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Found 16 with Last Name = 'blat' and Initial = 'd'
TargetCasein kinase II subunit alpha'/beta(Homo sapiens (Human))
Universit£T Zu K£Ln

Curated by ChEMBL
LigandPNGBDBM50530315(CHEMBL4520531)
Affinity DataKi:  86nMAssay Description:ATP competitive inhibition of recombinant human CK2alpha2 (1 to 335 residues)/CK2beta2 (1 to 193 residues) expressed in Escherichia coli BL21(DE3) us...More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha'/beta(Homo sapiens (Human))
Universit£T Zu K£Ln

Curated by ChEMBL
LigandPNGBDBM50540033(CHEMBL4635554)
Affinity DataKi:  206nMAssay Description:ATP competitive inhibition of recombinant human CK2alpha2 (1 to 335 residues)/CK2beta2 (1 to 193 residues) expressed in Escherichia coli BL21(DE3) us...More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha'/beta(Homo sapiens (Human))
Universit£T Zu K£Ln

Curated by ChEMBL
LigandPNGBDBM50540034(CHEMBL4647986)
Affinity DataKi:  1.47E+3nMAssay Description:ATP competitive inhibition of recombinant human CK2alpha2 (1 to 335 residues)/CK2beta2 (1 to 193 residues) expressed in Escherichia coli BL21(DE3) us...More data for this Ligand-Target Pair
TargetSomatostatin receptor type 2(Homo sapiens (Human))
The Weizmann Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50333670((3R,6S,9S,12S,15S,18S,21S,24S,27S,30S,33S,36R)-21-...)
Affinity DataIC50:  0.400nMAssay Description:Displacement of [125I-Tyr3]octreotide from sst2 receptor expressed in rat AR4-2J cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAtrial natriuretic peptide receptor 1(Homo sapiens (Human))
The Weizmann Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50333671(CHEMBL1643388)
Affinity DataIC50:  6nMAssay Description:Displacement of [125I]ANP from NPR-A expressed in HeLa cells after 3 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
The Weizmann Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50333669(CHEMBL1643384)
Affinity DataIC50:  8.10nMAssay Description:Displacement of [125I-Tyr3]octreotide from sst2 receptor expressed in rat AR4-2J cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
The Weizmann Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50333669(CHEMBL1643384)
Affinity DataIC50:  8.10nMAssay Description:Displacement of [125I-Tyr3]octreotide from sst2 receptor expressed in rat AR4-2J cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAtrial natriuretic peptide receptor 1(Homo sapiens (Human))
The Weizmann Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50333672(CHEMBL1643389)
Affinity DataIC50:  60nMAssay Description:Displacement of [125I]ANP from NPR-A expressed in HeLa cells after 3 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAtrial natriuretic peptide receptor 1(Homo sapiens (Human))
The Weizmann Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50333673(CHEMBL1643390)
Affinity DataIC50:  240nMAssay Description:Displacement of [125I]ANP from NPR-A expressed in HeLa cells after 3 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£T Zu K£Ln

Curated by ChEMBL
LigandPNGBDBM50252622(CHEMBL4070389)
Affinity DataIC50:  370nMAssay Description:Inhibition of human CK2alpha using RRRDDDSDDD peptide as substrate preincubated for 40 mins and measured after 70 mins in the presence of ATP by ADP ...More data for this Ligand-Target Pair
TargetSomatostatin receptor type 2(Homo sapiens (Human))
The Weizmann Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50333668(CHEMBL1643387)
Affinity DataIC50: >600nMAssay Description:Displacement of [125I-Tyr3]octreotide from sst2 receptor expressed in rat AR4-2J cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Tufts University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM578((2S)-N-[(2S,4S,5S)-5-[2-(2,6-dimethylphenoxy)aceta...)
Affinity DataIC50:  1.70E+3nMAssay Description:TP_TRANSPORTER: inhibition of Rhodamine 123 efflux in Caco-2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Tufts University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50069447(1-(3-(4-(m-Chlorophenyl)-1-piperazinyl)propyl)-3-e...)
Affinity DataIC50:  4.70E+3nMAssay Description:TP_TRANSPORTER: inhibition of Rhodamine 123 transepithelial transport (basal to apical) (R123: 5 uM) in Caco-2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Tufts University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM82507((+/-)-Methadone | CAS_5967-73-7 | METHADONE | Meth...)
Affinity DataIC50:  7.50E+3nMAssay Description:TP_TRANSPORTER: inhibition of Rhodamine 123 transepithelial transport (basal to apical) (Rhodamine 123: 5 uM) in Caco-2 cellsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Tufts University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM20607((2-{4-[(1Z)-1,2-diphenylbut-1-en-1-yl]phenoxy}ethy...)
Affinity DataIC50:  2.90E+4nMAssay Description:TP_TRANSPORTER: transepithelial transport of Rhodamine 123 (basal to apical) in Caco-2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Universit£T Zu K£Ln

Curated by ChEMBL
LigandPNGBDBM50602484(CHEMBL5195963)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of N-terminal GST-tagged human CK1epsilon (1 to 348 residues) expressed in baculovirus expression system in presence of peptide substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails PubMed