2K (unknown origin) using peptide MH-1 as substrate after 2 hrs by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50314418BDBM50314418(3-amino-4-(furan-2-yl)-5,6,7,8,9,10-hexahydrocyclo...)
Affinity DataIC50: 640nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50314430BDBM50314430(3-amino-4-(5-ethylfuran-2-yl)-5,6,7,8,9,10-hexahyd...)
Affinity DataIC50: 660nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 293954BDBM293954(US10106552, Compound 29)
Affinity DataIC50: 700nMAssay Description:To determine the IC50 of compounds of the invention, recombinant eEF2K was diluted in an assay buffer in the presence of calmodulin, a calcium-bindin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2019
Entry Details
US Patent

TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50464814BDBM50464814(CHEMBL4281348)
Affinity DataIC50: 760nMAssay Description:Inhibition of eEF2K (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50464814BDBM50464814(CHEMBL4281348)
Affinity DataIC50: 762nMAssay Description:Inhibition of GST-tagged EEF2K (unknown origin) using biotinylated EEF2 peptide substrate by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 293959BDBM293959(US10106552, Compound 34)
Affinity DataIC50: 800nMAssay Description:To determine the IC50 of compounds of the invention, recombinant eEF2K was diluted in an assay buffer in the presence of calmodulin, a calcium-bindin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2019
Entry Details
US Patent

TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50314431BDBM50314431(3-amino-4-(5-(hydroxymethyl)furan-2-yl)-5,6,7,8,9,...)
Affinity DataIC50: 800nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 293950BDBM293950(US10106552, Compound 25)
Affinity DataIC50: 800nMAssay Description:To determine the IC50 of compounds of the invention, recombinant eEF2K was diluted in an assay buffer in the presence of calmodulin, a calcium-bindin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2019
Entry Details
US Patent

TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50314415BDBM50314415(4-(3-amino-2-carbamoyl-5,6,7,8,9,10-hexahydrocyclo...)
Affinity DataIC50: 860nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50314409BDBM50314409(3-amino-4-isobutyl-5,6,7,8,9,10-hexahydrocycloocta...)
Affinity DataIC50: 860nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Nerviano Medical Sciences Srl

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 293943BDBM293943(US10106552, Compound 18)
Affinity DataIC50: 900nMAssay Description:To determine the IC50 of compounds of the invention, recombinant eEF2K was diluted in an assay buffer in the presence of calmodulin, a calcium-bindin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2019
Entry Details
US Patent

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