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TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 86139BDBM86139(CAS_235433-36-0 | PrRP31 | CAS_99566-27-5 | NSC_0 ...)
Affinity DataKi:  0.680nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2012
Entry Details Article
PubMed
TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 86148BDBM86148(CAS_222988-10-5 | PrRP20)
In Depth
Date in BDB:
5/24/2012
Entry Details Article
PubMed
TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 195624BDBM195624(US9206173, 2386)
Affinity DataKi:  2nM ΔG°:  -49.7kJ/molepH: 7.4 T: 2°CAssay Description:Receptor-expressing HEK 293 cell membrane fraction was analyzed by modifying the methods of C. J. Langmead et al. (see Langmead C J, Szekeres P G; Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details
US Patent

TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 195673BDBM195673(US9206173, 2435)
Affinity DataKi:  2nM ΔG°:  -49.7kJ/molepH: 7.4 T: 2°CAssay Description:Receptor-expressing HEK 293 cell membrane fraction was analyzed by modifying the methods of C. J. Langmead et al. (see Langmead C J, Szekeres P G; Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details
US Patent

TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 195644BDBM195644(US9206173, 2406)
Affinity DataKi:  2nM ΔG°:  -49.7kJ/molepH: 7.4 T: 2°CAssay Description:Receptor-expressing HEK 293 cell membrane fraction was analyzed by modifying the methods of C. J. Langmead et al. (see Langmead C J, Szekeres P G; Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details
US Patent

TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 195701BDBM195701(US9206173, 2463)
Affinity DataKi:  3nM ΔG°:  -48.6kJ/molepH: 7.4 T: 2°CAssay Description:Receptor-expressing HEK 293 cell membrane fraction was analyzed by modifying the methods of C. J. Langmead et al. (see Langmead C J, Szekeres P G; Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details
US Patent

TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 195733BDBM195733(US9206173, 2495)
Affinity DataKi:  3nM ΔG°:  -48.6kJ/molepH: 7.4 T: 2°CAssay Description:Receptor-expressing HEK 293 cell membrane fraction was analyzed by modifying the methods of C. J. Langmead et al. (see Langmead C J, Szekeres P G; Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details
US Patent

TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50553347BDBM50553347(CHEMBL4756509)
Affinity DataEC50:  3.90nMAssay Description:Activation of human GPR10 overexpressed in CHO-K1 cells assessed as increase in beta arrestin recruitment incubated for 90 mins by PathHunter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 195690BDBM195690(US9206173, 2452)
Affinity DataKi:  4nM ΔG°:  -47.9kJ/molepH: 7.4 T: 2°CAssay Description:Receptor-expressing HEK 293 cell membrane fraction was analyzed by modifying the methods of C. J. Langmead et al. (see Langmead C J, Szekeres P G; Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details
US Patent

TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 195613BDBM195613(US9206173, 1)
Affinity DataKi:  5nM ΔG°:  -47.4kJ/molepH: 7.4 T: 2°CAssay Description:Receptor-expressing HEK 293 cell membrane fraction was analyzed by modifying the methods of C. J. Langmead et al. (see Langmead C J, Szekeres P G; Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details
US Patent

TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 195749BDBM195749(US9206173, 95)
Affinity DataKi:  5nM ΔG°:  -47.4kJ/molepH: 7.4 T: 2°CAssay Description:Receptor-expressing HEK 293 cell membrane fraction was analyzed by modifying the methods of C. J. Langmead et al. (see Langmead C J, Szekeres P G; Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details
US Patent

TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 195671BDBM195671(US9206173, 2433)
Affinity DataKi:  5nM ΔG°:  -47.4kJ/molepH: 7.4 T: 2°CAssay Description:Receptor-expressing HEK 293 cell membrane fraction was analyzed by modifying the methods of C. J. Langmead et al. (see Langmead C J, Szekeres P G; Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details
US Patent

TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50553389BDBM50553389(CHEMBL4790047)
Affinity DataEC50:  5.10nMAssay Description:Activation of human GPR10 overexpressed in CHO-K1 cells assessed as increase in beta arrestin recruitment incubated for 90 mins by PathHunter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50553356BDBM50553356(CHEMBL4780405)
Affinity DataEC50:  5.20nMAssay Description:Activation of human GPR10 overexpressed in CHO-K1 cells assessed as increase in beta arrestin recruitment incubated for 90 mins by PathHunter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50553307BDBM50553307(CHEMBL4756913)
Affinity DataEC50:  5.90nMAssay Description:Activation of human GPR10 overexpressed in CHO-K1 cells assessed as increase in beta arrestin recruitment incubated for 90 mins by PathHunter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 195722BDBM195722(US9206173, 2484)
Affinity DataKi:  6nM ΔG°:  -46.9kJ/molepH: 7.4 T: 2°CAssay Description:Receptor-expressing HEK 293 cell membrane fraction was analyzed by modifying the methods of C. J. Langmead et al. (see Langmead C J, Szekeres P G; Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details
US Patent

TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 195753BDBM195753(US9206173, 166)
Affinity DataKi:  6nM ΔG°:  -46.9kJ/molepH: 7.4 T: 2°CAssay Description:Receptor-expressing HEK 293 cell membrane fraction was analyzed by modifying the methods of C. J. Langmead et al. (see Langmead C J, Szekeres P G; Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details
US Patent

TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 195694BDBM195694(US9206173, 2456)
Affinity DataKi:  6nM ΔG°:  -46.9kJ/molepH: 7.4 T: 2°CAssay Description:Receptor-expressing HEK 293 cell membrane fraction was analyzed by modifying the methods of C. J. Langmead et al. (see Langmead C J, Szekeres P G; Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details
US Patent

TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 195706BDBM195706(US9206173, 2468)
Affinity DataKi:  6nM ΔG°:  -46.9kJ/molepH: 7.4 T: 2°CAssay Description:Receptor-expressing HEK 293 cell membrane fraction was analyzed by modifying the methods of C. J. Langmead et al. (see Langmead C J, Szekeres P G; Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details
US Patent

TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 195640BDBM195640(US9206173, 2402)
Affinity DataKi:  6nM ΔG°:  -46.9kJ/molepH: 7.4 T: 2°CAssay Description:Receptor-expressing HEK 293 cell membrane fraction was analyzed by modifying the methods of C. J. Langmead et al. (see Langmead C J, Szekeres P G; Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details
US Patent

TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50553376BDBM50553376(CHEMBL4752167)
Affinity DataEC50:  6.10nMAssay Description:Activation of human GPR10 overexpressed in CHO-K1 cells assessed as increase in beta arrestin recruitment incubated for 90 mins by PathHunter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 195657BDBM195657(US9206173, 2419)
Affinity DataKi:  7nM ΔG°:  -46.5kJ/molepH: 7.4 T: 2°CAssay Description:Receptor-expressing HEK 293 cell membrane fraction was analyzed by modifying the methods of C. J. Langmead et al. (see Langmead C J, Szekeres P G; Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details
US Patent

TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50553346BDBM50553346(CHEMBL4782739)
Affinity DataEC50:  7.30nMAssay Description:Activation of human GPR10 overexpressed in CHO-K1 cells assessed as increase in beta arrestin recruitment incubated for 90 mins by PathHunter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50553384BDBM50553384(CHEMBL4746959)
Affinity DataEC50:  7.5nMAssay Description:Activation of human GPR10 overexpressed in CHO-K1 cells assessed as increase in beta arrestin recruitment incubated for 90 mins by PathHunter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50553310BDBM50553310(CHEMBL4792908)
Affinity DataEC50:  7.80nMAssay Description:Activation of human GPR10 overexpressed in CHO-K1 cells assessed as increase in beta arrestin recruitment incubated for 90 mins by PathHunter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 195627BDBM195627(US9206173, 2389)
Affinity DataKi:  8nM ΔG°:  -46.2kJ/molepH: 7.4 T: 2°CAssay Description:Receptor-expressing HEK 293 cell membrane fraction was analyzed by modifying the methods of C. J. Langmead et al. (see Langmead C J, Szekeres P G; Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details
US Patent

TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 195617BDBM195617(US9206173, 5)
Affinity DataKi:  8nM ΔG°:  -46.2kJ/molepH: 7.4 T: 2°CAssay Description:Receptor-expressing HEK 293 cell membrane fraction was analyzed by modifying the methods of C. J. Langmead et al. (see Langmead C J, Szekeres P G; Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details
US Patent

TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 195628BDBM195628(US9206173, 2390)
Affinity DataKi:  8nM ΔG°:  -46.2kJ/molepH: 7.4 T: 2°CAssay Description:Receptor-expressing HEK 293 cell membrane fraction was analyzed by modifying the methods of C. J. Langmead et al. (see Langmead C J, Szekeres P G; Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details
US Patent

TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50553308BDBM50553308(CHEMBL4742191)
Affinity DataEC50:  8nMAssay Description:Activation of human GPR10 overexpressed in CHO-K1 cells assessed as increase in beta arrestin recruitment incubated for 90 mins by PathHunter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 195650BDBM195650(US9206173, 2412)
Affinity DataKi:  8nM ΔG°:  -46.2kJ/molepH: 7.4 T: 2°CAssay Description:Receptor-expressing HEK 293 cell membrane fraction was analyzed by modifying the methods of C. J. Langmead et al. (see Langmead C J, Szekeres P G; Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details
US Patent

TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 195720BDBM195720(US9206173, 2482)
Affinity DataKi:  8nM ΔG°:  -46.2kJ/molepH: 7.4 T: 2°CAssay Description:Receptor-expressing HEK 293 cell membrane fraction was analyzed by modifying the methods of C. J. Langmead et al. (see Langmead C J, Szekeres P G; Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details
US Patent

TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 195645BDBM195645(US9206173, 2407)
Affinity DataKi:  8nM ΔG°:  -46.2kJ/molepH: 7.4 T: 2°CAssay Description:Receptor-expressing HEK 293 cell membrane fraction was analyzed by modifying the methods of C. J. Langmead et al. (see Langmead C J, Szekeres P G; Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details
US Patent

TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 195695BDBM195695(US9206173, 2457)
Affinity DataKi:  8nM ΔG°:  -46.2kJ/molepH: 7.4 T: 2°CAssay Description:Receptor-expressing HEK 293 cell membrane fraction was analyzed by modifying the methods of C. J. Langmead et al. (see Langmead C J, Szekeres P G; Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details
US Patent

TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 195656BDBM195656(US9206173, 2418)
Affinity DataKi:  8nM ΔG°:  -46.2kJ/molepH: 7.4 T: 2°CAssay Description:Receptor-expressing HEK 293 cell membrane fraction was analyzed by modifying the methods of C. J. Langmead et al. (see Langmead C J, Szekeres P G; Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details
US Patent

TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50553314BDBM50553314(CHEMBL4741249)
Affinity DataEC50:  8.20nMAssay Description:Activation of human GPR10 overexpressed in CHO-K1 cells assessed as increase in beta arrestin recruitment incubated for 90 mins by PathHunter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50553393BDBM50553393(CHEMBL4792592)
Affinity DataEC50:  8.80nMAssay Description:Activation of human GPR10 overexpressed in CHO-K1 cells assessed as increase in beta arrestin recruitment incubated for 90 mins by PathHunter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 195653BDBM195653(US9206173, 2415)
Affinity DataKi:  9nM ΔG°:  -45.9kJ/molepH: 7.4 T: 2°CAssay Description:Receptor-expressing HEK 293 cell membrane fraction was analyzed by modifying the methods of C. J. Langmead et al. (see Langmead C J, Szekeres P G; Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details
US Patent

TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 195716BDBM195716(US9206173, 2478)
Affinity DataKi:  9nM ΔG°:  -45.9kJ/molepH: 7.4 T: 2°CAssay Description:Receptor-expressing HEK 293 cell membrane fraction was analyzed by modifying the methods of C. J. Langmead et al. (see Langmead C J, Szekeres P G; Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details
US Patent

TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 195672BDBM195672(US9206173, 2434)
Affinity DataKi:  9nM ΔG°:  -45.9kJ/molepH: 7.4 T: 2°CAssay Description:Receptor-expressing HEK 293 cell membrane fraction was analyzed by modifying the methods of C. J. Langmead et al. (see Langmead C J, Szekeres P G; Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details
US Patent

TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 195714BDBM195714(US9206173, 2476)
Affinity DataKi:  9nM ΔG°:  -45.9kJ/molepH: 7.4 T: 2°CAssay Description:Receptor-expressing HEK 293 cell membrane fraction was analyzed by modifying the methods of C. J. Langmead et al. (see Langmead C J, Szekeres P G; Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details
US Patent

TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 195689BDBM195689(US9206173, 2451)
Affinity DataKi:  9nM ΔG°:  -45.9kJ/molepH: 7.4 T: 2°CAssay Description:Receptor-expressing HEK 293 cell membrane fraction was analyzed by modifying the methods of C. J. Langmead et al. (see Langmead C J, Szekeres P G; Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details
US Patent

TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50553312BDBM50553312(CHEMBL4745052)
Affinity DataEC50:  9nMAssay Description:Activation of human GPR10 overexpressed in CHO-K1 cells assessed as increase in beta arrestin recruitment incubated for 90 mins by PathHunter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50553308BDBM50553308(CHEMBL4742191)
Affinity DataEC50:  9.10nMAssay Description:Activation of human GPR10 overexpressed in CHO-K1 cells assessed as increase in beta arrestin recruitment incubated for 90 mins in presence of 10% FB...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 195703BDBM195703(US9206173, 2465)
Affinity DataKi:  10nM ΔG°:  -45.7kJ/molepH: 7.4 T: 2°CAssay Description:Receptor-expressing HEK 293 cell membrane fraction was analyzed by modifying the methods of C. J. Langmead et al. (see Langmead C J, Szekeres P G; Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details
US Patent

TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50553397BDBM50553397(CHEMBL4740406)
Affinity DataEC50:  10nMAssay Description:Activation of human GPR10 overexpressed in CHO-K1 cells assessed as increase in beta arrestin recruitment incubated for 90 mins by PathHunter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 195648BDBM195648(US9206173, 2410)
Affinity DataKi:  10nM ΔG°:  -45.7kJ/molepH: 7.4 T: 2°CAssay Description:Receptor-expressing HEK 293 cell membrane fraction was analyzed by modifying the methods of C. J. Langmead et al. (see Langmead C J, Szekeres P G; Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details
US Patent

TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 195697BDBM195697(US9206173, 2459)
Affinity DataKi:  10nM ΔG°:  -45.7kJ/molepH: 7.4 T: 2°CAssay Description:Receptor-expressing HEK 293 cell membrane fraction was analyzed by modifying the methods of C. J. Langmead et al. (see Langmead C J, Szekeres P G; Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details
US Patent

TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 195752BDBM195752(US9206173, 163)
Affinity DataKi:  10nM ΔG°:  -45.7kJ/molepH: 7.4 T: 2°CAssay Description:Receptor-expressing HEK 293 cell membrane fraction was analyzed by modifying the methods of C. J. Langmead et al. (see Langmead C J, Szekeres P G; Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details
US Patent

TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50553307BDBM50553307(CHEMBL4756913)
Affinity DataEC50:  10nMAssay Description:Activation of human GPR10 overexpressed in CHO-K1 cells assessed as increase in beta arrestin recruitment incubated for 90 mins in presence of 10% FB...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProlactin-releasing peptide receptor(Human)
Juvantia Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 195642BDBM195642(US9206173, 2404)
Affinity DataKi:  10nM ΔG°:  -45.7kJ/molepH: 7.4 T: 2°CAssay Description:Receptor-expressing HEK 293 cell membrane fraction was analyzed by modifying the methods of C. J. Langmead et al. (see Langmead C J, Szekeres P G; Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details
US Patent

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