BindingDB PrimarySearch_ki

Found 242 with Last Name = 'christ' and Initial = 'cd'

N-lysine methyltransferase SMYD2(Homo sapiens (Human))
Bayer Pharma

Curated by ChEMBL

PNG

BDBM50180955(CHEMBL3818617)

Ki: 8nMAssay Description:Competitive inhibition of full length 6xHis-tagged SMYD2 (unknown origin) expressed in Escherichia coli using varying levels of Btn-Ahx-GSRAHSSHLKSKK...More data for this Ligand-Target Pair

PDB Reactome pathway
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N-lysine methyltransferase SMYD2(Homo sapiens (Human))
Bayer Pharma

Curated by ChEMBL

PNG

BDBM50180955(CHEMBL3818617)

Ki: 28nMAssay Description:Uncompetitive inhibition of full length 6xHis-tagged SMYD2 (unknown origin) expressed in Escherichia coli using fixed levels of Btn-Ahx-GSRAHSSHLKSKK...More data for this Ligand-Target Pair

PDB Reactome pathway
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Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha(Homo sapiens)TBA

PNG

BDBM50611048(BAY-091)

IC50: 1nMAssay Description:Inhibition of recombinant full length His-tagged PIP4K2A (unknown origin) expressed in sf21 cells assessed as reduction in ADP production preincubate...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Details PubMed PDB

3D Structure (crystal)

Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha(Homo sapiens)TBA

PNG

BDBM50611049(CHEMBL5280127)

IC50: 2nMAssay Description:Inhibition of recombinant full length His-tagged PIP4K2A (unknown origin) expressed in sf21 cells assessed as reduction in ADP production preincubate...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
GoogleScholar

Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha(Homo sapiens)TBA

PNG

BDBM50611049(CHEMBL5280127)

IC50: 3nMAssay Description:Inhibition of recombinant full length His-tagged PIP4K2A (unknown origin) expressed in sf21 cells assessed as reduction in ADP production preincubate...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha(Homo sapiens)TBA

PNG

BDBM50611048(BAY-091)

IC50: 3nMAssay Description:Inhibition of recombinant full length His-tagged PIP4K2A (unknown origin) expressed in sf21 cells assessed as reduction in ADP production preincubate...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Details PubMed PDB

3D Structure (crystal)

Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha(Homo sapiens)TBA

PNG

BDBM50610997(CHEMBL5276719)

IC50: 5nMAssay Description:Inhibition of recombinant full length His-tagged PIP4K2A (unknown origin) expressed in sf21 cells assessed as reduction in ADP production preincubate...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
GoogleScholar

Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha(Homo sapiens)TBA

PNG

BDBM50610997(CHEMBL5276719)

IC50: 5.5nMAssay Description:Inhibition of recombinant full length His-tagged PIP4K2A (unknown origin) expressed in sf21 cells assessed as reduction in ADP production preincubate...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
GoogleScholar

Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha(Homo sapiens)TBA

PNG

BDBM50611050(CHEMBL5270765)

IC50: 7nMAssay Description:Inhibition of recombinant full length His-tagged PIP4K2A (unknown origin) expressed in sf21 cells assessed as reduction in ADP production preincubate...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha(Homo sapiens)TBA

PNG

BDBM50611048(BAY-091)

IC50: 8nMAssay Description:Inhibition of recombinant full length His-tagged PIP4K2A (unknown origin) expressed in sf21 assessed as reduction in PI4,5P2 production preincubated ...More data for this Ligand-Target Pair

PDB Reactome pathway
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Details PubMed PDB

3D Structure (crystal)

Proteinase-activated receptor 1(Homo sapiens (Human))
Bayer Pharma

Curated by ChEMBL

PNG

BDBM50181506(CHEMBL3819038)

IC50: 10nMAssay Description:Antagonist activity at PAR1 (unknown origin)More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha(Homo sapiens)TBA

PNG

BDBM50611046(CHEMBL5290005)

IC50: 13nMAssay Description:Inhibition of recombinant full length His-tagged PIP4K2A (unknown origin) expressed in sf21 cells assessed as reduction in ADP production preincubate...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Details PubMed PDB

3D Structure (crystal)

Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha(Homo sapiens)TBA

PNG

BDBM50611049(CHEMBL5280127)

IC50: 14nMAssay Description:Inhibition of recombinant full length His-tagged PIP4K2A (unknown origin) expressed in sf21 assessed as reduction in PI4,5P2 production preincubated ...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha(Homo sapiens)TBA

PNG

BDBM50610996(CHEMBL5271652)

IC50: 14nMAssay Description:Inhibition of recombinant full length His-tagged PIP4K2A (unknown origin) expressed in sf21 cells assessed as reduction in ADP production preincubate...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
GoogleScholar

N-lysine methyltransferase SMYD2(Homo sapiens (Human))
Bayer Pharma

Curated by ChEMBL

PNG

BDBM50075102(CHEMBL3414623)

IC50: <15nMAssay Description:Inhibition of SMYD2 (unknown origin) expressed in Escherichia coli BL21 (DE3) using Biotinaminohexanoyl-GSRAHSSHLKSKKGQSTSRH as substrate after 75 mi...More data for this Ligand-Target Pair

PDB Reactome pathway
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3D Structure (crystal)

Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha(Homo sapiens)TBA

PNG

BDBM50611048(BAY-091)

IC50: 16nMAssay Description:Inhibition of recombinant full length His-tagged PIP4K2A (unknown origin) expressed in sf21 assessed as reduction in PI4,5P2 production preincubated ...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Details PubMed PDB

3D Structure (crystal)

Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha(Homo sapiens)TBA

PNG

BDBM50611047(CHEMBL5277824)

IC50: 19nMAssay Description:Inhibition of recombinant full length His-tagged PIP4K2A (unknown origin) expressed in sf21 cells assessed as reduction in ADP production preincubate...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
GoogleScholar

N-lysine methyltransferase SMYD2(Homo sapiens (Human))
Bayer Pharma

Curated by ChEMBL

PNG

BDBM50180967(CHEMBL3818487)

IC50: 19nMAssay Description:Inhibition of SMYD2 (unknown origin) using H4 as substrate after 2hrs in presence 3H-SAM of by scintillation proximity assayMore data for this Ligand-Target Pair

PDB Reactome pathway
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Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha(Homo sapiens)TBA

PNG

BDBM50611050(CHEMBL5270765)

IC50: 20nMAssay Description:Inhibition of recombinant full length His-tagged PIP4K2A (unknown origin) expressed in sf21 cells assessed as reduction in ADP production preincubate...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
GoogleScholar

Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha(Homo sapiens)TBA

PNG

BDBM50610997(CHEMBL5276719)

IC50: 27nMAssay Description:Inhibition of recombinant full length His-tagged PIP4K2A (unknown origin) expressed in sf21 assessed as reduction in PI4,5P2 production preincubated ...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
GoogleScholar

N-lysine methyltransferase SMYD2(Homo sapiens (Human))
Bayer Pharma

Curated by ChEMBL

PNG

BDBM50180955(CHEMBL3818617)

IC50: 27nMAssay Description:Inhibition of full length 6xHis-tagged SMYD2 (unknown origin) expressed in Escherichia coli using Btn-Ahx GSRAHSSHLKSKKGQSTSRH-amide as substrate aft...More data for this Ligand-Target Pair

PDB Reactome pathway
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Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha(Homo sapiens)TBA

PNG

BDBM50611049(CHEMBL5280127)

IC50: 29nMAssay Description:Inhibition of recombinant full length His-tagged PIP4K2A (unknown origin) expressed in sf21 assessed as reduction in PI4,5P2 production preincubated ...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
GoogleScholar

Proteinase-activated receptor 1(Homo sapiens (Human))
Bayer Pharma

Curated by ChEMBL

PNG

BDBM50181504(CHEMBL3818898)

IC50: 30nMAssay Description:Antagonist activity at PAR1 (unknown origin)More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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Proteinase-activated receptor 1(Homo sapiens (Human))
Bayer Pharma

Curated by ChEMBL

PNG

BDBM50181502(CHEMBL3818510)

IC50: 30nMAssay Description:Antagonist activity at PAR1 (unknown origin)More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha(Homo sapiens)TBA

PNG

BDBM50611013(CHEMBL5288492)

IC50: 30nMAssay Description:Inhibition of recombinant full length His-tagged PIP4K2A (unknown origin) expressed in sf21 cells assessed as reduction in ADP production preincubate...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
GoogleScholar

Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha(Homo sapiens)TBA

PNG

BDBM50611050(CHEMBL5270765)

IC50: 30nMAssay Description:Inhibition of recombinant full length His-tagged PIP4K2A (unknown origin) expressed in sf21 assessed as reduction in PI4,5P2 production preincubated ...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
GoogleScholar

Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha(Homo sapiens)TBA

PNG

BDBM50611020(CHEMBL5282226)

IC50: 37nMAssay Description:Inhibition of recombinant full length His-tagged PIP4K2A (unknown origin) expressed in sf21 cells assessed as reduction in ADP production preincubate...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
GoogleScholar

N-lysine methyltransferase SMYD2(Homo sapiens (Human))
Bayer Pharma

Curated by ChEMBL

PNG

BDBM50180973(CHEMBL3819284)

IC50: 38nMAssay Description:Inhibition of SMYD2 (unknown origin) using H4 as substrate after 2hrs in presence 3H-SAM of by scintillation proximity assayMore data for this Ligand-Target Pair

PDB Reactome pathway
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Proteinase-activated receptor 1(Homo sapiens (Human))
Bayer Pharma

Curated by ChEMBL

PNG

BDBM50181505(CHEMBL3819204)

IC50: 40nMAssay Description:Antagonist activity at PAR1 (unknown origin)More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha(Homo sapiens)TBA

PNG

BDBM50611012(CHEMBL5284796)

IC50: 40nMAssay Description:Inhibition of recombinant full length His-tagged PIP4K2A (unknown origin) expressed in sf21 cells assessed as reduction in ADP production preincubate...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha(Homo sapiens)TBA

PNG

BDBM50611023(CHEMBL5273876)

IC50: 42nMAssay Description:Inhibition of recombinant full length His-tagged PIP4K2A (unknown origin) expressed in sf21 cells assessed as reduction in ADP production preincubate...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
GoogleScholar

N-lysine methyltransferase SMYD2(Homo sapiens (Human))
Bayer Pharma

Curated by ChEMBL

PNG

BDBM50180968(CHEMBL3818080)

IC50: 44nMAssay Description:Inhibition of SMYD2 (unknown origin) using H4 as substrate after 2hrs in presence 3H-SAM of by scintillation proximity assayMore data for this Ligand-Target Pair

PDB Reactome pathway
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Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha(Homo sapiens)TBA

PNG

BDBM50611043(CHEMBL5272762)

IC50: 47nMAssay Description:Inhibition of recombinant full length His-tagged PIP4K2A (unknown origin) expressed in sf21 cells assessed as reduction in ADP production preincubate...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
GoogleScholar

Proteinase-activated receptor 1(Homo sapiens (Human))
Bayer Pharma

Curated by ChEMBL

PNG

BDBM50181513(CHEMBL3819237)

IC50: 50nMAssay Description:Antagonist activity at PAR1 (unknown origin)More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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N-lysine methyltransferase SMYD2(Homo sapiens (Human))
Bayer Pharma

Curated by ChEMBL

PNG

BDBM50180971(CHEMBL3818322)

IC50: 50nMAssay Description:Inhibition of SMYD2 (unknown origin) using H4 as substrate after 2hrs in presence 3H-SAM of by scintillation proximity assayMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Details Article PubMed

Proteinase-activated receptor 1(Homo sapiens (Human))
Bayer Pharma

Curated by ChEMBL

PNG

BDBM50181507(CHEMBL3818421)

IC50: 50nMAssay Description:Antagonist activity at PAR1 (unknown origin)More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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B.MOAD DrugBank antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha(Homo sapiens)TBA

PNG

BDBM50610996(CHEMBL5271652)

IC50: 51nMAssay Description:Inhibition of recombinant full length His-tagged PIP4K2A (unknown origin) expressed in sf21 cells assessed as reduction in ADP production preincubate...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
GoogleScholar

Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha(Homo sapiens)TBA

PNG

BDBM50610997(CHEMBL5276719)

IC50: 59nMAssay Description:Inhibition of recombinant full length His-tagged PIP4K2A (unknown origin) expressed in sf21 cells assessed as reduction in ADP production preincubate...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
GoogleScholar

Proteinase-activated receptor 1(Homo sapiens (Human))
Bayer Pharma

Curated by ChEMBL

PNG

BDBM50181509(CHEMBL3817930)

IC50: 60nMAssay Description:Antagonist activity at PAR1 (unknown origin)More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Details Article PubMed

N-lysine methyltransferase SMYD2(Homo sapiens (Human))
Bayer Pharma

Curated by ChEMBL

PNG

BDBM50180955(CHEMBL3818617)

IC50: 60nMAssay Description:Inhibition of N-terminal 2xc-myc-tagged human SMYD2 transfected in human MDA-MB-231 cells assessed as reduction in AHNAK methylation after 72 hrs by ...More data for this Ligand-Target Pair

PDB Reactome pathway
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Proteinase-activated receptor 1(Homo sapiens (Human))
Bayer Pharma

Curated by ChEMBL

PNG

BDBM50181511(CHEMBL3819343)

IC50: 60nMAssay Description:Antagonist activity at PAR1 (unknown origin)More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
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Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha(Homo sapiens)TBA

PNG

BDBM50611033(CHEMBL5265849)

IC50: 61nMAssay Description:Inhibition of recombinant full length His-tagged PIP4K2A (unknown origin) expressed in sf21 cells assessed as reduction in ADP production preincubate...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
GoogleScholar

Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha(Homo sapiens)TBA

PNG

BDBM50610998(CHEMBL5274835)

IC50: 66nMAssay Description:Inhibition of recombinant full length His-tagged PIP4K2A (unknown origin) expressed in sf21 cells assessed as reduction in ADP production preincubate...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
GoogleScholar

Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha(Homo sapiens)TBA

PNG

BDBM50611046(CHEMBL5290005)

IC50: 69nMAssay Description:Inhibition of recombinant full length His-tagged PIP4K2A (unknown origin) expressed in sf21 cells assessed as reduction in ADP production preincubate...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
GoogleScholar

Details PubMed PDB

3D Structure (crystal)

Proteinase-activated receptor 1(Homo sapiens (Human))
Bayer Pharma

Curated by ChEMBL

PNG

BDBM50181512(CHEMBL3819277 | US10023539, Example WO 2006/07235...)

IC50: 70nMAssay Description:Antagonist activity at PAR1 (unknown origin)More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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N-lysine methyltransferase SMYD2(Homo sapiens (Human))
Bayer Pharma

Curated by ChEMBL

PNG

BDBM50180970(CHEMBL3819554)

IC50: 71nMAssay Description:Inhibition of SMYD2 (unknown origin) using H4 as substrate after 2hrs in presence 3H-SAM of by scintillation proximity assayMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha(Homo sapiens)TBA

PNG

BDBM50611047(CHEMBL5277824)

IC50: 71nMAssay Description:Inhibition of recombinant full length His-tagged PIP4K2A (unknown origin) expressed in sf21 cells assessed as reduction in ADP production preincubate...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
GoogleScholar

Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha(Homo sapiens)TBA

PNG

BDBM50611032(CHEMBL5275703)

IC50: 74nMAssay Description:Inhibition of recombinant full length His-tagged PIP4K2A (unknown origin) expressed in sf21 cells assessed as reduction in ADP production preincubate...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
GoogleScholar

N-lysine methyltransferase SMYD2(Homo sapiens (Human))
Bayer Pharma

Curated by ChEMBL

PNG

BDBM50180974(CHEMBL3818092 | US10023539, Example 33.2)

IC50: 80nMAssay Description:Inhibition of SMYD2 (unknown origin) using H4 as substrate after 2hrs in presence 3H-SAM of by scintillation proximity assayMore data for this Ligand-Target Pair

PDB Reactome pathway
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Proteinase-activated receptor 1(Homo sapiens (Human))
Bayer Pharma

Curated by ChEMBL

PNG

BDBM50181510(CHEMBL3818750)

IC50: 80nMAssay Description:Antagonist activity at PAR1 (unknown origin)More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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