Compile Data Set for Download or QSAR
Report error Found 136 of affinity data for UniProtKB/TrEMBL: Q14330
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50056486(((5Z,8Z,11Z,14Z)-Icosa-5,8,11,14-tetraenoylamino)-...)
Affinity DataEC50:  20nMAssay Description:Agonist activity at recombinant full length human GPR18 expressed in CHO cells assessed as forskolin-stimulated cAMP accumulation after 10 mins by en...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50056486(((5Z,8Z,11Z,14Z)-Icosa-5,8,11,14-tetraenoylamino)-...)
Affinity DataEC50:  44nMAssay Description:Agonist activity at recombinant human GPR18 expressed in HEK293 cells assessed as induction of p44/42 MAPK phosphorylation after 5 mins by Western bl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449597(CHEMBL4174825)
Affinity DataIC50: 238nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50561705(CHEMBL4758188)
Affinity DataEC50:  454nMAssay Description:Agonist activity at Prolink1-tagged human GPR18 receptor expressed in CHO cells assessed as induction of beta-arrestin recruitment after 90 mins by b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50221691(9-(2-(1H-indol-3-yl)ethyl)-1,3-dimethyl-6,7,8,9-te...)
Affinity DataEC50:  562nMAssay Description:Agonist activity at Prolink1-tagged human GPR18 receptor expressed in CHO cells assessed as induction of beta-arrestin recruitment after 90 mins by b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449561(CHEMBL4168457)
Affinity DataIC50: 650nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50221691(9-(2-(1H-indol-3-yl)ethyl)-1,3-dimethyl-6,7,8,9-te...)
Affinity DataIC50: 944nMAssay Description:Agonist activity at Prolink1-tagged human GPR18 receptor expressed in CHO cells assessed as induction of beta-arrestin recruitment by measuring 2-(3-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449598(CHEMBL4176317)
Affinity DataIC50: 1.14E+3nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449584(CHEMBL4169939)
Affinity DataIC50: 1.15E+3nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449599(CHEMBL4169536)
Affinity DataIC50: 1.49E+3nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449578(CHEMBL4159298)
Affinity DataIC50: 1.71E+3nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449560(CHEMBL4168388)
Affinity DataIC50: 1.73E+3nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449577(CHEMBL4162436)
Affinity DataIC50: 2.29E+3nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449564(CHEMBL4171815)
Affinity DataIC50: 2.38E+3nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449587(CHEMBL4161205)
Affinity DataIC50: 3.25E+3nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449579(CHEMBL4172931)
Affinity DataIC50: 3.59E+3nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM60994((10R,10aR)-6,6,9-Trimethyl-3-pentyl-6a,7,8,10a-tet...)
Affinity DataEC50:  4.61E+3nMAssay Description:Agonist activity at human GPR18 transfected in CHO cells after 90 mins by beta-arrestin translocation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449565(CHEMBL4177155)
Affinity DataIC50: 4.78E+3nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449563(CHEMBL4161619)
Affinity DataIC50: 5.00E+3nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50561706(CHEMBL4780863)
Affinity DataEC50:  5.68E+3nMAssay Description:Agonist activity at Prolink1-tagged human GPR18 receptor expressed in CHO cells assessed as induction of beta-arrestin recruitment after 90 mins by b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50072775(ChEMBL_75020 | 5-(1,1-Dimethyl-heptyl)-2-[(1R,2R,5...)
Affinity DataIC50: 5.99E+3nMAssay Description:Antagonist activity at human GPR18 transfected in CHO cells assessed as delta9-THC-induced beta-arrestin recruitment incubated 60 mins prior to delta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50398222(CHEMBL2177264)
Affinity DataIC50: 8.10E+3nMAssay Description:Antagonist activity at human GPR18 transfected in CHO cells assessed as delta9-THC-induced beta-arrestin recruitment incubated 60 mins prior to delta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50448075(CHEMBL1258979)
Affinity DataIC50: 9.91E+3nMAssay Description:Inverse agonist activity at human GPR18 expressed in CHO cells assessed as inhibition of 7.5 uM THC-mediated beta-arrestin recruitment after 90 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449583(CHEMBL4160778)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449582(CHEMBL4170355)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at recombinant human GPR18 expressed in CHO cells assessed as increase in beta-arrestin recruitment incubated for 60 mins measured f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449591(CHEMBL4165882)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449590(CHEMBL4160494)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at recombinant human GPR18 expressed in CHO cells assessed as increase in beta-arrestin recruitment incubated for 60 mins measured f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449580(CHEMBL4174205)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at recombinant human GPR18 expressed in CHO cells assessed as increase in beta-arrestin recruitment incubated for 60 mins measured f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449577(CHEMBL4162436)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at recombinant human GPR18 expressed in CHO cells assessed as increase in beta-arrestin recruitment incubated for 60 mins measured f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449588(CHEMBL4169314)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at recombinant human GPR18 expressed in CHO cells assessed as increase in beta-arrestin recruitment incubated for 60 mins measured f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449580(CHEMBL4174205)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449587(CHEMBL4161205)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at recombinant human GPR18 expressed in CHO cells assessed as increase in beta-arrestin recruitment incubated for 60 mins measured f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449578(CHEMBL4159298)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at recombinant human GPR18 expressed in CHO cells assessed as increase in beta-arrestin recruitment incubated for 60 mins measured f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50056486(((5Z,8Z,11Z,14Z)-Icosa-5,8,11,14-tetraenoylamino)-...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at Prolink1-tagged human GPR18 receptor expressed in CHO cells assessed as induction of beta-arrestin recruitment after 90 mins by b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449589(CHEMBL4173561)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at recombinant human GPR18 expressed in CHO cells assessed as increase in beta-arrestin recruitment incubated for 60 mins measured f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50552130(CHEMBL499876)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at Prolink1-tagged human GPR18 receptor expressed in CHO cells assessed as induction of beta-arrestin recruitment after 90 mins by b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50398229(CHEMBL2177257)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human GPR18 transfected in CHO cells assessed as delta9-THC-induced beta-arrestin recruitment incubated 60 mins prior to delta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50398237(CHEMBL2177249)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human GPR18 transfected in CHO cells assessed as delta9-THC-induced beta-arrestin recruitment incubated 60 mins prior to delta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449586(CHEMBL4171382)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449589(CHEMBL4173561)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50434879(CHEMBL2387535)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human GPR18 transfected in CHO cells assessed as delta9-THC-induced beta-arrestin recruitment incubated 60 mins prior to delta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50434878(CHEMBL2387536)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human GPR18 transfected in CHO cells assessed as delta9-THC-induced beta-arrestin recruitment incubated 60 mins prior to delta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50434877(CHEMBL2387538)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human GPR18 transfected in CHO cells assessed as delta9-THC-induced beta-arrestin recruitment incubated 60 mins prior to delta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50434876(CHEMBL2387539)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human GPR18 transfected in CHO cells assessed as delta9-THC-induced beta-arrestin recruitment incubated 60 mins prior to delta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449562(CHEMBL4165036)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449585(CHEMBL4159707)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at recombinant human GPR18 expressed in CHO cells assessed as increase in beta-arrestin recruitment incubated for 60 mins measured f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449593(CHEMBL4163505)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at recombinant human GPR18 expressed in CHO cells assessed as increase in beta-arrestin recruitment incubated for 60 mins measured f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449565(CHEMBL4177155)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at recombinant human GPR18 expressed in CHO cells assessed as increase in beta-arrestin recruitment incubated for 60 mins measured f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449588(CHEMBL4169314)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449579(CHEMBL4172931)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at recombinant human GPR18 expressed in CHO cells assessed as increase in beta-arrestin recruitment incubated for 60 mins measured f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
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