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TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50044777(CHEBI:34543 | Arginine Vasopressin | Beta-Hypopham...)
Affinity DataEC50:  0.00350nMAssay Description:Agonist activity at recombinant human V1b receptor expressed in HEK293 cells assessed as increase in intracellular calcium level measured at 3 secs i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50345133((S)-1-((R)-5-chloro-3-(2-methoxy-5-(pyrrolidin-1-y...)
Affinity DataKi:  0.0300nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50345134((S)-1-((R)-5-chloro-3-(2-methoxy-5-((4-methylpiper...)
Affinity DataKi:  0.0300nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50345131((S)-1-((R)-5-chloro-3-(2-methoxy-4-((4-methylpiper...)
Affinity DataKi:  0.0400nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50345130((S)-1-((R)-5-chloro-3-(2-methoxy-4-(pyrrolidin-1-y...)
Affinity DataKi:  0.0800nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM260242(US9522914, A-44)
Affinity DataIC50: 0.160nMpH: 7.4 T: 2°CAssay Description:Human V1b receptor was transiently expressed in 293FT cells (Invitrogen). The cells were collected and then homogenated in a 15 mmol/L tris-hydrochlo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2017
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM260242(US9522914, A-44)
Affinity DataIC50: 0.160nMpH: 7.4 T: 2°CAssay Description:Human V1b receptor was transiently expressed in 293FT cells (Invitrogen). The cells were collected and then homogenated in a 15 mmol/L tris-hydrochlo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at human V1B receptor expressed in HEK293 cells assessed as intracellular calcium level measured at 3 secs interval for 5 mins by fu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50145126((2S)-2-{[(2R)-1-{[(4S,7R,10S,13R,16S)-13-benzyl-7-...)
Affinity DataKi:  0.230nMAssay Description:Binding affinity against human vasopressin V1b receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataEC50:  0.240nMAssay Description:Agonist activity at recombinant human V1b receptor expressed in HEK293 cells assessed as increase in intracellular calcium level measured at 3 secs i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50345132((S)-1-((R)-5-chloro-1-(2,4-dimethoxyphenylsulfonyl...)
Affinity DataKi:  0.260nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50145118(d[Val4]AVP | CHEMBL412353)
Affinity DataKi:  0.290nMAssay Description:Binding affinity against human vasopressin V1b receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50145112((2S)-2-{[(2R)-1-{[(4S,7R,13R,16S)-13-benzyl-7-(car...)
Affinity DataKi:  0.370nMAssay Description:Binding affinity against human vasopressin V1b receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50370387(CHEMBL1790575)
Affinity DataKi:  0.420nMAssay Description:Binding affinity against human vasopressin V1b receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM260267(US9522914, B-20)
Affinity DataIC50: 0.430nMpH: 7.4 T: 2°CAssay Description:Human V1b receptor was transiently expressed in 293FT cells (Invitrogen). The cells were collected and then homogenated in a 15 mmol/L tris-hydrochlo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2017
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM260267(US9522914, B-20)
Affinity DataIC50: 0.430nMpH: 7.4 T: 2°CAssay Description:Human V1b receptor was transiently expressed in 293FT cells (Invitrogen). The cells were collected and then homogenated in a 15 mmol/L tris-hydrochlo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50145124((2S)-2-{[(2R)-1-{[(4S,7R,13R,16S)-13-benzyl-10-but...)
Affinity DataKi:  0.430nMAssay Description:Binding affinity against human vasopressin V1b receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50145107((2S)-2-{[(2R)-1-{[(4S,7R,13R,16S)-10-(3-aminopropy...)
Affinity DataKi:  0.490nMAssay Description:Binding affinity against human vasopressin V1b receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM260241(US9522914, A-43)
Affinity DataIC50: 0.490nMpH: 7.4 T: 2°CAssay Description:Human V1b receptor was transiently expressed in 293FT cells (Invitrogen). The cells were collected and then homogenated in a 15 mmol/L tris-hydrochlo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2017
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM260241(US9522914, A-43)
Affinity DataIC50: 0.490nMpH: 7.4 T: 2°CAssay Description:Human V1b receptor was transiently expressed in 293FT cells (Invitrogen). The cells were collected and then homogenated in a 15 mmol/L tris-hydrochlo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM35667([3H]Argipressin tannate | AVP | [3H]Arginine vasop...)
Affinity DataKi:  0.490nMAssay Description:Displacement of [3H]-AVP from human vasopressin V1b receptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50523555(CHEMBL4474284)
Affinity DataEC50:  0.5nMAssay Description:Agonist activity at recombinant human V1b receptor expressed in HEK293 cells assessed as increase in intracellular calcium level measured at 3 secs i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50342028(2-((S)-6-amino-2-((S)-1-((4R,7S,10S,13S,16S)-7-(2-...)
Affinity DataKi:  0.520nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed CHO cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50145117((2S)-2-{[(2R)-1-{[(4S,7R,13R,16S)-13-benzyl-7-(car...)
Affinity DataKi:  0.520nMAssay Description:Binding affinity against human vasopressin V1b receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM35667([3H]Argipressin tannate | AVP | [3H]Arginine vasop...)
Affinity DataKi:  0.590nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details
PubMed
TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50299343(SSR149415 | (2S,4R)-1-[5-Chloro-1-[(2,4-dimethoxyp...)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]Arg8-vasopressin from human vasopressin V1b receptor expressed in CHO-K1 cells by Packard Topcount scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50299343(SSR149415 | (2S,4R)-1-[5-Chloro-1-[(2,4-dimethoxyp...)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells by whole cell binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50342032(2-((S)-2-((S)-1-((4R,7S,10S,13S,16S)-7-(2-amino-2-...)
Affinity DataKi:  0.610nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed CHO cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM260347(US9522914, D-36)
Affinity DataIC50: 0.610nMpH: 7.4 T: 2°CAssay Description:Human V1b receptor was transiently expressed in 293FT cells (Invitrogen). The cells were collected and then homogenated in a 15 mmol/L tris-hydrochlo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2017
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM260347(US9522914, D-36)
Affinity DataIC50: 0.610nMpH: 7.4 T: 2°CAssay Description:Human V1b receptor was transiently expressed in 293FT cells (Invitrogen). The cells were collected and then homogenated in a 15 mmol/L tris-hydrochlo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50342029(2-((S)-2-((S)-1-((4R,7S,10S,13S,16S)-7-(2-amino-2-...)
Affinity DataKi:  0.650nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed CHO cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50299343(SSR149415 | (2S,4R)-1-[5-Chloro-1-[(2,4-dimethoxyp...)
Affinity DataKi:  0.740nMAssay Description:Test compounds were tested for binding to the V1b human vasopressin receptor using a human V1b (agonist radioligand) Receptor Binding Assay, with the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2025
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50145108((2S)-2-{[(2R)-1-{[(4S,7R,13R,16S)-13-benzyl-7-(car...)
Affinity DataKi:  0.780nMAssay Description:Binding affinity against human vasopressin V1b receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50523556(CHEMBL4458988)
Affinity DataEC50:  0.800nMAssay Description:Agonist activity at recombinant human V1b receptor expressed in HEK293 cells assessed as increase in intracellular calcium level measured at 3 secs i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50345129((S)-1-((R)-5-chloro-1-(2,4-dimethoxyphenylsulfonyl...)
Affinity DataKi:  0.810nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM260206(US9522914, A-08)
Affinity DataIC50: 0.820nMpH: 7.4 T: 2°CAssay Description:Human V1b receptor was transiently expressed in 293FT cells (Invitrogen). The cells were collected and then homogenated in a 15 mmol/L tris-hydrochlo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2017
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM260206(US9522914, A-08)
Affinity DataIC50: 0.820nMpH: 7.4 T: 2°CAssay Description:Human V1b receptor was transiently expressed in 293FT cells (Invitrogen). The cells were collected and then homogenated in a 15 mmol/L tris-hydrochlo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM716486(US20250034117, Compound Example 2)
Affinity DataKi:  0.960nMAssay Description:Test compounds were tested for binding to the V1b human vasopressin receptor using a human V1b (agonist radioligand) Receptor Binding Assay, with the...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2025
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM717676(US20250034117, Example 3)
Affinity DataKi:  0.980nMAssay Description:Test compounds were tested for binding to the V1b human vasopressin receptor using a human V1b (agonist radioligand) Receptor Binding Assay, with the...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2025
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50345056(2-(6-(3-((dimethylamino)methyl)phenyl)-2-(4-fluoro...)
Affinity DataIC50: 1nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM175039(US9688678, 11 (+)-3-(2-ethoxy-5-methoxyphenyl)-1-(...)
Affinity DataKi: <1nM ΔG°: <-51.4kJ/molepH: 7.4 T: 2°CAssay Description:The binding assay was carried out by the method based on that of Tahara et al. (Tahara A et al., Brit. J. Pharmacol. 125, 1463-1470 (1998)). The incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2018
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM175037(US9688678, 9A (+)-3-(2-ethoxy-3-pyridyl)-1-[(5-met...)
Affinity DataKi: <1nM ΔG°: <-51.4kJ/molepH: 7.4 T: 2°CAssay Description:The binding assay was carried out by the method based on that of Tahara et al. (Tahara A et al., Brit. J. Pharmacol. 125, 1463-1470 (1998)). The incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2018
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM260237(US9522914, A-39)
Affinity DataIC50: 1nMpH: 7.4 T: 2°CAssay Description:Human V1b receptor was transiently expressed in 293FT cells (Invitrogen). The cells were collected and then homogenated in a 15 mmol/L tris-hydrochlo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM175060(US9688678, 21 (+-)-3-(2,5-dimethoxyphenyl)-1-[(5-m...)
Affinity DataKi: <1nM ΔG°: <-51.4kJ/molepH: 7.4 T: 2°CAssay Description:The binding assay was carried out by the method based on that of Tahara et al. (Tahara A et al., Brit. J. Pharmacol. 125, 1463-1470 (1998)). The incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2018
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM175058(US9688678, 19 (+-)-3-(2-ethoxy-5-methoxy-phenyl)-3...)
Affinity DataKi: <1nM ΔG°: <-51.4kJ/molepH: 7.4 T: 2°CAssay Description:The binding assay was carried out by the method based on that of Tahara et al. (Tahara A et al., Brit. J. Pharmacol. 125, 1463-1470 (1998)). The incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2018
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM175057(US9688678, 18A (+)-3-(2-methoxyphenyl)-1-[(5-metho...)
Affinity DataKi: <1nM ΔG°: <-51.4kJ/molepH: 7.4 T: 2°CAssay Description:The binding assay was carried out by the method based on that of Tahara et al. (Tahara A et al., Brit. J. Pharmacol. 125, 1463-1470 (1998)). The incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2018
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM175056(US9688678, 18 (+-)3-(2-methoxyphenyl)-1-[(5-methox...)
Affinity DataKi: <1nM ΔG°: <-51.4kJ/molepH: 7.4 T: 2°CAssay Description:The binding assay was carried out by the method based on that of Tahara et al. (Tahara A et al., Brit. J. Pharmacol. 125, 1463-1470 (1998)). The incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2018
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM175055(US9688678, 17B (+)-3-(2-ethoxy-5-methoxy-phenyl)-1...)
Affinity DataKi: <1nM ΔG°: <-51.4kJ/molepH: 7.4 T: 2°CAssay Description:The binding assay was carried out by the method based on that of Tahara et al. (Tahara A et al., Brit. J. Pharmacol. 125, 1463-1470 (1998)). The incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2018
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM175054(US9688678, 17 (+-)-3-(2-ethoxy-5-methoxy-phenyl)-1...)
Affinity DataKi: <1nM ΔG°: <-51.4kJ/molepH: 7.4 T: 2°CAssay Description:The binding assay was carried out by the method based on that of Tahara et al. (Tahara A et al., Brit. J. Pharmacol. 125, 1463-1470 (1998)). The incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2018
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM175064(US9688678, 25 (+)-3-(2-ethoxy-5-methoxy-phenyl)-1-...)
Affinity DataKi: <1nM ΔG°: <-51.4kJ/molepH: 7.4 T: 2°CAssay Description:The binding assay was carried out by the method based on that of Tahara et al. (Tahara A et al., Brit. J. Pharmacol. 125, 1463-1470 (1998)). The incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2018
Entry Details
US Patent

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