Compile Data Set for Download or QSAR
Report error Found 380 Enz. Inhib. hit(s) with Target = 'Gamma-aminobutyric acid receptor subunit beta'
TargetGamma-aminobutyric acid receptor subunit beta-3(Human)
Shimane University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50214664BDBM50214664(5-chloromethyl-1-(2,6-dichloro-4-trifluoromethylph...)
Affinity DataKi:  0.659nMAssay Description:Displacement of [3H]EBOB from human recombinant GABAbeta3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit beta-3(Human)
Shimane University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50214659BDBM50214659(1-(2,6-dichloro-4-trifluoromethylphenyl)-5-methyl-...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]EBOB from human recombinant GABAbeta3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit beta-3(Human)
Shimane University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50214673BDBM50214673(1-(2,6-dichloro-4-trifluoromethylphenyl)-5-hydroxy...)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]EBOB from human recombinant GABAbeta3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit beta-3(Human)
Shimane University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50214650BDBM50214650(1-(2,6-dichloro-4-trifluoromethylphenyl)-4,5-dieth...)
Affinity DataKi:  4.30nMAssay Description:Displacement of [3H]EBOB from human recombinant GABAbeta3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit beta-3(Human)
Shimane University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50214662BDBM50214662(1-(2,6-dichloro-4-trifluoromethylphenyl)-4-ethyl-5...)
Affinity DataKi:  7.10nMAssay Description:Displacement of [3H]EBOB from human recombinant GABAbeta3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit beta-3(Human)
Shimane University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50214670BDBM50214670(1-(2,6-dichloro-4-trifluoromethylphenyl)-5-ethyl-4...)
Affinity DataKi:  8.10nMAssay Description:Displacement of [3H]EBOB from human recombinant GABAbeta3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit beta-3(Human)
Shimane University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50214665BDBM50214665(1-(2,6-dibromo-4-trifluoromethylphenyl)-5-methyl-4...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]EBOB from human recombinant GABAbeta3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit beta-3(Human)
Shimane University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50106148BDBM50106148(5-amino-1-[2,6-dichloro-4-(trifluoromethyl)phenyl]...)
Affinity DataIC50: 28nMAssay Description:Inhibition of [3H]EBOB binding to human GABA-A receptor beta3 subunit (range 1-28)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit beta-3(Human)
Shimane University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50106149BDBM50106149(1-(2,6-Dichloro-4-trifluoromethyl-phenyl)-4-(3-tri...)
Affinity DataIC50: 28nMAssay Description:Inhibition of [3H]EBOB binding to human GABA-A receptor beta3 subunit (range 1-28)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit beta-3(Human)
Shimane University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50106149BDBM50106149(1-(2,6-Dichloro-4-trifluoromethyl-phenyl)-4-(3-tri...)
Affinity DataIC50: 28nMAssay Description:Inhibition of [3H]EBOB binding to drosophila GABA-A receptor (range 1-28)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit beta-3(Human)
Shimane University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50106148BDBM50106148(5-amino-1-[2,6-dichloro-4-(trifluoromethyl)phenyl]...)
Affinity DataIC50: 28nMAssay Description:Inhibition of [3H]EBOB binding to human GABA-A receptor beta3 subunit (range 1-28)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit beta(House fly)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179909BDBM50179909(2-(2,6-dichloro-4-(trifluoromethyl)phenyl)-4-methy...)
Affinity DataIC50: 30nMAssay Description:Displacement of [3H]EBOB from housefly neuronal membrane GABA receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit beta-3(Human)
Shimane University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50214653BDBM50214653(1-(2,6-dichloro-4-trifluoromethylphenyl)-4-ethyl-5...)
Affinity DataKi:  47nMAssay Description:Displacement of [3H]EBOB from human recombinant GABAbeta3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit beta-3(Human)
Shimane University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50214661BDBM50214661(4-chloromethyl-1-(2,6-dichloro-4-trifluoromethylph...)
Affinity DataKi:  67nMAssay Description:Displacement of [3H]EBOB from human recombinant GABAbeta3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit beta-3(Human)
Shimane University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50214647BDBM50214647(1-(2,6-dichloro-4-(trifluoromethyl)phenyl)-5-ethyl...)
Affinity DataKi:  70.1nMAssay Description:Displacement of [3H]EBOB from human recombinant GABAbeta3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit beta(House fly)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179898BDBM50179898(2-(2,6-dichloro-4-(trifluoromethyl)phenyl)-4,4,6,6...)
Affinity DataIC50: 74nMAssay Description:Displacement of [3H]EBOB from housefly neuronal membrane GABA receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit beta(House fly)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179896BDBM50179896(2-(2,6-dichloro-4-(trifluoromethyl)phenyl)-2,4,5,6...)
Affinity DataIC50: 83nMAssay Description:Displacement of [3H]EBOB from housefly neuronal membrane GABA receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit beta-1(Rat)
Sage Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 625778BDBM625778(US20230322846, Example 267)
Affinity DataIC50: 100nMAssay Description:Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2023
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit beta-1(Rat)
Sage Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 625779BDBM625779(US20230322846, Example 268)
Affinity DataIC50: 100nMAssay Description:Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2023
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit beta-1(Rat)
Sage Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 625780BDBM625780(US20230322846, Example 269 | Synthesis of 1-((R)-2...)
Affinity DataIC50: 100nMAssay Description:Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2023
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit beta-1(Rat)
Sage Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 625781BDBM625781(US20230322846, Example 270)
Affinity DataIC50: 100nMAssay Description:Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2023
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit beta-1(Rat)
Sage Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 625774BDBM625774(US20230322846, Example 263)
Affinity DataIC50: 100nMAssay Description:Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2023
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit beta(House fly)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179903BDBM50179903(2-(2,6-dichloro-4-(trifluoromethyl)phenyl)-5,5-dif...)
Affinity DataIC50: 100nMAssay Description:Displacement of [3H]EBOB from housefly neuronal membrane GABA receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit beta-1(Rat)
Sage Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 625786BDBM625786(US20230322846, Example 275)
Affinity DataIC50: 100nMAssay Description:Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2023
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit beta-1(Rat)
Sage Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 625787BDBM625787(US20230322846, Example 276)
Affinity DataIC50: 100nMAssay Description:Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2023
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit beta-1(Rat)
Sage Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 625788BDBM625788(US20230322846, Example 278)
Affinity DataIC50: 100nMAssay Description:Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2023
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit beta-1(Rat)
Sage Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 625789BDBM625789(US20230322846, Example 279)
Affinity DataIC50: 100nMAssay Description:Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2023
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit beta-1(Rat)
Sage Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 625782BDBM625782(US20230322846, Example 271)
Affinity DataIC50: 100nMAssay Description:Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2023
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit beta(House fly)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179912BDBM50179912(2-(2,6-dichloro-4-(trifluoromethyl)phenyl)-4,4-dif...)
Affinity DataIC50: 100nMAssay Description:Displacement of [3H]EBOB from housefly neuronal membrane GABA receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit beta-1(Rat)
Sage Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 625783BDBM625783(US20230322846, Example 272)
Affinity DataIC50: 100nMAssay Description:Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2023
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit beta-1(Rat)
Sage Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 625784BDBM625784(US20230322846, Example 273)
Affinity DataIC50: 100nMAssay Description:Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2023
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit beta-1(Rat)
Sage Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 625763BDBM625763(US20230322846, Example 252)
Affinity DataIC50: 100nMAssay Description:Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2023
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit beta-1(Rat)
Sage Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 625765BDBM625765(US20230322846, Example 254)
Affinity DataIC50: 100nMAssay Description:Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2023
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit beta-1(Rat)
Sage Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 625761BDBM625761(US20230322846, Example 250)
Affinity DataIC50: 100nMAssay Description:Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2023
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit beta-1(Rat)
Sage Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 625770BDBM625770(US20230322846, Example 259)
Affinity DataIC50: 100nMAssay Description:Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2023
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit beta-1(Rat)
Sage Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 625771BDBM625771(US20230322846, Example 260)
Affinity DataIC50: 100nMAssay Description:Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2023
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit beta-1(Rat)
Sage Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 625773BDBM625773(US20230322846, Example 262)
Affinity DataIC50: 100nMAssay Description:Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2023
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit beta-1(Rat)
Sage Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 625767BDBM625767(US20230322846, Example 256)
Affinity DataIC50: 100nMAssay Description:Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2023
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit beta-1(Rat)
Sage Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 625810BDBM625810(US20230322846, Example 304)
Affinity DataIC50: 100nMAssay Description:Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2023
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit beta-1(Rat)
Sage Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 625811BDBM625811(US20230322846, Example 305 | Synthesis of 1-((R)-2...)
Affinity DataIC50: 100nMAssay Description:Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2023
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit beta-1(Rat)
Sage Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 625812BDBM625812(US20230322846, Example 306)
Affinity DataIC50: 100nMAssay Description:Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2023
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit beta-1(Rat)
Sage Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 625813BDBM625813(US20230322846, Example 307 | Synthesis of 1-((R)-2...)
Affinity DataIC50: 100nMAssay Description:Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2023
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit beta-1(Rat)
Sage Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 625806BDBM625806(US20230322846, Example 300)
Affinity DataIC50: 100nMAssay Description:Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2023
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit beta-1(Rat)
Sage Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 625807BDBM625807(US20230322846, Example 301 | Synthesis of 1-((R)-2...)
Affinity DataIC50: 100nMAssay Description:Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2023
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit beta-1(Rat)
Sage Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 625808BDBM625808(US20230322846, Example 302)
Affinity DataIC50: 100nMAssay Description:Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2023
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit beta-1(Rat)
Sage Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 625809BDBM625809(US20230322846, Example 303 | Synthesis of 1-((R)-2...)
Affinity DataIC50: 100nMAssay Description:Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2023
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit beta-1(Rat)
Sage Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 625818BDBM625818(US20230322846, Example 312)
Affinity DataIC50: 100nMAssay Description:Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2023
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit beta-1(Rat)
Sage Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 625819BDBM625819(US20230322846, Example 313)
Affinity DataIC50: 100nMAssay Description:Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2023
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit beta-1(Rat)
Sage Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 625821BDBM625821(US20230322846, Example 315)
Affinity DataIC50: 100nMAssay Description:Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2023
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit beta-1(Rat)
Sage Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 625814BDBM625814(US20230322846, Example 308)
Affinity DataIC50: 100nMAssay Description:Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2023
Entry Details
US Patent

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