Compile Data Set for Download or QSAR
Report error Found 262 of affinity data for UniProtKB/TrEMBL: O70526
TargetB2 bradykinin receptor(Guinea pig)
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Curated by ChEMBL
LigandPNGBDBM50419902(CHEMBL1956722)
Affinity DataKd:  0.0631nMAssay Description:Antagonist activity at guinea pig bradykinin B2 receptor in longitudinal smooth muscle assessed as inhibition of bradykinin-induced contractile respo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50036833(D-Arg-Arg-Pro-Hyp-Gly-Phe-Ser-D-Tic-Oic-Arg | CHEM...)
Affinity DataKi:  0.0800nMAssay Description:Binding affinity against [3H]bradykinin binding to bradykinin receptor B2 in guinea pig ileal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50403371(Firazyr | HOE-140 | ICATIBANT)
Affinity DataIC50: 0.0900nMAssay Description:Concentration required to inhibit specific binding of [ 3H]BK (0.06 nM) to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50403371(Firazyr | HOE-140 | ICATIBANT)
Affinity DataIC50: 0.0900nMAssay Description:Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50074978(2-[3-(4-Amino-butyl)-ureido]-N-[4-chloro-2-cyano-3...)
Affinity DataKi:  0.100nMAssay Description:Inhibition of specific binding of [3H]BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50075000((E)-N-({[4-Chloro-2-cyano-3-(2-methyl-quinolin-8-y...)
Affinity DataKi:  0.100nMAssay Description:Inhibition of specific binding of [3H]BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50036833(D-Arg-Arg-Pro-Hyp-Gly-Phe-Ser-D-Tic-Oic-Arg | CHEM...)
Affinity DataKi:  0.110nMAssay Description:Binding affinity towards bradykinin receptor B2 using [3H]bradykininMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50406750(Firazyr | HOE-140 | Icatibant)
Affinity DataKi:  0.110nMAssay Description:In vitro binding affinity against bradykinin receptor B2 from guinea pig ileum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50067317(N-({[2,4-Dichloro-3-(2-methyl-quinolin-8-yloxymeth...)
Affinity DataIC50: 0.130nMAssay Description:Concentration required to inhibit specific binding of [ 3H]BK (0.06 nM) to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50406751(CHEMBL2369941)
Affinity DataKi:  0.160nMAssay Description:In vitro binding affinity against bradykinin receptor B2 from guinea pig ileum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50067929(4-(2-{[(E)-3-(4-Dimethylcarbamoyl-phenyl)-acryloyl...)
Affinity DataIC50: 0.25nMAssay Description:Inhibition of the specific binding of [3H]BK to Bradykinin receptor B2 in guinea pig ileum membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50074986(N-(2-((4-chloro-2-cyano-3-((2-methylquinolin-8-ylo...)
Affinity DataIC50: 0.300nMAssay Description:Displacement of [3H]bradykinin from guinea pig B2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50074986(N-(2-((4-chloro-2-cyano-3-((2-methylquinolin-8-ylo...)
Affinity DataKi:  0.300nMAssay Description:Inhibition of specific binding of [3H]BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50067263(5-{2-[({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin...)
Affinity DataIC50: 0.360nMAssay Description:Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50067242(3-(6-Acetylamino-pyridin-3-yl)-N-({[3-(3-bromo-2-m...)
Affinity DataIC50: 0.380nMAssay Description:Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50121684(CHEMBL3616944)
Affinity DataKi:  0.430nMAssay Description:Displacement of [3H]BK from B2R in guinea pig ileum membranes by liquid scintillation counting in based radioligand competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2016
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50067248(5-{2-[({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin...)
Affinity DataIC50: 0.440nMAssay Description:Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50067290(5-{2-[({[2,4-Dichloro-3-(2-methyl-quinolin-8-yloxy...)
Affinity DataIC50: 0.460nMAssay Description:Displacement of [3H]BK from Bradykinin B2 Receptor in guinea pig ileum by liquid scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50067301(FK-3657 | (E)-3-(6-Acetylamino-pyridin-3-yl)-N-({[...)
Affinity DataIC50: 0.460nMAssay Description:Inhibition of the specific binding of [3H]BK to Bradykinin receptor B2 in guinea pig ileum membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50067301(FK-3657 | (E)-3-(6-Acetylamino-pyridin-3-yl)-N-({[...)
Affinity DataIC50: 0.460nMAssay Description:Concentration required to inhibit specific binding of [ 3H]BK (0.06 nM) to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50067305((E)-N-({[2,4-Dimethyl-3-(2-methyl-quinolin-8-yloxy...)
Affinity DataIC50: 0.470nMAssay Description:Concentration required to inhibit specific binding of [ 3H]BK (0.06 nM) to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50067247(4-{(E)-2-[({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyr...)
Affinity DataIC50: 0.5nMAssay Description:Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50067283((E)-3-(4-Acetylamino-phenyl)-N-({[2,4-dichloro-3-(...)
Affinity DataIC50: 0.5nMAssay Description:Concentration required to inhibit specific binding of [ 3H]BK (0.06 nM) to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50067247(4-{(E)-2-[({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyr...)
Affinity DataIC50: 0.5nMAssay Description:Concentration required to inhibit specific binding of [ 3H]BK (0.06 nM) to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50067281(CHEMBL439737 | CHEMBL542096 | 4-{(E)-2-[({[2,4-Dic...)
Affinity DataIC50: 0.510nMAssay Description:Inhibition of the specific binding of [3H]BK to Bradykinin receptor B2 in guinea pig ileum membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50067281(CHEMBL439737 | CHEMBL542096 | 4-{(E)-2-[({[2,4-Dic...)
Affinity DataIC50: 0.510nMAssay Description:Concentration required to inhibit specific binding of [ 3H]BK (0.06 nM) to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50045210(D-Arg-Arg-Pro-Hyp-Calpha-methylGly-Calpha-methylPh...)
Affinity DataKi:  0.540nMAssay Description:Binding affinity against [3H]bradykinin binding to bradykinin receptor B2 in guinea pig ileal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50067274((E)-N-({[2,4-Dichloro-3-(2-methyl-quinolin-8-yloxy...)
Affinity DataIC50: 0.550nMAssay Description:Concentration required to inhibit specific binding of [ 3H]BK (0.06 nM) to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50067253((E)-3-(4-Acetylamino-phenyl)-N-({[3-(3-bromo-2-met...)
Affinity DataIC50: 0.550nMAssay Description:Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50067932((E)-N-({Methyl-[3-(2-methyl-quinolin-8-yloxymethyl...)
Affinity DataIC50: 0.550nMAssay Description:Inhibition of the specific binding of [3H]BK to Bradykinin receptor B2 in guinea pig ileum membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50067923(3-(6-Acetylamino-pyridin-3-yl)-N-{1-[2,4-bis-acety...)
Affinity DataIC50: 0.560nMAssay Description:Inhibition of the specific binding of [3H]BK to Bradykinin receptor B2 in guinea pig ileum membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50067917((E)-N-{1-[3-(2-Methyl-quinolin-8-yloxymethyl)-2,4-...)
Affinity DataIC50: 0.580nMAssay Description:Inhibition of the specific binding of [3H]BK to Bradykinin receptor B2 in guinea pig ileum membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50067240((E)-N-({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin...)
Affinity DataIC50: 0.590nMAssay Description:Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50074997((E)-3-(6-Acetylamino-pyridin-3-yl)-N-({[4-methoxy-...)
Affinity DataKi:  0.600nMAssay Description:Inhibition of specific binding of [3H]BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50067294(4-{2-[({[2,4-Dichloro-3-(2-methyl-quinolin-8-yloxy...)
Affinity DataIC50: 0.620nMAssay Description:Concentration required to inhibit specific binding of [ 3H]BK (0.06 nM) to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50067930(4-[(E)-2-({1-[2,4-Dichloro-3-(2-methyl-quinolin-8-...)
Affinity DataIC50: 0.640nMAssay Description:Inhibition of the specific binding of [3H]BK to Bradykinin receptor B2 in guinea pig ileum membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50067289((E)-3-(6-Acetylamino-pyridin-3-yl)-N-({[2,4-dichlo...)
Affinity DataIC50: 0.650nMAssay Description:Concentration required to inhibit specific binding of [ 3H]BK (0.06 nM) to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50067251(4-{(E)-2-[({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyr...)
Affinity DataIC50: 0.660nMAssay Description:Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50067251(4-{(E)-2-[({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyr...)
Affinity DataIC50: 0.660nMAssay Description:Concentration required to inhibit specific binding of [ 3H]BK (0.06 nM) to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50067290(5-{2-[({[2,4-Dichloro-3-(2-methyl-quinolin-8-yloxy...)
Affinity DataIC50: 0.680nMAssay Description:Concentration required to inhibit specific binding of [ 3H]BK (0.06 nM) to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50067922(N*1*,N*3*-Dimethyl-4-(methyl-{2-[3-(6-methylcarbam...)
Affinity DataIC50: 0.680nMAssay Description:Inhibition of the specific binding of [3H]BK to Bradykinin receptor B2 in guinea pig ileum membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50067308((E)-N-({[2,4-Dichloro-3-(2-methyl-quinolin-8-yloxy...)
Affinity DataIC50: 0.690nMAssay Description:Concentration required to inhibit specific binding of [ 3H]BK (0.06 nM) to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50075000((E)-N-({[4-Chloro-2-cyano-3-(2-methyl-quinolin-8-y...)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50406749(CHEMBL2028979)
Affinity DataKi:  0.75nMAssay Description:In vitro binding affinity against bradykinin receptor B2 from guinea pig ileum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50067915((E)-N-({Methyl-[3-(2-methyl-quinolin-8-yloxymethyl...)
Affinity DataIC50: 0.760nMAssay Description:Inhibition of the specific binding of [3H]BK to Bradykinin receptor B2 in guinea pig ileum membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50067296((E)-N-({[2,4-Dichloro-3-(2-methyl-quinolin-8-yloxy...)
Affinity DataIC50: 0.760nMAssay Description:Concentration required to inhibit specific binding of [ 3H]BK (0.06 nM) to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50067257(3-[3-({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin-...)
Affinity DataIC50: 0.760nMAssay Description:Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50067264((Z)-N-({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin...)
Affinity DataIC50: 0.780nMAssay Description:Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50067280(N-({[2,4-Dichloro-3-(2-methyl-quinolin-8-yloxymeth...)
Affinity DataIC50: 0.790nMAssay Description:Concentration required to inhibit specific binding of [ 3H]BK (0.06 nM) to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50067235(3-[3-({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin-...)
Affinity DataIC50: 0.790nMAssay Description:Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
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