TargetCasein kinase II subunit alpha'/beta(Homo sapiens (Human))
Universit£T Zu K£Ln
Curated by ChEMBL
Universit£T Zu K£Ln
Curated by ChEMBL
Affinity DataKi: 86nMAssay Description:ATP competitive inhibition of recombinant human CK2alpha2 (1 to 335 residues)/CK2beta2 (1 to 193 residues) expressed in Escherichia coli BL21(DE3) us...More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha'/beta(Homo sapiens (Human))
Universit£T Zu K£Ln
Curated by ChEMBL
Universit£T Zu K£Ln
Curated by ChEMBL
Affinity DataKi: 206nMAssay Description:ATP competitive inhibition of recombinant human CK2alpha2 (1 to 335 residues)/CK2beta2 (1 to 193 residues) expressed in Escherichia coli BL21(DE3) us...More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha'/beta(Homo sapiens (Human))
Universit£T Zu K£Ln
Curated by ChEMBL
Universit£T Zu K£Ln
Curated by ChEMBL
Affinity DataKi: 1.47E+3nMAssay Description:ATP competitive inhibition of recombinant human CK2alpha2 (1 to 335 residues)/CK2beta2 (1 to 193 residues) expressed in Escherichia coli BL21(DE3) us...More data for this Ligand-Target Pair
TargetSomatostatin receptor type 2(Homo sapiens (Human))
The Weizmann Institute Of Science
Curated by ChEMBL
The Weizmann Institute Of Science
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:Displacement of [125I-Tyr3]octreotide from sst2 receptor expressed in rat AR4-2J cellsMore data for this Ligand-Target Pair
TargetAtrial natriuretic peptide receptor 1(Homo sapiens (Human))
The Weizmann Institute Of Science
Curated by ChEMBL
The Weizmann Institute Of Science
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Displacement of [125I]ANP from NPR-A expressed in HeLa cells after 3 hrs by gamma countingMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 2(Homo sapiens (Human))
The Weizmann Institute Of Science
Curated by ChEMBL
The Weizmann Institute Of Science
Curated by ChEMBL
Affinity DataIC50: 8.10nMAssay Description:Displacement of [125I-Tyr3]octreotide from sst2 receptor expressed in rat AR4-2J cellsMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 2(Homo sapiens (Human))
The Weizmann Institute Of Science
Curated by ChEMBL
The Weizmann Institute Of Science
Curated by ChEMBL
Affinity DataIC50: 8.10nMAssay Description:Displacement of [125I-Tyr3]octreotide from sst2 receptor expressed in rat AR4-2J cellsMore data for this Ligand-Target Pair
TargetAtrial natriuretic peptide receptor 1(Homo sapiens (Human))
The Weizmann Institute Of Science
Curated by ChEMBL
The Weizmann Institute Of Science
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Displacement of [125I]ANP from NPR-A expressed in HeLa cells after 3 hrs by gamma countingMore data for this Ligand-Target Pair
TargetAtrial natriuretic peptide receptor 1(Homo sapiens (Human))
The Weizmann Institute Of Science
Curated by ChEMBL
The Weizmann Institute Of Science
Curated by ChEMBL
Affinity DataIC50: 240nMAssay Description:Displacement of [125I]ANP from NPR-A expressed in HeLa cells after 3 hrs by gamma countingMore data for this Ligand-Target Pair
Affinity DataIC50: 370nMAssay Description:Inhibition of human CK2alpha using RRRDDDSDDD peptide as substrate preincubated for 40 mins and measured after 70 mins in the presence of ATP by ADP ...More data for this Ligand-Target Pair
TargetSomatostatin receptor type 2(Homo sapiens (Human))
The Weizmann Institute Of Science
Curated by ChEMBL
The Weizmann Institute Of Science
Curated by ChEMBL
Affinity DataIC50: >600nMAssay Description:Displacement of [125I-Tyr3]octreotide from sst2 receptor expressed in rat AR4-2J cellsMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Tufts University School Of Medicine
Curated by ChEMBL
Tufts University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:TP_TRANSPORTER: inhibition of Rhodamine 123 efflux in Caco-2 cellsMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Tufts University School Of Medicine
Curated by ChEMBL
Tufts University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 4.70E+3nMAssay Description:TP_TRANSPORTER: inhibition of Rhodamine 123 transepithelial transport (basal to apical) (R123: 5 uM) in Caco-2 cellsMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Tufts University School Of Medicine
Curated by ChEMBL
Tufts University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 7.50E+3nMAssay Description:TP_TRANSPORTER: inhibition of Rhodamine 123 transepithelial transport (basal to apical) (Rhodamine 123: 5 uM) in Caco-2 cellsMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Tufts University School Of Medicine
Curated by ChEMBL
Tufts University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 2.90E+4nMAssay Description:TP_TRANSPORTER: transepithelial transport of Rhodamine 123 (basal to apical) in Caco-2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of N-terminal GST-tagged human CK1epsilon (1 to 348 residues) expressed in baculovirus expression system in presence of peptide substrate ...More data for this Ligand-Target Pair