Compile Data Set for Download or QSAR
Report error Found 36 Enz. Inhib. hit(s) with Target = 'Bromodomain testis-specific protein [287-359]'
TargetBromodomain testis-specific protein [287-359](Human)
University Of Texas

US Patent
LigandChemical structure of BindingDB Monomer ID 205429BDBM205429( (R)-JQ1 (3) | US9320741, (R)-JQ1 | US10407441, Co...)
Affinity DataIC50: 217nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2022
Entry Details
US Patent

TargetBromodomain testis-specific protein [287-359](Human)
University Of Texas

US Patent
LigandChemical structure of BindingDB Monomer ID 50103503BDBM50103503(CHEMBL2393130 | US11117865, Compound RVX-208 | US2...)
Affinity DataIC50: 708nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2022
Entry Details
US Patent

TargetBromodomain testis-specific protein [287-359](Human)
University Of Texas

US Patent
LigandChemical structure of BindingDB Monomer ID 674640BDBM674640(US20240158355, Compound 80)
Affinity DataIC50: 1.02E+3nMAssay Description:No details are given.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2024
Entry Details
US Patent

TargetBromodomain testis-specific protein [287-359](Human)
University Of Texas

US Patent
LigandChemical structure of BindingDB Monomer ID 518731BDBM518731(US11117865, Compound ZL0590)
Affinity DataIC50: 1.86E+3nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2022
Entry Details
US Patent

TargetBromodomain testis-specific protein [287-359](Human)
University Of Texas

US Patent
LigandChemical structure of BindingDB Monomer ID 518731BDBM518731(US11117865, Compound ZL0590)
Affinity DataIC50: 1.86E+3nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2022
Entry Details
US Patent

TargetBromodomain testis-specific protein [287-359](Human)
University Of Texas

US Patent
LigandChemical structure of BindingDB Monomer ID 518799BDBM518799(US11117865, Compound ZL0591)
Affinity DataIC50: 1.95E+3nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2022
Entry Details
US Patent

TargetBromodomain testis-specific protein [287-359](Human)
University Of Texas

US Patent
LigandChemical structure of BindingDB Monomer ID 518799BDBM518799(US11117865, Compound ZL0591)
Affinity DataIC50: 1.95E+3nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2022
Entry Details
US Patent

TargetBromodomain testis-specific protein [287-359](Human)
University Of Texas

US Patent
LigandChemical structure of BindingDB Monomer ID 674638BDBM674638(US20240158355, Compound 78)
Affinity DataIC50: 2.45E+3nMAssay Description:No details are given.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2024
Entry Details
US Patent

TargetBromodomain testis-specific protein [287-359](Human)
University Of Texas

US Patent
LigandChemical structure of BindingDB Monomer ID 50370182BDBM50370182(CHEMBL4176038 | US11117865, Compound ZL0420)
Affinity DataIC50: 2.78E+3nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2022
Entry Details
US Patent

TargetBromodomain testis-specific protein [287-359](Human)
University Of Texas

US Patent
LigandChemical structure of BindingDB Monomer ID 50370181BDBM50370181(CHEMBL4159382 | US11117865, Compound ZL0454)
Affinity DataIC50: 3.08E+3nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2022
Entry Details
US Patent

TargetBromodomain testis-specific protein [287-359](Human)
University Of Texas

US Patent
LigandChemical structure of BindingDB Monomer ID 50527819BDBM50527819(CHEMBL4557050 | US11117865, Compound ZL0516)
Affinity DataIC50: 3.18E+3nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2022
Entry Details
US Patent

TargetBromodomain testis-specific protein [287-359](Human)
University Of Texas

US Patent
LigandChemical structure of BindingDB Monomer ID 50527819BDBM50527819(CHEMBL4557050 | US11117865, Compound ZL0516)
Affinity DataIC50: 3.18E+3nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2022
Entry Details
US Patent

TargetBromodomain testis-specific protein [287-359](Human)
University Of Texas

US Patent
LigandChemical structure of BindingDB Monomer ID 674639BDBM674639(US20240158355, Compound 79)
Affinity DataIC50: 3.21E+3nMAssay Description:No details are given.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2024
Entry Details
US Patent

TargetBromodomain testis-specific protein [287-359](Human)
University Of Texas

US Patent
LigandChemical structure of BindingDB Monomer ID 674566BDBM674566(US20240158355, Compound 6)
Affinity DataIC50: 6.30E+3nMAssay Description:No details are given.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2024
Entry Details
US Patent

TargetBromodomain testis-specific protein [287-359](Human)
University Of Texas

US Patent
LigandChemical structure of BindingDB Monomer ID 674636BDBM674636(US20240158355, Compound 76)
Affinity DataIC50: 9.48E+3nMAssay Description:No details are given.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2024
Entry Details
US Patent

TargetBromodomain testis-specific protein [287-359](Human)
University Of Texas

US Patent
LigandChemical structure of BindingDB Monomer ID 674570BDBM674570(US20240158355, Compound 11 | US20240158355, Compou...)
Affinity DataIC50: 1.00E+4nMAssay Description:No details are given.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2024
Entry Details
US Patent

TargetBromodomain testis-specific protein [287-359](Human)
University Of Texas

US Patent
LigandChemical structure of BindingDB Monomer ID 674625BDBM674625(US20240158355, Compound 65)
Affinity DataIC50: 1.00E+4nMAssay Description:No details are given.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2024
Entry Details
US Patent

TargetBromodomain testis-specific protein [287-359](Human)
University Of Texas

US Patent
LigandChemical structure of BindingDB Monomer ID 674569BDBM674569(US20240158355, Compound 9)
Affinity DataIC50: 1.00E+4nMAssay Description:No details are given.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2024
Entry Details
US Patent

TargetBromodomain testis-specific protein [287-359](Human)
University Of Texas

US Patent
LigandChemical structure of BindingDB Monomer ID 674570BDBM674570(US20240158355, Compound 11 | US20240158355, Compou...)
Affinity DataIC50: 1.00E+4nMAssay Description:No details are given.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2024
Entry Details
US Patent

TargetBromodomain testis-specific protein [287-359](Human)
University Of Texas

US Patent
LigandChemical structure of BindingDB Monomer ID 674577BDBM674577(US20240158355, Compound 17)
Affinity DataIC50: 1.00E+4nMAssay Description:No details are given.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2024
Entry Details
US Patent

TargetBromodomain testis-specific protein [287-359](Human)
University Of Texas

US Patent
LigandChemical structure of BindingDB Monomer ID 674578BDBM674578(US20240158355, Compound 18)
Affinity DataIC50: 1.00E+4nMAssay Description:No details are given.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2024
Entry Details
US Patent

TargetBromodomain testis-specific protein [287-359](Human)
University Of Texas

US Patent
LigandChemical structure of BindingDB Monomer ID 518854BDBM518854(US11117865, Compound ZL0497)
Affinity DataIC50: 1.00E+4nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2022
Entry Details
US Patent

TargetBromodomain testis-specific protein [287-359](Human)
University Of Texas

US Patent
LigandChemical structure of BindingDB Monomer ID 674573BDBM674573(US20240158355, Compound 13)
Affinity DataIC50: 1.00E+4nMAssay Description:No details are given.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2024
Entry Details
US Patent

TargetBromodomain testis-specific protein [287-359](Human)
University Of Texas

US Patent
LigandChemical structure of BindingDB Monomer ID 674627BDBM674627(US20240158355, Compound 67)
Affinity DataIC50: 1.00E+4nMAssay Description:No details are given.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2024
Entry Details
US Patent

TargetBromodomain testis-specific protein [287-359](Human)
University Of Texas

US Patent
LigandChemical structure of BindingDB Monomer ID 674581BDBM674581(US20240158355, Compound 21)
Affinity DataIC50: 1.00E+4nMAssay Description:No details are given.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2024
Entry Details
US Patent

TargetBromodomain testis-specific protein [287-359](Human)
University Of Texas

US Patent
LigandChemical structure of BindingDB Monomer ID 674582BDBM674582(US20240158355, Compound 22)
Affinity DataIC50: 1.00E+4nMAssay Description:No details are given.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2024
Entry Details
US Patent

TargetBromodomain testis-specific protein [287-359](Human)
University Of Texas

US Patent
LigandChemical structure of BindingDB Monomer ID 674637BDBM674637(US20240158355, Compound 77)
Affinity DataIC50: 1.00E+4nMAssay Description:No details are given.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2024
Entry Details
US Patent

TargetBromodomain testis-specific protein [287-359](Human)
University Of Texas

US Patent
LigandChemical structure of BindingDB Monomer ID 674579BDBM674579(US20240158355, Compound 19)
Affinity DataIC50: 1.00E+4nMAssay Description:No details are given.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2024
Entry Details
US Patent

TargetBromodomain testis-specific protein [287-359](Human)
University Of Texas

US Patent
LigandChemical structure of BindingDB Monomer ID 674580BDBM674580(US20240158355, Compound 20)
Affinity DataIC50: 1.00E+4nMAssay Description:No details are given.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2024
Entry Details
US Patent

TargetBromodomain testis-specific protein [287-359](Human)
University Of Texas

US Patent
LigandChemical structure of BindingDB Monomer ID 674586BDBM674586(US20240158355, Compound 26)
Affinity DataIC50: 1.00E+4nMAssay Description:No details are given.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2024
Entry Details
US Patent

TargetBromodomain testis-specific protein [287-359](Human)
University Of Texas

US Patent
LigandChemical structure of BindingDB Monomer ID 674567BDBM674567(US20240158355, Compound 7)
Affinity DataIC50: 1.00E+4nMAssay Description:No details are given.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2024
Entry Details
US Patent

TargetBromodomain testis-specific protein [287-359](Human)
University Of Texas

US Patent
LigandChemical structure of BindingDB Monomer ID 674615BDBM674615(US20240158355, Compound 55)
Affinity DataIC50: 1.00E+4nMAssay Description:No details are given.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2024
Entry Details
US Patent

TargetBromodomain testis-specific protein [287-359](Human)
University Of Texas

US Patent
LigandChemical structure of BindingDB Monomer ID 674587BDBM674587(US20240158355, Compound 27)
Affinity DataIC50: 1.00E+4nMAssay Description:No details are given.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2024
Entry Details
US Patent

TargetBromodomain testis-specific protein [287-359](Human)
University Of Texas

US Patent
LigandChemical structure of BindingDB Monomer ID 674568BDBM674568(US20240158355, Compound 8)
Affinity DataIC50: 1.00E+4nMAssay Description:No details are given.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2024
Entry Details
US Patent

TargetBromodomain testis-specific protein [287-359](Human)
University Of Texas

US Patent
LigandChemical structure of BindingDB Monomer ID 674564BDBM674564(US20240158355, Compound 4)
Affinity DataIC50: 1.00E+4nMAssay Description:No details are given.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2024
Entry Details
US Patent

TargetBromodomain testis-specific protein [287-359](Human)
University Of Texas

US Patent
LigandChemical structure of BindingDB Monomer ID 674585BDBM674585(US20240158355, Compound 25)
Affinity DataIC50: 1.00E+4nMAssay Description:No details are given.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2024
Entry Details
US Patent