Compile Data Set for Download or QSAR
Report error Found 1190 of affinity data for UniProtKB/TrEMBL: Q5L478
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50458018BDBM50458018(CHEMBL4216436)
Affinity DataEC50:  0.000100nMAssay Description:Inhibition of NS5A in HCV genotype 4a infected in human HuH7 replicon cells expressing HCV genotype 1b chimeric replicon assessed as reduction in vir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50458023BDBM50458023(CHEMBL4214282)
Affinity DataEC50:  0.000100nMAssay Description:Inhibition of NS5A in HCV genotype 4a infected in human HuH7 replicon cells expressing HCV genotype 1b chimeric replicon assessed as reduction in vir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50458020BDBM50458020(CHEMBL4203791)
Affinity DataEC50:  0.000100nMAssay Description:Inhibition of NS5A in HCV genotype 4a infected in human HuH7 replicon cells expressing HCV genotype 1b chimeric replicon assessed as reduction in vir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50453112BDBM50453112(CHEBI:85183 | ABT-267 | Ombitasvir)
Affinity DataEC50:  0.000300nMAssay Description:Inhibition of NS5A in HCV genotype 4a infected in human HuH7 replicon cells expressing HCV genotype 1b chimeric replicon assessed as reduction in vir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50453103BDBM50453103(CHEMBL4218872)
Affinity DataEC50:  0.00100nMAssay Description:Inhibition of NS5A in HuH7 cell infected HCV genotype 1a H77 assessed as decrease in viral replication after 3 days by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595029BDBM50595029(CHEMBL5191072)
Affinity DataEC50:  0.00100nMAssay Description:Inhibition of HCV genotype 4a NS5AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595029BDBM50595029(CHEMBL5191072)
Affinity DataEC50:  0.00100nMAssay Description:Inhibition of HCV genotype 6a NS5AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50547638BDBM50547638(CHEMBL4782728)
Affinity DataIC50: 0.00100nMAssay Description:Inhibition of HCV genotype 1b NS5A infected in Huh7 cells assessed as reduction in viral replication incubated 3 days and measured by Celltiter Glo a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50458018BDBM50458018(CHEMBL4216436)
Affinity DataEC50:  0.00100nMAssay Description:Inhibition of NS5A in HCV genotype 5a infected in human HuH7 replicon cells expressing HCV genotype 1b chimeric replicon assessed as reduction in vir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50547628BDBM50547628(CHEMBL4753603)
Affinity DataIC50: 0.00100nMAssay Description:Inhibition of HCV genotype 2a NS5A infected in Huh7 cells assessed as reduction in viral replication incubated 3 days and measured by bright Glo-luci...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50547630BDBM50547630(CHEMBL4758660)
Affinity DataIC50: 0.00100nMAssay Description:Inhibition of HCV genotype 1b NS5A infected in Huh7 cells assessed as reduction in viral replication incubated 3 days and measured by Celltiter Glo a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50547646BDBM50547646(CHEMBL4780371)
Affinity DataIC50: 0.00100nMAssay Description:Inhibition of HCV genotype 1b NS5A infected in Huh7 cells assessed as reduction in viral replication incubated 3 days and measured by Celltiter Glo a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50458020BDBM50458020(CHEMBL4203791)
Affinity DataEC50:  0.00100nMAssay Description:Inhibition of NS5A in HCV genotype 5a infected in human HuH7 replicon cells expressing HCV genotype 1b chimeric replicon assessed as reduction in vir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50458023BDBM50458023(CHEMBL4214282)
Affinity DataEC50:  0.00100nMAssay Description:Inhibition of NS5A in HCV genotype 5a infected in human HuH7 replicon cells expressing HCV genotype 1b chimeric replicon assessed as reduction in vir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50547634BDBM50547634(CHEMBL4747100)
Affinity DataIC50: 0.00100nMAssay Description:Inhibition of HCV genotype 1b NS5A infected in Huh7 cells assessed as reduction in viral replication incubated 3 days and measured by Celltiter Glo a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50453109BDBM50453109(CHEMBL4205352)
Affinity DataEC50:  0.00100nMAssay Description:Inhibition of NS5A in HuH7 cell infected HCV genotype 1a H77 assessed as decrease in viral replication after 3 days by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595029BDBM50595029(CHEMBL5191072)
Affinity DataEC50:  0.00100nMAssay Description:Inhibition of HCV genotype 1a NS5AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595029BDBM50595029(CHEMBL5191072)
Affinity DataEC50:  0.00100nMAssay Description:Inhibition of HCV genotype 2a NS5AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531965BDBM50531965(CHEMBL4542548)
Affinity DataEC50:  0.00160nMAssay Description:Inhibition of NS5A in HCV genotype 1b assessed as decrease in viral replicationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50453100BDBM50453100(A-1325912.0 | ABT-530 | Pibrentasvir)
Affinity DataEC50:  0.00180nMAssay Description:Inhibition of NS5A in HuH7 cell infected HCV genotype 1a H77 assessed as decrease in viral replication after 3 days by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531953BDBM50531953(CHEMBL3360472)
Affinity DataEC50:  0.00200nMAssay Description:Inhibition of NS5A in HCV genotype 1b assessed as decrease in viral replicationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595029BDBM50595029(CHEMBL5191072)
Affinity DataEC50:  0.00200nMAssay Description:Inhibition of HCV genotype 5a NS5AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50547627BDBM50547627(CHEMBL4755593)
Affinity DataIC50: 0.00200nMAssay Description:Inhibition of HCV genotype 1b NS5A infected in Huh7 cells assessed as reduction in viral replication incubated 3 days and measured by Celltiter Glo a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50453117BDBM50453117(CHEMBL4211486)
Affinity DataEC50:  0.00200nMAssay Description:Inhibition of NS5A in HuH7 cell infected HCV genotype 1a H77 assessed as decrease in viral replication after 3 days by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50547640BDBM50547640(CHEMBL4746579)
Affinity DataIC50: 0.00200nMAssay Description:Inhibition of HCV genotype 1b NS5A infected in Huh7 cells assessed as reduction in viral replication incubated 3 days and measured by Celltiter Glo a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50547639BDBM50547639(CHEMBL4744183)
Affinity DataIC50: 0.00200nMAssay Description:Inhibition of HCV genotype 1b NS5A infected in Huh7 cells assessed as reduction in viral replication incubated 3 days and measured by Celltiter Glo a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50547629BDBM50547629(CHEMBL4763617)
Affinity DataIC50: 0.00200nMAssay Description:Inhibition of HCV genotype 1b NS5A infected in Huh7 cells assessed as reduction in viral replication incubated 3 days and measured by Celltiter Glo a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50547643BDBM50547643(CHEMBL4764688)
Affinity DataIC50: 0.00200nMAssay Description:Inhibition of HCV genotype 1b NS5A infected in Huh7 cells assessed as reduction in viral replication incubated 3 days and measured by Celltiter Glo a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50547642BDBM50547642(CHEMBL4780002)
Affinity DataIC50: 0.00200nMAssay Description:Inhibition of HCV genotype 1b NS5A infected in Huh7 cells assessed as reduction in viral replication incubated 3 days and measured by Celltiter Glo a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50453106BDBM50453106(CHEMBL4215923)
Affinity DataEC50:  0.00200nMAssay Description:Inhibition of NS5A in HuH7 cell infected HCV genotype 1a H77 assessed as decrease in viral replication after 3 days by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50547631BDBM50547631(CHEMBL4798211)
Affinity DataIC50: 0.00200nMAssay Description:Inhibition of HCV genotype 1b NS5A infected in Huh7 cells assessed as reduction in viral replication incubated 3 days and measured by Celltiter Glo a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531947BDBM50531947(CHEMBL4566096)
Affinity DataEC50:  0.00200nMAssay Description:Inhibition of NS5A in HCV genotype 1a assessed as decrease in viral replicationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531957BDBM50531957(CHEMBL4582225)
Affinity DataEC50:  0.00200nMAssay Description:Inhibition of NS5A in HCV genotype 1a assessed as decrease in viral replicationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531962BDBM50531962(CHEMBL4577346)
Affinity DataEC50:  0.00200nMAssay Description:Inhibition of NS5A in HCV genotype 1a assessed as decrease in viral replicationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50547636BDBM50547636(CHEMBL4744064)
Affinity DataIC50: 0.00200nMAssay Description:Inhibition of HCV genotype 1b NS5A infected in Huh7 cells assessed as reduction in viral replication incubated 3 days and measured by Celltiter Glo a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50547635BDBM50547635(CHEMBL4798433)
Affinity DataIC50: 0.00200nMAssay Description:Inhibition of HCV genotype 1b NS5A infected in Huh7 cells assessed as reduction in viral replication incubated 3 days and measured by Celltiter Glo a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50547650BDBM50547650(CHEMBL4797491)
Affinity DataIC50: 0.00200nMAssay Description:Inhibition of HCV genotype 1b NS5A infected in Huh7 cells assessed as reduction in viral replication incubated 3 days and measured by Celltiter Glo a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50547649BDBM50547649(CHEMBL4793304)
Affinity DataIC50: 0.00200nMAssay Description:Inhibition of HCV genotype 1b NS5A infected in Huh7 cells assessed as reduction in viral replication incubated 3 days and measured by Celltiter Glo a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595029BDBM50595029(CHEMBL5191072)
Affinity DataEC50:  0.00200nMAssay Description:Inhibition of HCV genotype 1b NS5AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50547637BDBM50547637(CHEMBL4745761)
Affinity DataIC50: 0.00200nMAssay Description:Inhibition of HCV genotype 1b NS5A infected in Huh7 cells assessed as reduction in viral replication incubated 3 days and measured by Celltiter Glo a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531965BDBM50531965(CHEMBL4542548)
Affinity DataEC50:  0.00220nMAssay Description:Inhibition of NS5A in HCV genotype 1a assessed as decrease in viral replicationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531966BDBM50531966(CHEMBL4450175)
Affinity DataEC50:  0.00270nMAssay Description:Inhibition of NS5A in HCV genotype 1a assessed as decrease in viral replicationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531942BDBM50531942(CHEMBL4454064)
Affinity DataEC50:  0.00290nMAssay Description:Inhibition of NS5A in HCV genotype 1a assessed as decrease in viral replicationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50458020BDBM50458020(CHEMBL4203791)
Affinity DataEC50:  0.00300nMAssay Description:Inhibition of NS5A in HCV genotype 1b infected in human HuH7 replicon cells assessed as reduction in viral replication after 3 days by luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50458023BDBM50458023(CHEMBL4214282)
Affinity DataEC50:  0.00300nMAssay Description:Inhibition of NS5A in HCV genotype 1b infected in human HuH7 replicon cells assessed as reduction in viral replication after 3 days by luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50547628BDBM50547628(CHEMBL4753603)
Affinity DataIC50: 0.00300nMAssay Description:Inhibition of HCV genotype 1b NS5A infected in Huh7 cells assessed as reduction in viral replication incubated 3 days and measured by Celltiter Glo a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50514776BDBM50514776(CHEMBL4465921)
Affinity DataEC50:  0.00300nMAssay Description:Inhibition of NS5A in HCV genotype 1b infected in HuH-Lcu-Neo cells assessed as reduction in viral replication incubated for 48 hrs by luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531960BDBM50531960(CHEMBL4438612)
Affinity DataEC50:  0.00300nMAssay Description:Inhibition of NS5A in HCV genotype 1b assessed as decrease in viral replicationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50533598BDBM50533598(CHEMBL4580319)
Affinity DataEC50:  0.00300nMAssay Description:Inhibition of HCV genotype 1b replicons NS5A infected in human Huh7 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetNonstructural protein 5A(Hepacivirus C)
Chia Tai Tianqing Pharmaceutical Group

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50505975BDBM50505975(CHEMBL4473049)
Affinity DataIC50: 0.00300nMAssay Description:Inhibition of NS5A in HCV genotype 4a infected in human HuH7.5/Con1/SG-Neo(I)-hRluc2aUb cells assessed as inhibition of replicon levels incubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
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