Compile Data Set for Download or QSAR
Report error Found 1120 of affinity data for UniProtKB/TrEMBL: P30969
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50105862(pGlu-His-Trp-Ser-Tyr-D-Lys(2-(hydroxymethyl)anthra...)
Affinity DataIC50: 0.00200nMAssay Description:Evaluated for gonadotropin-releasing hormone receptor binding by displacing the 50% of the bound tracer [125I][D-Lys6]-GnRH radioligand in rat pituit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50470113(CHEMBL439134)
Affinity DataKi:  0.00200nMAssay Description:Inhibition of the in vitro binding of [125I]-labeled leuprolide to the rat pituitary luteinizing hormone releasing hormone (LHRH) receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50470098(CHEMBL2371296)
Affinity DataKi:  0.0100nMAssay Description:Inhibition of the in vitro binding of [125I]-labeled leuprolide to the rat pituitary luteinizing hormone releasing hormone (LHRH) receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50470117(CHEMBL264989)
Affinity DataKi:  0.0120nMAssay Description:Inhibition of the in vitro binding of [125I]-labeled leuprolide to the rat pituitary luteinizing hormone releasing hormone (LHRH) receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50469862(CHEMBL409219)
Affinity DataKi:  0.0135nMAssay Description:The negative logarithm of the concentration of antagonist that inhibits 50% of the binding of 125 I-labeled leuprolide to the rat pituitary LHRH rece...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50470118(CHEMBL412751)
Affinity DataKi:  0.0160nMAssay Description:Inhibition of the in vitro binding of [125I]-labeled leuprolide to the rat pituitary luteinizing hormone releasing hormone (LHRH) receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50470097(CHEMBL262235)
Affinity DataKi:  0.0170nMAssay Description:Inhibition of the in vitro binding of [125I]-labeled leuprolide to the rat pituitary luteinizing hormone releasing hormone (LHRH) receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50470082(CHEMBL408861)
Affinity DataKi:  0.0170nMAssay Description:Inhibition of the in vitro binding of [125I]-labeled leuprolide to the rat pituitary luteinizing hormone releasing hormone (LHRH) receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50470080(CHEMBL266475)
Affinity DataKi:  0.0170nMAssay Description:Inhibition of the in vitro binding of [125I]-labeled leuprolide to the rat pituitary luteinizing hormone releasing hormone (LHRH) receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50470086(CHEMBL2369140)
Affinity DataKi:  0.0180nMAssay Description:Inhibition of the in vitro binding of [125I]-labeled leuprolide to the rat pituitary luteinizing hormone releasing hormone (LHRH) receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50470099(CHEMBL2371295)
Affinity DataKi:  0.0180nMAssay Description:Inhibition of the in vitro binding of [125I]-labeled leuprolide to the rat pituitary luteinizing hormone releasing hormone (LHRH) receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50470085(CHEMBL438195)
Affinity DataKi:  0.0200nMAssay Description:Inhibition of the in vitro binding of [125I]-labeled leuprolide to the rat pituitary luteinizing hormone releasing hormone (LHRH) receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50470083(CHEMBL267709)
Affinity DataKi:  0.0200nMAssay Description:Inhibition of the in vitro binding of [125I]-labeled leuprolide to the rat pituitary luteinizing hormone releasing hormone (LHRH) receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50470084(CHEMBL428299)
Affinity DataKi:  0.0200nMAssay Description:Inhibition of the in vitro binding of [125I]-labeled leuprolide to the rat pituitary luteinizing hormone releasing hormone (LHRH) receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50470106(CHEMBL413660)
Affinity DataKi:  0.0220nMAssay Description:Inhibition of the in vitro binding of [125I]-labeled leuprolide to the rat pituitary luteinizing hormone releasing hormone (LHRH) receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50470105(CHEMBL405993)
Affinity DataKi:  0.0230nMAssay Description:Inhibition of the in vitro binding of [125I]-labeled leuprolide to the rat pituitary luteinizing hormone releasing hormone (LHRH) receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50469858(CHEMBL268397)
Affinity DataKi:  0.0234nMAssay Description:The negative logarithm of the concentration of antagonist that inhibits 50% of the binding of 125 I-labeled leuprolide to the rat pituitary LHRH rece...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50470132(CHEMBL2370208)
Affinity DataKi:  0.0250nMAssay Description:Inhibition of the in vitro binding of [125I]-labeled leuprolide to the rat pituitary luteinizing hormone releasing hormone (LHRH) receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50470101(CHEMBL406887)
Affinity DataKi:  0.0260nMAssay Description:Inhibition of the in vitro binding of [125I]-labeled leuprolide to the rat pituitary luteinizing hormone releasing hormone (LHRH) receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50470127(CHEMBL2369141)
Affinity DataKi:  0.0290nMAssay Description:Inhibition of the in vitro binding of [125I]-labeled leuprolide to the rat pituitary luteinizing hormone releasing hormone (LHRH) receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50469859(CHEMBL263839 | A-75998)
Affinity DataKi:  0.0316nMAssay Description:The negative logarithm of the concentration of antagonist that inhibits 50% of the binding of 125 I-labeled leuprolide to the rat pituitary LHRH rece...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50470121(CHEMBL268173)
Affinity DataKi:  0.0320nMAssay Description:Inhibition of the in vitro binding of [125I]-labeled leuprolide to the rat pituitary luteinizing hormone releasing hormone (LHRH) receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50470124(CHEMBL437632)
Affinity DataKi:  0.0330nMAssay Description:Inhibition of the in vitro binding of [125I]-labeled leuprolide to the rat pituitary luteinizing hormone releasing hormone (LHRH) receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50470079(CHEMBL445681)
Affinity DataKi:  0.0330nMAssay Description:Inhibition of the in vitro binding of [125I]-labeled leuprolide to the rat pituitary luteinizing hormone releasing hormone (LHRH) receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50469856(CHEMBL263840 | ORG-30850)
Affinity DataKi:  0.0331nMAssay Description:The negative logarithm of the concentration of antagonist that inhibits 50% of the binding of 125 I-labeled leuprolide to the rat pituitary LHRH rece...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50470107(CHEMBL2371292)
Affinity DataKi:  0.0380nMAssay Description:Inhibition of the in vitro binding of [125I]-labeled leuprolide to the rat pituitary luteinizing hormone releasing hormone (LHRH) receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50470122(CHEMBL265538)
Affinity DataKi:  0.0390nMAssay Description:Inhibition of the in vitro binding of [125I]-labeled leuprolide to the rat pituitary luteinizing hormone releasing hormone (LHRH) receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50470103(CHEMBL384341)
Affinity DataKi:  0.0400nMAssay Description:Inhibition of the in vitro binding of [125I]-labeled leuprolide to the rat pituitary luteinizing hormone releasing hormone (LHRH) receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50470130(CHEMBL217175)
Affinity DataKi:  0.0480nMAssay Description:Inhibition of the in vitro binding of [125I]-labeled leuprolide to the rat pituitary luteinizing hormone releasing hormone (LHRH) receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50470078(CHEMBL413393)
Affinity DataKi:  0.0520nMAssay Description:Inhibition of the in vitro binding of [125I]-labeled leuprolide to the rat pituitary luteinizing hormone releasing hormone (LHRH) receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50470089(CHEMBL429365)
Affinity DataKi:  0.0520nMAssay Description:Inhibition of the in vitro binding of [125I]-labeled leuprolide to the rat pituitary luteinizing hormone releasing hormone (LHRH) receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50470092(CHEMBL428138)
Affinity DataKi:  0.0520nMAssay Description:Inhibition of the in vitro binding of [125I]-labeled leuprolide to the rat pituitary luteinizing hormone releasing hormone (LHRH) receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50469857(CHEMBL268319)
Affinity DataKi:  0.0525nMAssay Description:The negative logarithm of the concentration of antagonist that inhibits 50% of the binding of 125 I-labeled leuprolide to the rat pituitary LHRH rece...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50470081(CHEMBL267843)
Affinity DataKi:  0.0560nMAssay Description:Inhibition of the in vitro binding of [125I]-labeled leuprolide to the rat pituitary luteinizing hormone releasing hormone (LHRH) receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50060785([D or LAgl (hydroxyacetic acid)4]acyline | CHEMBL2...)
Affinity DataIC50: 0.0560nMAssay Description:Inhibition of binding of radiolabeled histrelin to Gonadotropin-releasing hormone receptor (GnRHr) in rat pituitary gland membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50470120(CHEMBL405994)
Affinity DataKi:  0.0580nMAssay Description:Inhibition of the in vitro binding of [125I]-labeled leuprolide to the rat pituitary luteinizing hormone releasing hormone (LHRH) receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50469860(CHEMBL409990)
Affinity DataKi:  0.0617nMAssay Description:The negative logarithm of the concentration of antagonist that inhibits 50% of the binding of 125 I-labeled leuprolide to the rat pituitary LHRH rece...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50470119(CHEMBL383952)
Affinity DataKi:  0.0710nMAssay Description:Inhibition of the in vitro binding of [125I]-labeled leuprolide to the rat pituitary luteinizing hormone releasing hormone (LHRH) receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50470087(CHEMBL428093)
Affinity DataKi:  0.0760nMAssay Description:Inhibition of the in vitro binding of [125I]-labeled leuprolide to the rat pituitary luteinizing hormone releasing hormone (LHRH) receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50470114(CHEMBL268620)
Affinity DataKi:  0.0760nMAssay Description:Inhibition of the in vitro binding of [125I]-labeled leuprolide to the rat pituitary luteinizing hormone releasing hormone (LHRH) receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50470096(CHEMBL2369142)
Affinity DataKi:  0.0760nMAssay Description:Inhibition of the in vitro binding of [125I]-labeled leuprolide to the rat pituitary luteinizing hormone releasing hormone (LHRH) receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50470088(CHEMBL278704)
Affinity DataKi:  0.0780nMAssay Description:Inhibition of the in vitro binding of [125I]-labeled leuprolide to the rat pituitary luteinizing hormone releasing hormone (LHRH) receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50105860(pGlu-His-Trp-Ser-Tyr-D-Lys-Leu-Arg-Pro-Gly-NH2([D-...)
Affinity DataIC50: 0.0800nMAssay Description:Evaluated for gonadotropin-releasing hormone receptor binding by displacing the 50% of the bound tracer [125I][D-Lys6]-GnRH radioligand in rat pituit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50007953(CHEMBL414113 | pGlu-His-DPal-Ser-Tyr-DPal-Leu-ILys...)
Affinity DataKd:  0.0800nMAssay Description:In vitro binding affinity of Gonadotropin-releasing hormone antagonist was measured in rat pituitary cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50470123(CHEMBL415643)
Affinity DataKi:  0.0850nMAssay Description:Inhibition of the in vitro binding of [125I]-labeled leuprolide to the rat pituitary luteinizing hormone releasing hormone (LHRH) receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50470095(CHEMBL216589)
Affinity DataKi:  0.0890nMAssay Description:Inhibition of the in vitro binding of [125I]-labeled leuprolide to the rat pituitary luteinizing hormone releasing hormone (LHRH) receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50105861(pGlu-His-Trp-Ser-Tyr-D-Lys(N-(2 chloro-1,4-naphtho...)
Affinity DataIC50: 0.0900nMAssay Description:Evaluated for gonadotropin-releasing hormone receptor binding by displacing the 50% of the bound tracer [125I][D-Lys6]-GnRH radioligand in rat pituit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50101189(N-{4-[4-(2-{2-(3,5-Dimethyl-phenyl)-5-[2-(2,5-dime...)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of [125I]buserelin binding to rat pituitary Gonadotropin-releasing hormone receptor, in the presence of 0.1% bovine serum albumin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50101187(2-(2-(3,5-Dimethyl-phenyl)-3-{2-[4-(4-methanesulfo...)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of [125I]buserelin binding to rat pituitary Gonadotropin-releasing hormone receptor, in the presence of 0.1% bovine serum albumin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50085734(DiCyclo (4-10/5,5'-8) [Ac-D Nal, D Cpa, D Pal, Asp...)
Affinity DataKi:  0.100nMAssay Description:Competitive radioligand binding assay, in human HEK293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Displayed 1 to 50 (of 1120 total ) | Next | Last >>
Jump to: