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Report error Found 92 Enz. Inhib. hit(s) with all data for entry = 50016511
TargetAdenosine receptor A2b(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50150074(2-Amino-4-(4-hydroxy-phenyl)-6-(1H-imidazol-2-ylme...)
Affinity DataKi:  1nMAssay Description:Binding affinity to human wild type adenosine A2B receptor expressed in Expi293F cells assessed as inhibition constant by surface plasmon resonance a...More data for this Ligand-Target Pair
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TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM82022(2-(Phenylamino)ado (CV-1808) | 2-[6-Amino-2-(3-cyc...)
Affinity DataKi:  76nMAssay Description:Binding affinity to human wild type adenosine A2A receptor expressed in Expi293F cells assessed as inhibition constant by surface plasmon resonance a...More data for this Ligand-Target Pair
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TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM14487((2R,3R,4S,5R)-2-(6-amino-9H-purin-9-yl)-5-(hydroxy...)
Affinity DataKi:  150nMAssay Description:Binding affinity to human wild type adenosine A2A receptor expressed in Expi293F cells assessed as inhibition constant by surface plasmon resonance a...More data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM14487((2R,3R,4S,5R)-2-(6-amino-9H-purin-9-yl)-5-(hydroxy...)
Affinity DataKi:  290nMAssay Description:Binding affinity to human wild type adenosine A3 receptor expressed in Expi293F cells assessed as inhibition constant by surface plasmon resonance as...More data for this Ligand-Target Pair
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TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM21190(4-(2-{[5-amino-2-(furan-2-yl)-[1,2,4]triazolo[1,5-...)
Affinity DataKi:  395nMAssay Description:Binding affinity to human wild type adenosine A2A receptor expressed in Expi293F cells assessed as inhibition constant by surface plasmon resonance a...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM21190(4-(2-{[5-amino-2-(furan-2-yl)-[1,2,4]triazolo[1,5-...)
Affinity DataIC50:  1.5nMAssay Description:Antagonist activity at human adenosine A2A receptor expressed in HEK293T cells assessed as inhibition of NECA-induced Gs short protein activation by ...More data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 alpha(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM8392(CHEMBL408564 | N-[5-bromo-6-(furan-2-yl)-1H-pyrazo...)
Affinity DataIC50:  7nMAssay Description:Inhibition of recombinant human GSKalphaMore data for this Ligand-Target Pair
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TargetGlycogen synthase kinase-3 alpha(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM8246(3-[(3-chloro-4-hydroxyphenyl)amino]-4-(3-chlorophe...)
Affinity DataIC50:  94nMAssay Description:Inhibition of recombinant human GSKalphaMore data for this Ligand-Target Pair
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TargetGlycogen synthase kinase-3 alpha(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50595384(CHEMBL63803)
Affinity DataIC50:  100nMAssay Description:Inhibition of recombinant human GSKalphaMore data for this Ligand-Target Pair
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TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50520329(CHEMBL4550896)
Affinity DataIC50:  166nMAssay Description:Antagonist activity at human adenosine A2A receptor expressed in HEK293T cells assessed as inhibition of NECA-induced Gs short protein activation by ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM14487((2R,3R,4S,5R)-2-(6-amino-9H-purin-9-yl)-5-(hydroxy...)
Affinity DataKd:  17nMAssay Description:Binding affinity to human wild type adenosine A2A receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM21190(4-(2-{[5-amino-2-(furan-2-yl)-[1,2,4]triazolo[1,5-...)
Affinity DataKd:  286nMAssay Description:Binding affinity to human wild type adenosine A2A receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM10847(1,3-dimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-dion...)
Affinity DataKd:  3.63E+3nMAssay Description:Binding affinity to human wild type adenosine A2A receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50140241(Allopurinol | Aloral | Aluline 100 | Aluline 300 |...)
Affinity DataKd:  7.70E+4nMAssay Description:Binding affinity to human wild type adenosine A2A receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM10849(1,3,7-trimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-d...)
Affinity DataKd:  5.51E+3nMAssay Description:Binding affinity to human wild type adenosine A2A receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM82022(2-(Phenylamino)ado (CV-1808) | 2-[6-Amino-2-(3-cyc...)
Affinity DataKd:  9.10nMAssay Description:Binding affinity to human wild type adenosine A2A receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50595371(CHEMBL5193006)
Affinity DataKd:  1.39E+5nMAssay Description:Binding affinity to human wild type adenosine A2A receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance...More data for this Ligand-Target Pair
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TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM152260(US8993552, 1F4 Compound 44)
Affinity DataKd:  4.10E+5nMAssay Description:Binding affinity to human wild type adenosine A2A receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50595372(CHEMBL5195119)
Affinity DataKd:  1.00E+5nMAssay Description:Binding affinity to human wild type adenosine A2A receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50520329(CHEMBL4550896)
Affinity DataKd:  4.00E+4nMAssay Description:Binding affinity to human wild type adenosine A2A receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50207720(CHEMBL3954022)
Affinity DataKd:  1.11E+3nMAssay Description:Binding affinity to human wild type adenosine A2A receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50595373(CHEMBL5197657)
Affinity DataKd:  3.18E+4nMAssay Description:Binding affinity to human wild type adenosine A2A receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50595374(CHEMBL5197070)
Affinity DataKd:  2.10E+5nMAssay Description:Binding affinity to human wild type adenosine A2A receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50595375(CHEMBL1573515)
Affinity DataKd:  1.31E+5nMAssay Description:Binding affinity to human wild type adenosine A2A receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50595376(CHEMBL47633)
Affinity DataKd:  1.30E+5nMAssay Description:Binding affinity to human wild type adenosine A2A receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50595377(CHEMBL336555 | Pteridine-2,4-Diamine)
Affinity DataKd:  9.60E+3nMAssay Description:Binding affinity to human wild type adenosine A2A receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50595378(CHEMBL5204663)
Affinity DataKd:  2.88E+4nMAssay Description:Binding affinity to human wild type adenosine A2A receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50595379(CHEMBL5193059)
Affinity DataKd:  4.90E+4nMAssay Description:Binding affinity to human wild type adenosine A2A receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50595380(BENZOGUANAMINE)
Affinity DataKd:  1.50E+3nMAssay Description:Binding affinity to human wild type adenosine A2A receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50595381(CHEMBL5184937)
Affinity DataKd:  2.18E+4nMAssay Description:Binding affinity to human wild type adenosine A2A receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50595382(CHEMBL5208068)
Affinity DataKd:  1.35E+4nMAssay Description:Binding affinity to human wild type adenosine A2A receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50595383(CHEMBL5201800)
Affinity DataKd:  5.00E+4nMAssay Description:Binding affinity to human wild type adenosine A2A receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM6659(1-phenyl-3-pyridin-2-ylurea | Diarylurea deriv. 14...)
Affinity DataKd:  5.09E+4nMAssay Description:Binding affinity to human wild type adenosine A2A receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM8392(CHEMBL408564 | N-[5-bromo-6-(furan-2-yl)-1H-pyrazo...)
Affinity DataKd:  560nMAssay Description:Binding affinity to human wild type adenosine A2A receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM8246(3-[(3-chloro-4-hydroxyphenyl)amino]-4-(3-chlorophe...)
Affinity DataKd:  110nMAssay Description:Binding affinity to human wild type adenosine A2A receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance...More data for this Ligand-Target Pair
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TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50275499(2-(4-fluorophenyl)-3-(4-pyridinyl)pyrazolo-[1,5-a]...)
Affinity DataKd:  8.90E+3nMAssay Description:Binding affinity to human wild type adenosine A2A receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50581950(CHEMBL4204703)
Affinity DataKd:  5.5nMAssay Description:Binding affinity to human wild type adenosine A1 receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50595371(CHEMBL5193006)
Affinity DataKd:  1.22E+5nMAssay Description:Binding affinity to human wild type adenosine A1 receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM152260(US8993552, 1F4 Compound 44)
Affinity DataKd:  7.80E+4nMAssay Description:Binding affinity to human wild type adenosine A1 receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50595372(CHEMBL5195119)
Affinity DataKd:  9.20E+4nMAssay Description:Binding affinity to human wild type adenosine A1 receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A1(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50520329(CHEMBL4550896)
Affinity DataKd:  5.90E+4nMAssay Description:Binding affinity to human wild type adenosine A1 receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50207720(CHEMBL3954022)
Affinity DataKd:  2.29E+4nMAssay Description:Binding affinity to human wild type adenosine A1 receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50595374(CHEMBL5197070)
Affinity DataKd:  2.70E+4nMAssay Description:Binding affinity to human wild type adenosine A1 receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50595375(CHEMBL1573515)
Affinity DataKd:  1.54E+5nMAssay Description:Binding affinity to human wild type adenosine A1 receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50595376(CHEMBL47633)
Affinity DataKd:  5.17E+4nMAssay Description:Binding affinity to human wild type adenosine A1 receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A1(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50595378(CHEMBL5204663)
Affinity DataKd:  3.43E+4nMAssay Description:Binding affinity to human wild type adenosine A1 receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50595379(CHEMBL5193059)
Affinity DataKd:  7.00E+4nMAssay Description:Binding affinity to human wild type adenosine A1 receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50595380(BENZOGUANAMINE)
Affinity DataKd:  2.21E+3nMAssay Description:Binding affinity to human wild type adenosine A1 receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50595381(CHEMBL5184937)
Affinity DataKd:  2.07E+4nMAssay Description:Binding affinity to human wild type adenosine A1 receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A1(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50595382(CHEMBL5208068)
Affinity DataKd:  7.60E+3nMAssay Description:Binding affinity to human wild type adenosine A1 receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
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