Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Homo sapiens (Human))
Universidad Nacional AutóNoma De MéXico
Curated by ChEMBL
Universidad Nacional AutóNoma De MéXico
Curated by ChEMBL
Affinity DataKi: 0.900nMAssay Description:Inhibitory constant against HMG-CoA reductaseMore data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Homo sapiens (Human))
Universidad Nacional AutóNoma De MéXico
Curated by ChEMBL
Universidad Nacional AutóNoma De MéXico
Curated by ChEMBL
Affinity DataKi: 2.60nMAssay Description:Inhibitory constant against HMG-CoA reductaseMore data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Homo sapiens (Human))
Universidad Nacional AutóNoma De MéXico
Curated by ChEMBL
Universidad Nacional AutóNoma De MéXico
Curated by ChEMBL
Affinity DataKi: 23.5nMAssay Description:Inhibitory constant against HMG-CoA reductaseMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Universidad Aut£Noma Del Estado De Morelos
Curated by ChEMBL
Universidad Aut£Noma Del Estado De Morelos
Curated by ChEMBL
Affinity DataKi: 3.40E+3nMAssay Description:Mixed type inhibition of human recombinant PTP-1B expressed in Escherichia coli TB1 using p-nitrophenyl phosphate as substrateMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Universidad Aut£Noma Del Estado De Morelos
Curated by ChEMBL
Universidad Aut£Noma Del Estado De Morelos
Curated by ChEMBL
Affinity DataKi: 6.00E+3nMAssay Description:Mixed type inhibition of human recombinant PTP-1B expressed in Escherichia coli TB1 using p-nitrophenyl phosphate as substrateMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Universidad Aut£Noma Del Estado De Morelos
Curated by ChEMBL
Universidad Aut£Noma Del Estado De Morelos
Curated by ChEMBL
Affinity DataKi: 6.20E+3nMAssay Description:Mixed-type inhibition of human recombinant GST-tagged PTP1B expressed in Escherichia coli TB1 cells using p-NPP as substrate by double reciprocal plo...More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Universidad Aut£Noma Del Estado De Morelos
Curated by ChEMBL
Universidad Aut£Noma Del Estado De Morelos
Curated by ChEMBL
Affinity DataKi: 7.10E+3nMAssay Description:Inhibition of human recombinant PTP1B expressed in Escherichia coli TB1 by double reciprocal plot analysisMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Universidad Aut£Noma Del Estado De Morelos
Curated by ChEMBL
Universidad Aut£Noma Del Estado De Morelos
Curated by ChEMBL
Affinity DataKi: 7.10E+3nMAssay Description:Non-competitive inhibition of human recombinant PTP-1B expressed in Escherichia coli TB1 using p-nitrophenyl phosphate as substrateMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Universidad Aut£Noma Del Estado De Morelos
Curated by ChEMBL
Universidad Aut£Noma Del Estado De Morelos
Curated by ChEMBL
Affinity DataKi: 7.90E+3nMAssay Description:Mixed-type inhibition of human recombinant GST-tagged PTP1B expressed in Escherichia coli TB1 cells using p-NPP as substrate by double reciprocal plo...More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Universidad Aut£Noma Del Estado De Morelos
Curated by ChEMBL
Universidad Aut£Noma Del Estado De Morelos
Curated by ChEMBL
Affinity DataKi: 7.90E+3nMAssay Description:Mixed-type inhibition of human recombinant GST-tagged PTP1B expressed in Escherichia coli TB1 cells using p-NPP as substrate by double reciprocal plo...More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Universidad Aut£Noma Del Estado De Morelos
Curated by ChEMBL
Universidad Aut£Noma Del Estado De Morelos
Curated by ChEMBL
Affinity DataKi: 8.00E+3nMAssay Description:Mixed type inhibition of human recombinant PTP-1B expressed in Escherichia coli TB1 using p-nitrophenyl phosphate as substrateMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Universidad Aut£Noma Del Estado De Morelos
Curated by ChEMBL
Universidad Aut£Noma Del Estado De Morelos
Curated by ChEMBL
Affinity DataKi: 2.04E+4nMAssay Description:Inhibition of human recombinant PTP1B expressed in Escherichia coli TB1 by double reciprocal plot analysisMore data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Homo sapiens (Human))
Universidad Nacional AutóNoma De MéXico
Curated by ChEMBL
Universidad Nacional AutóNoma De MéXico
Curated by ChEMBL
Affinity DataKi: 6.80E+4nMAssay Description:Inhibitory constant against HMG-CoA reductase with alpha asaroneMore data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Homo sapiens (Human))
Universidad Nacional AutóNoma De MéXico
Curated by ChEMBL
Universidad Nacional AutóNoma De MéXico
Curated by ChEMBL
Affinity DataKi: 7.10E+4nMAssay Description:Inhibitory constant against HMG-CoA reductase with alpha asaroneMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 1.70nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 1.70nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 3.60nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair