Affinity DataIC50: 0.180nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Ghent University
Curated by ChEMBL
Ghent University
Curated by ChEMBL
Affinity DataIC50: 3.5nMAssay Description:Inhibition of human KDR using and Ulight-CAGAGAIETDKEYYTVKD as substrate after 1 hr by FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 220nMAssay Description:Inhibition of rabbit skeletal muscle myosin 2More data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibition of rabbit skeletal muscle myosin 2More data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization assessed as microtubule assembly after 15 mins by DAPI stainingMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of pig beta cardiac myosin 2 by NADH-coupled spectrophotometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of CYP1A2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of chicken non-muscle myosin 2b by NADH-coupled spectrophotometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of Dictyostelium discoideum myosin 2 ATPase activityMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of Dictyostelium discoideum myosin 2 ATPase activity by NADH-coupled assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of mouse non-muscle myosin 2cMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of human non-muscle myosin 2aMore data for this Ligand-Target Pair
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of human non-muscle myosin 2bMore data for this Ligand-Target Pair
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of RLC-phosphorylated Dictyostelium discoideum myosin 2 ATPase activity by NADH-coupled spectrophotometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of Dictyostelium discoideum myosin 2 ATPase activity by NADH-coupled assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.80E+4nMAssay Description:Inhibition of human myosin 2a ATPase activityMore data for this Ligand-Target Pair
Affinity DataIC50: 8.30E+4nMAssay Description:Inhibition of dephosphorylated Acanthamoeba non muscle myosin 2 by NADH-coupled spectrophotometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human myosin 15 by NADH-coupled spectrophotometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: >1.50E+5nMAssay Description:Inhibition of bovine myosin x by NADH-coupled spectrophotometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: >1.50E+5nMAssay Description:Inhibition of mouse myosin 5a by NADH-coupled spectrophotometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: >1.50E+5nMAssay Description:Inhibition of rat myosin 1b by NADH-coupled spectrophotometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: >1.50E+5nMAssay Description:Inhibition of dephosphorylated Acanthamoeba muscle myosin 1c by NADH-coupled spectrophotometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of fruit fly non-muscle myosin 2More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Ghent University
Curated by ChEMBL
Ghent University
Curated by ChEMBL
Affinity DataEC50: 25nMAssay Description:Inhibition of human ERG assessed as reduction of tail currentMore data for this Ligand-Target Pair