Compile Data Set for Download or QSAR
maximum 50k data
Found 46 with Last Name = 'kishore kumar' and Initial = 'm'
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50177100(3-Cycloheptyl-9-dimethylamino-3H-pyrido[3',2':4,5]...)
Affinity DataIC50:  1nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50177053(9-Dimethylamino-3-(4-ethyl-phenyl)-3H-pyrido[3',2'...)
Affinity DataIC50:  3nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50177063(3-(4-Bromo-phenyl)-9-dimethylamino-3H-pyrido[3',2'...)
Affinity DataIC50:  4nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50177097(9-Dimethylamino-3-p-tolyl-3H-pyrido[3',2':4,5]thie...)
Affinity DataIC50:  5nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50177085(3-Cyclopentyl-9-dimethylamino-3H-pyrido[3',2':4,5]...)
Affinity DataIC50:  5nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50177055(9-Dimethylamino-3-(3-ethyl-phenyl)-3H-pyrido[3',2'...)
Affinity DataIC50:  9nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50177080(3-azepan-1-yl-9-dimethylamino-3H-pyrido[3',2':4,5]...)
Affinity DataIC50:  10nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50177059(3-Cyclooctyl-9-dimethylamino-3H-pyrido[3',2':4,5]t...)
Affinity DataIC50:  13nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50177076(3-(4-Chloro-phenyl)-9-dimethylamino-3H-pyrido[3',2...)
Affinity DataIC50:  16nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50177065(9-Dimethylamino-3-(2,4-dimethyl-phenyl)-3H-pyrido[...)
Affinity DataIC50:  17nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50177079(9-dimethylamino-3-phenyl-3H-pyrido[3',2':4,5]thien...)
Affinity DataIC50:  20nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50177078(9-Dimethylamino-3-(4-fluoro-phenyl)-3H-pyrido[3',2...)
Affinity DataIC50:  23nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50177098(3-Cyclopentylmethyl-9-dimethylamino-3H-pyrido[3',2...)
Affinity DataIC50:  26nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50177057(9-Dimethylamino-3-(4-trifluoromethyl-phenyl)-3H-py...)
Affinity DataIC50:  32nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50177074(9-(Ethyl-methyl-amino)-3-(4-ethyl-phenyl)-3H-pyrid...)
Affinity DataIC50:  37nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50177084(9-Dimethylamino-3-(6-methoxy-pyridin-3-yl)-3H-pyri...)
Affinity DataIC50:  39nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50177061(9-Cyclopropylamino-3-(4-ethyl-phenyl)-3H-pyrido[3'...)
Affinity DataIC50:  41nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50177054(9-(1'-cyanomethylamino)-3-(4'-ethylphenyl)-3H-5-th...)
Affinity DataIC50:  43nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50177093(9-Dimethylamino-3-(4-ethyl-phenyl)-2-methyl-3H-pyr...)
Affinity DataIC50:  44nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50177081(3-(2,4-Dichloro-phenyl)-9-dimethylamino-3H-pyrido[...)
Affinity DataIC50:  45nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50177067(9-Dimethylamino-3-(2-hydroxy-phenyl)-3H-pyrido[3',...)
Affinity DataIC50:  50nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50177070(3-Cyclohexyl-9-dimethylamino-3H-pyrido[3',2':4,5]t...)
Affinity DataIC50:  50nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50190237(3-(4-Ethyl-phenyl)-9-[methyl-(2-pyridin-2-yl-ethyl...)
Affinity DataIC50:  52nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50177083(3-(4-ethylphenyl)-9-[(2-methoxyethyl)(methyl)amino...)
Affinity DataIC50:  71nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50177068(3-Adamantan-1-yl-9-dimethylamino-3H-pyrido[3',2':4...)
Affinity DataIC50:  76nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50177095(9-Dimethylamino-2-ethyl-3-(4-ethyl-phenyl)-3H-pyri...)
Affinity DataIC50:  84nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50177066(3-(4-Cyclopropyl-phenyl)-9-dimethylamino-3H-pyrido...)
Affinity DataIC50:  87nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50177086(3-(4-Ethyl-phenyl)-9-methylamino-3H-pyrido[3',2':4...)
Affinity DataIC50:  98nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50177071(3-(4-Ethyl-phenyl)-9-(2,2,2-trifluoro-ethylamino)-...)
Affinity DataIC50:  99nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50177073(2-Butyl-9-dimethylamino-3-(4-ethyl-phenyl)-3H-pyri...)
Affinity DataIC50:  101nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50177058(9-Azetidin-1-yl-3-(4-ethyl-phenyl)-3H-pyrido[3',2'...)
Affinity DataIC50:  113nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50245682(9-Dimethylamino-3-(1H-indol-6-yl)-3H-pyrido[3',2':...)
Affinity DataIC50:  122nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50177094(9-Dimethylamino-3-(2-methyl-cyclohexyl)-3H-pyrido[...)
Affinity DataIC50:  130nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50177075(3-Cyclohexylmethyl-9-dimethylamino-3H-pyrido[3',2'...)
Affinity DataIC50:  139nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50177072(9-Dimethylamino-3-(4-methyl-cyclohexyl)-3H-pyrido[...)
Affinity DataIC50:  140nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50245379(3-cycloheptyl-9-(dimethylnitroryl)pyrido[3',2':4,5...)
Affinity DataIC50:  167nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50177060(3-Cyclobutyl-9-dimethylamino-3H-pyrido[3',2':4,5]t...)
Affinity DataIC50:  167nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50177102(9-Dimethylamino-3-(4-propyl-phenyl)-3H-pyrido[3',2...)
Affinity DataIC50:  180nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50177056(9-Dimethylamino-3-(2-ethyl-phenyl)-3H-pyrido[3',2'...)
Affinity DataIC50:  251nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50177064(3-Benzyl-9-dimethylamino-3H-pyrido[3',2':4,5]thien...)
Affinity DataIC50:  281nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50177069(9-(N,N,-dimethyl-N-oxyamino)-3-(4'-ethylphenyl)-3H...)
Affinity DataIC50:  306nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50177077(9-Dimethylamino-3-(1-ethyl-propyl)-3H-pyrido[3',2'...)
Affinity DataIC50:  335nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50177092(9-Dimethylamino-3-(4-isopropyl-phenyl)-3H-pyrido[3...)
Affinity DataIC50:  407nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50177099(9-Dimethylamino-3-(3-methyl-cyclohexyl)-3H-pyrido[...)
Affinity DataIC50:  482nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50177101(3-Cyclopropyl-9-dimethylamino-3H-pyrido[3',2':4,5]...)
Affinity DataIC50:  632nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50177091(3-(4-tert-Butyl-phenyl)-9-dimethylamino-3H-pyrido[...)
Affinity DataIC50:  8.50E+3nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed