Affinity DataIC50: 9nMAssay Description:Inhibition of IL-17A (unknown origin) measured by FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: <100nMAssay Description:Inhibition of IL-17A (unknown origin) by ELISA IIMore data for this Ligand-Target Pair
Affinity DataIC50: <100nMAssay Description:Inhibition of IL-17A (unknown origin) by ELISA IIMore data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Inhibition of IL-17A (unknown origin) measured by AlphaLISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Inhibition of IL-17A (unknown origin) measured by AlphaLISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition of human recombinant CYP3A4 using DEF as substrate preincubated for 5 to 10 mins before substrate additionMore data for this Ligand-Target Pair
Affinity DataIC50: 700nMAssay Description:Inhibition of human recombinant CYP3A4 using DEF as substrate preincubated for 5 to 10 mins before substrate additionMore data for this Ligand-Target Pair
Affinity DataIC50: 700nMAssay Description:Inhibition of human recombinant CYP3A4 using DEF as substrate preincubated for 5 to 10 mins before substrate additionMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human recombinant CYP3A4 using DEF as substrate preincubated for 5 to 10 mins before substrate additionMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human recombinant CYP3A4 using DEF as substrate preincubated for 5 to 10 mins before substrate additionMore data for this Ligand-Target Pair
Affinity DataIC50: 1.14E+3nMAssay Description:Inhibition of IL-17A (unknown origin) measured by FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.33E+3nMAssay Description:Inhibition of human recombinant CYP3A4 using DEF as substrate preincubated for 5 to 10 mins before substrate additionMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human recombinant CYP3A4 using DEF as substrate preincubated for 5 to 10 mins before substrate additionMore data for this Ligand-Target Pair
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of human recombinant CYP3A4 using 7-BQ as substrate preincubated for 5 to 10 mins before substrate additionMore data for this Ligand-Target Pair
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of human recombinant CYP3A4 using 7-BQ as substrate preincubated for 5 to 10 mins before substrate additionMore data for this Ligand-Target Pair
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of human recombinant CYP3A4 using 7-BQ as substrate preincubated for 5 to 10 mins before substrate additionMore data for this Ligand-Target Pair
Affinity DataIC50: 7.80E+3nMAssay Description:Inhibition of human recombinant CYP3A4 using DEF as substrate preincubated for 5 to 10 mins before substrate additionMore data for this Ligand-Target Pair
Affinity DataIC50: 7.90E+3nMAssay Description:Inhibition of human recombinant CYP3A4 using DEF as substrate preincubated for 5 to 10 mins before substrate additionMore data for this Ligand-Target Pair
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of human recombinant CYP3A4 using 7-BQ as substrate preincubated for 5 to 10 mins before substrate additionMore data for this Ligand-Target Pair
Affinity DataIC50: 9.80E+3nMAssay Description:Inhibition of human recombinant CYP3A4 using 7-BQ as substrate preincubated for 5 to 10 mins before substrate additionMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CYP3A4 using 7-BQ as substrate preincubated for 5 to 10 mins before substrate additionMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CYP3A4 using 7-BQ as substrate preincubated for 5 to 10 mins before substrate additionMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CYP3A4 using 7-BQ as substrate preincubated for 5 to 10 mins before substrate additionMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CYP3A4 using DEF as substrate preincubated for 5 to 10 mins before substrate additionMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Fidelta
Curated by ChEMBL
Fidelta
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human ERG by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Fidelta
Curated by ChEMBL
Fidelta
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human ERG by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Fidelta
Curated by ChEMBL
Fidelta
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human ERG by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Fidelta
Curated by ChEMBL
Fidelta
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human ERG by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CYP3A4 using 7-BQ as substrate preincubated for 5 to 10 mins before substrate additionMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CYP3A4 using 7-BQ as substrate preincubated for 5 to 10 mins before substrate additionMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CYP3A4 using 7-BQ as substrate preincubated for 5 to 10 mins before substrate additionMore data for this Ligand-Target Pair
Affinity DataEC50: 90nMAssay Description:Binding affinity to glucocorticoid receptor (unknown origin) by fluorescence polarization competitive binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: >2.50E+4nMAssay Description:Displacement of [3H]-dexamethasone human glucocorticoid receptor alpha expressed in 293 MSR cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataEC50: 910nMAssay Description:Binding affinity to glucocorticoid receptor (unknown origin) by fluorescence polarization competitive binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: >2.50E+4nMAssay Description:Displacement of [3H]-dexamethasone human glucocorticoid receptor alpha expressed in 293 MSR cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Binding affinity to glucocorticoid receptor (unknown origin) by fluorescence polarization competitive binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: >2.50E+4nMAssay Description:Displacement of [3H]-dexamethasone human glucocorticoid receptor alpha expressed in 293 MSR cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataEC50: 1.44E+3nMAssay Description:Binding affinity to glucocorticoid receptor (unknown origin) by fluorescence polarization competitive binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 9.70nMAssay Description:Inhibition of glucocorticoid receptor in human H13 cells assessed as inhibition of glucocorticoid-induced cell proliferation after 3 hrs by [3H]-thym...More data for this Ligand-Target Pair
Affinity DataEC50: 13nMAssay Description:Displacement of [3H]-dexamethasone human glucocorticoid receptor alpha expressed in 293 MSR cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataEC50: 3.70nMAssay Description:Binding affinity to glucocorticoid receptor (unknown origin) by fluorescence polarization competitive binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Inhibition of glucocorticoid receptor in human H13 cells assessed as inhibition of glucocorticoid-induced cell proliferation after 3 hrs by [3H]-thym...More data for this Ligand-Target Pair
Affinity DataEC50: 430nMAssay Description:Displacement of [3H]-dexamethasone human glucocorticoid receptor alpha expressed in 293 MSR cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataEC50: 4.16E+3nMAssay Description:Binding affinity to glucocorticoid receptor (unknown origin) by fluorescence polarization competitive binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.30E+4nMAssay Description:Displacement of [3H]-dexamethasone human glucocorticoid receptor alpha expressed in 293 MSR cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataEC50: 2.09E+3nMAssay Description:Binding affinity to glucocorticoid receptor (unknown origin) by fluorescence polarization competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKd: <500nMAssay Description:Binding affinity to IL-17A (unknown origin) measured by SPR assayMore data for this Ligand-Target Pair
Affinity DataKd: <500nMAssay Description:Binding affinity to IL-17A (unknown origin) measured by SPR assayMore data for this Ligand-Target Pair
Affinity DataKd: <660nMAssay Description:Binding affinity to IL-17A (unknown origin) measured by SPR assayMore data for this Ligand-Target Pair
Affinity DataKd: <141nMAssay Description:Binding affinity to IL-17A (unknown origin) measured by SPR assayMore data for this Ligand-Target Pair