Affinity DataKi: 0.0410nMAssay Description:Inhibition of human plasmin using Ac-RM(O2)YR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0510nMAssay Description:Inhibition of human plasmin using Ac-RM(O2)YR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 0.140nMAssay Description:Inhibition of human plasmin using Ac-RM(O2)YR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Inhibition of trypsin (unknown origin) using Bz-FVRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 0.210nMAssay Description:Inhibition of human plasmin using Ac-RM(O2)YR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 0.450nMAssay Description:Inhibition of human plasmin using Ac-RM(O2)YR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 0.610nMAssay Description:Inhibition of human plasmin using Ac-RM(O2)YR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 0.660nMAssay Description:Inhibition of human plasmin using Ac-RM(O2)YR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 0.660nMAssay Description:Inhibition of human plasmin using Ac-RM(O2)YR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Inhibition of human plasmin using Ac-RM(O2)YR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Inhibition of human plasmin using Ac-RM(O2)YR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Inhibition of human plasmin using Ac-RM(O2)YR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of human plasmin using Ac-RM(O2)YR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Inhibition of human plasmin using Ac-RM(O2)YR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:Inhibition of human plasmin using Ac-RM(O2)YR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 6.90nMAssay Description:Inhibition of trypsin (unknown origin) using Bz-FVRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 8.30nMAssay Description:Inhibition of human plasmin using Ac-RM(O2)YR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Inhibition of bovine cationic trypsin using Bz-FVR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Inhibition of human plasmin using Ac-RM(O2)YR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Inhibition of human plasmin using Ac-RM(O2)YR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Inhibition of bovine cationic trypsin using Bz-FVR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Inhibition of plasmin (unknown origin) using Ac-RM(O2)YRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Inhibition of factor 12a (unknown origin) using Ac-QRFRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Inhibition of human plasmin using Ac-RM(O2)YR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 160nMAssay Description:Inhibition of bovine cationic trypsin using Bz-FVR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 180nMAssay Description:Inhibition of factor 12a (unknown origin) using Ac-QRFRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Inhibition of recombinant human matriptase catalytic domain pre-incubated for 60 mins before Boc QAR-AMC substrate additionMore data for this Ligand-Target Pair
Affinity DataKi: 270nMAssay Description:Inhibition of plasmin (unknown origin) using Ac-RM(O2)YRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 360nMAssay Description:Inhibition of factor 10a (unknown origin) using Ac-QRSRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 460nMAssay Description:Inhibition of factor 10a (unknown origin) using Ac-QRSRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 490nMAssay Description:Inhibition of factor 12a (unknown origin) using Ac-QRFRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 510nMAssay Description:Inhibition of factor 12a (unknown origin) using Ac-QRFRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 570nMAssay Description:Inhibition of factor 10a (unknown origin) using Ac-QRSRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 750nMAssay Description:Inhibition of factor 12a (unknown origin) using Ac-QRFRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.50E+3nMAssay Description:Inhibition of plasmin (unknown origin) using Ac-RM(O2)YRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 2.16E+3nMAssay Description:Inhibition of factor 12a (unknown origin) using Ac-QRFRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 2.24E+3nMAssay Description:Inhibition of trypsin (unknown origin) using Bz-FVRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 2.39E+3nMAssay Description:Inhibition of factor 12a (unknown origin) using Ac-QRFRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 4.54E+3nMAssay Description:Inhibition of plasmin (unknown origin) using Ac-RM(O2)YRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 6.24E+3nMAssay Description:Inhibition of trypsin (unknown origin) using Bz-FVRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 7.80E+3nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate after 30 minsMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of uPA (unknown origin) incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
TargetTissue-type plasminogen activator(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of tPA (unknown origin) incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
TargetTissue-type plasminogen activator(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of tPA (unknown origin) incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of factor 11a (unknown origin) using Bz-FVRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human plasma kallikrein using Ac-RM(O2)YRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of uPA (unknown origin) incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of factor 9a (unknown origin) using Ac-QGRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of factor 11a (unknown origin) using Bz-FVRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of factor 9a (unknown origin) using Ac-QGRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair