Affinity DataIC50: 4.30nMAssay Description:Tested for Oxidosqualene-lanosterol cyclase inhibition in T. bruceiMore data for this Ligand-Target Pair
Affinity DataIC50: 4.60nMAssay Description:Tested for Oxidosqualene-lanosterol cyclase inhibition in P. cariniiMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Tested for Oxidosqualene-lanosterol cyclase inhibition in T. bruceiMore data for this Ligand-Target Pair
Affinity DataIC50: 49nMAssay Description:Tested for Oxidosqualene-lanosterol cyclase inhibition in ratMore data for this Ligand-Target Pair
Affinity DataIC50: 71nMAssay Description:Tested for Oxidosqualene-lanosterol cyclase inhibition in T. cruziMore data for this Ligand-Target Pair
Affinity DataIC50: 92nMAssay Description:Tested for Oxidosqualene-lanosterol cyclase inhibition in P. cariniiMore data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Tested for Oxidosqualene-lanosterol cyclase inhibition in ratMore data for this Ligand-Target Pair
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: 260nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
Affinity DataIC50: 280nMAssay Description:Tested for Oxidosqualene-lanosterol cyclase inhibition in T. bruceiMore data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Tested for Oxidosqualene-lanosterol cyclase inhibition in T. cruziMore data for this Ligand-Target Pair
Affinity DataIC50: 750nMAssay Description:Tested for Oxidosqualene-lanosterol cyclase inhibition in T. cruziMore data for this Ligand-Target Pair
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+3nMAssay Description:Tested for Oxidosqualene-lanosterol cyclase inhibition in ratMore data for this Ligand-Target Pair
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: 2.60E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: 4.80E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: 8.00E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: 1.20E+4nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+4nMAssay Description:Tested for Oxidosqualene-lanosterol cyclase inhibition in P. cariniiMore data for this Ligand-Target Pair
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: 2.10E+4nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: 2.30E+4nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: 3.00E+4nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: 1.10E+5nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: >1.00E+6nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: >1.00E+6nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair