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Report error Found 119 Enz. Inhib. hit(s) with Target = 'Peptidase'
TargetPeptidase(Staphylococcus aureus)
Ain Shams University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50611988BDBM50611988(CEFTAROLINE | Ceftaroline | T 91825 | T-91825)
Affinity DataIC50: 0.160nMAssay Description:Binding affinity to methicillin resistant Staphylococcus aureus PBP2aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetPeptidase(Staphylococcus aureus)
Ain Shams University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50611989BDBM50611989(CHEMBL5271107)
Affinity DataIC50: 1.20nMAssay Description:Displacement of [3H]-penicillin from Staphylococcus aureus PBP2aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50031688BDBM50031688(CHEMBL3360299)
Affinity DataIC50: 3nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50031689BDBM50031689(CHEMBL3360298)
Affinity DataIC50: 3nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50031695BDBM50031695(CHEMBL3360292)
Affinity DataIC50: 4nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50031685BDBM50031685(CHEMBL3360301)
Affinity DataIC50: 4nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50031687BDBM50031687(CHEMBL3360300)
Affinity DataIC50: 4nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50031684BDBM50031684(CHEMBL3360302)
Affinity DataIC50: 4nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50031690BDBM50031690(CHEMBL3360297)
Affinity DataIC50: 5nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50031635BDBM50031635(CHEMBL3359786)
Affinity DataIC50: 6nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50031632BDBM50031632(CHEMBL3359790)
Affinity DataIC50: 6nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50031693BDBM50031693(CHEMBL3360294)
Affinity DataIC50: 6nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50031713BDBM50031713(CHEMBL3360282)
Affinity DataIC50: 6nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 103023BDBM103023(US8541363, PVA-039)
Affinity DataIC50: 6.30nMAssay Description:The fluorogenic substrate used for measuring Der p 1 proteolytic activity was 2-aminobenzoylvalylalanylnorleucylseryl-(3-nitro)tyrosinyl aspartamide....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2013
Entry Details
US Patent

TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50031668BDBM50031668(CHEMBL3359782)
Affinity DataIC50: 7nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 103022BDBM103022(US8541363, PVA-037)
Affinity DataIC50: 7.85nMAssay Description:The fluorogenic substrate used for measuring Der p 1 proteolytic activity was 2-aminobenzoylvalylalanylnorleucylseryl-(3-nitro)tyrosinyl aspartamide....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2013
Entry Details
US Patent

TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50031719BDBM50031719(CHEMBL3359772)
Affinity DataIC50: 8nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50031711BDBM50031711(CHEMBL3360284)
Affinity DataIC50: 8nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50031697BDBM50031697(CHEMBL3360290)
Affinity DataIC50: 9nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50031714BDBM50031714(CHEMBL3360281)
Affinity DataIC50: 9nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50031694BDBM50031694(CHEMBL3360293)
Affinity DataIC50: 10nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50031700BDBM50031700(CHEMBL3360287)
Affinity DataIC50: 11nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50031682BDBM50031682(CHEMBL3359775)
Affinity DataIC50: 12nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50031673BDBM50031673(CHEMBL3359780)
Affinity DataIC50: 13nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 103021BDBM103021(US8541363, PVA-038)
Affinity DataIC50: 13nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 103021BDBM103021(US8541363, PVA-038)
Affinity DataIC50: 13.3nMAssay Description:The fluorogenic substrate used for measuring Der p 1 proteolytic activity was 2-aminobenzoylvalylalanylnorleucylseryl-(3-nitro)tyrosinyl aspartamide....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2013
Entry Details
US Patent

TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50031696BDBM50031696(CHEMBL3360291)
Affinity DataIC50: 14nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 103020BDBM103020(US8541363, PVA-026)
Affinity DataIC50: 14nMAssay Description:The fluorogenic substrate used for measuring Der p 1 proteolytic activity was 2-aminobenzoylvalylalanylnorleucylseryl-(3-nitro)tyrosinyl aspartamide....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2013
Entry Details
US Patent

TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 103020BDBM103020(US8541363, PVA-026)
Affinity DataIC50: 14nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50031698BDBM50031698(CHEMBL3360289)
Affinity DataIC50: 14nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50031699BDBM50031699(CHEMBL3360288)
Affinity DataIC50: 14nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase(Staphylococcus aureus)
Ain Shams University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50482776BDBM50482776(CHEBI:70718 | Ceftaroline Fosamil | PPI-0903 | TAK...)
Affinity DataIC50: 14.6nMAssay Description:Binding affinity to against methicillin-, daptomycin-resistant, vancomycin-intermediate, beta-lactamase-positive Staphylococcus aureus 25 PBP2a by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50031719BDBM50031719(CHEMBL3359772)
Affinity DataIC50: 17nMAssay Description:Reversible inhibition of house dust mite Derp-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50031692BDBM50031692(CHEMBL3360295)
Affinity DataIC50: 17nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50031633BDBM50031633(CHEMBL3359789)
Affinity DataIC50: 17nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50031710BDBM50031710(CHEMBL3360285)
Affinity DataIC50: 17nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50031683BDBM50031683(CHEMBL3359773)
Affinity DataIC50: 18nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50031670BDBM50031670(CHEMBL3359781)
Affinity DataIC50: 18nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50031691BDBM50031691(CHEMBL3360296)
Affinity DataIC50: 20nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50031678BDBM50031678(CHEMBL3359779)
Affinity DataIC50: 20nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50031715BDBM50031715(CHEMBL3359791)
Affinity DataIC50: 24nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50031681BDBM50031681(CHEMBL3359777)
Affinity DataIC50: 42nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50031712BDBM50031712(CHEMBL3360283)
Affinity DataIC50: 47nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50031634BDBM50031634(CHEMBL3359787)
Affinity DataIC50: 55nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50031722BDBM50031722(CHEMBL3359770)
Affinity DataIC50: 65nMAssay Description:Reversible inhibition of house dust mite Derp-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50031717BDBM50031717(CHEMBL3359784)
Affinity DataIC50: 67nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50031716BDBM50031716(CHEMBL3359788)
Affinity DataIC50: 115nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50031701BDBM50031701(CHEMBL3360286)
Affinity DataIC50: 117nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase, M28 family(Bacteroides forsythus)
Fraunhofer-Gesellschaft Zur Forderung Der Angewandten Forschung

US Patent
LigandChemical structure of BindingDB Monomer ID 667852BDBM667852(US11958871, Example 17)
Affinity DataKi:  123nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2024
Entry Details
US Patent

TargetPeptidase(Staphylococcus aureus)
Ain Shams University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50569542BDBM50569542(CHEMBL4847813)
Affinity DataKd:  129nMAssay Description:Binding affinity to Staphylococcus aureus PBP2a assessed as equilibrium dissociation constant by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
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