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Report error Found 68 Enz. Inhib. hit(s) with Target = 'C-C motif chemokine 2'
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50331728(N-(2-((3S,4S)-1-(cis-4-(benzo[d][1,3]dioxol-5-yl)-...)
Affinity DataKd:  0.230nMAssay Description:Displacement of [3H]INCB3344 from human CCR2 receptor expressed in human U2OS cell membranes assessed as association and dissociation of radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50331728(N-(2-((3S,4S)-1-(cis-4-(benzo[d][1,3]dioxol-5-yl)-...)
Affinity DataKd:  0.720nMAssay Description:Displacement of [3H]INCB3344 from human CCR2 receptor expressed in human U2OS cell membranes assessed as association and dissociation of compound by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50331728(N-(2-((3S,4S)-1-(cis-4-(benzo[d][1,3]dioxol-5-yl)-...)
Affinity DataKd:  0.900nMAssay Description:Displacement of [3H]INCB3344 from human CCR2 receptor expressed in human U2OS cell membranes by saturation binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50331728(N-(2-((3S,4S)-1-(cis-4-(benzo[d][1,3]dioxol-5-yl)-...)
Affinity DataKd:  1.20nMAssay Description:Displacement of [3H]INCB3344 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50440552(CHEMBL2426340)
Affinity DataKi:  3.60nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50440556(CHEMBL2426334)
Affinity DataKi:  3.90nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50440549(CHEMBL2426351)
Affinity DataKi:  6.10nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50440557(CHEMBL2426335)
Affinity DataKi:  6.30nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257898((1S,3R)-N-(3,5-bis(trifluoromethyl)benzyl)-1-isopr...)
Affinity DataKi:  6.80nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50440552(CHEMBL2426340)
Affinity DataKi:  7.20nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50440552(CHEMBL2426340)
Affinity DataKi:  7.20nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50607762(CHEMBL5220494)
Affinity DataIC50: 16nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50440551(CHEMBL2426354)
Affinity DataKi:  18nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50607758(CHEMBL5219991)
Affinity DataIC50: 20nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50607759(CHEMBL5218813)
Affinity DataIC50: 25nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50440558(CHEMBL2426336)
Affinity DataKi:  27nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50440550(CHEMBL2426352)
Affinity DataKi:  29nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257900((1S,3R)-N-(3,5-bis(trifluoromethyl)benzyl)-1-isopr...)
Affinity DataKi:  31nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50607770(CHEMBL5219919)
Affinity DataIC50: 32nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50607766(CHEMBL5220128)
Affinity DataIC50: 32nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50440545(CHEMBL2426345)
Affinity DataKi:  33nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50440559(CHEMBL2426337)
Affinity DataKi:  35nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50607757(CHEMBL5218822)
Affinity DataIC50: 40nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50607765(CHEMBL5218726)
Affinity DataIC50: 40nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50607767(CHEMBL5218909)
Affinity DataIC50: 40nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50607769(CHEMBL5219538)
Affinity DataIC50: 40nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50607768(CHEMBL5219602)
Affinity DataIC50: 40nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50440546(CHEMBL2426346)
Affinity DataKi:  43nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50607761(CHEMBL5221069)
Affinity DataIC50: 50nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50607763(CHEMBL5218817)
Affinity DataIC50: 50nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257992((1S,3R)-N-(3,5-bis(trifluoromethyl)benzyl)-3-(2,3-...)
Affinity DataKi:  50nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50440554(CHEMBL2426357)
Affinity DataKi:  54nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50440553(CHEMBL2426356)
Affinity DataKi:  55nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50440548(CHEMBL2426348)
Affinity DataKi:  70nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50440547(CHEMBL2426347)
Affinity DataKi:  86nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257792((1S,3R)-N-(3,5-bis(trifluoromethyl)benzyl)-3-(cycl...)
Affinity DataKi:  110nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50607760(CHEMBL5219194)
Affinity DataIC50: 126nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50440555(CHEMBL2426333)
Affinity DataKi:  130nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50440544(CHEMBL2426344)
Affinity DataKi:  134nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50607753(CHEMBL5219077)
Affinity DataIC50: 158nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50603097(CHEMBL5195288)
Affinity DataIC50: 200nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50603092(CHEMBL5190509)
Affinity DataIC50: 251nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50607747(CHEMBL5220077)
Affinity DataIC50: 398nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50607752(CHEMBL5220099)
Affinity DataIC50: 398nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50603089(CHEMBL5194720)
Affinity DataIC50: 398nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50440542(CHEMBL2426342)
Affinity DataKi:  437nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50607744(CHEMBL5220904)
Affinity DataIC50: 631nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50607746(CHEMBL5220753)
Affinity DataIC50: 631nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50607745(CHEMBL5220501)
Affinity DataIC50: 631nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetC-C motif chemokine 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50607750(CHEMBL5220275)
Affinity DataIC50: 631nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
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