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Found 32 with Last Name = 'suh' and Initial = 'dy'
TargetLanosterol synthase(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50133285((E)-3-Carboxy-acrylateallyl-{6-[4-(4-chloro-benzoy...)
Affinity DataIC50:  4.30nMAssay Description:Tested for Oxidosqualene-lanosterol cyclase inhibition in T. bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50133285((E)-3-Carboxy-acrylateallyl-{6-[4-(4-chloro-benzoy...)
Affinity DataIC50:  4.60nMAssay Description:Tested for Oxidosqualene-lanosterol cyclase inhibition in P. cariniiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50095601(CHEMBL25405 | [4-(1-Aza-bicyclo[2.2.2]oct-3-yloxy)...)
Affinity DataIC50:  22nMAssay Description:Tested for Oxidosqualene-lanosterol cyclase inhibition in T. bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Rattus norvegicus)
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50133285((E)-3-Carboxy-acrylateallyl-{6-[4-(4-chloro-benzoy...)
Affinity DataIC50:  49nMAssay Description:Tested for Oxidosqualene-lanosterol cyclase inhibition in ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50133285((E)-3-Carboxy-acrylateallyl-{6-[4-(4-chloro-benzoy...)
Affinity DataIC50:  71nMAssay Description:Tested for Oxidosqualene-lanosterol cyclase inhibition in T. cruziMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50095601(CHEMBL25405 | [4-(1-Aza-bicyclo[2.2.2]oct-3-yloxy)...)
Affinity DataIC50:  92nMAssay Description:Tested for Oxidosqualene-lanosterol cyclase inhibition in P. cariniiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Rattus norvegicus)
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50095601(CHEMBL25405 | [4-(1-Aza-bicyclo[2.2.2]oct-3-yloxy)...)
Affinity DataIC50:  160nMAssay Description:Tested for Oxidosqualene-lanosterol cyclase inhibition in ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065348((1S,4aR,5S)-1,4a-Dimethyl-6-methylene-5-[2-(2-oxo-...)
Affinity DataIC50:  250nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065336((1S,4aS,5R)-1,4a-Dimethyl-6-oxo-5-[2-(2-oxo-2,5-di...)
Affinity DataIC50:  260nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50133286(CHEMBL132091 | [3-(Biphenyl-4-yloxy)-propyl]-dimet...)
Affinity DataIC50:  280nMAssay Description:Tested for Oxidosqualene-lanosterol cyclase inhibition in T. bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50095601(CHEMBL25405 | [4-(1-Aza-bicyclo[2.2.2]oct-3-yloxy)...)
Affinity DataIC50:  400nMAssay Description:Tested for Oxidosqualene-lanosterol cyclase inhibition in T. cruziMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50133286(CHEMBL132091 | [3-(Biphenyl-4-yloxy)-propyl]-dimet...)
Affinity DataIC50:  750nMAssay Description:Tested for Oxidosqualene-lanosterol cyclase inhibition in T. cruziMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065344(CHEMBL89088 | methyl 5,8a-dimethyl-1-[2-(2-oxo-2,5...)
Affinity DataIC50:  1.00E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065343((1S,4aR,5S,6S)-6-Hydroxymethyl-1,4a-dimethyl-5-[2-...)
Affinity DataIC50:  1.60E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065347(3-[2-((1S,5S,8aR)-5-Methoxymethyl-5,8a-dimethyl-2-...)
Affinity DataIC50:  1.70E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065339((1S,4aS)-6-Formyl-1,4a-dimethyl-5-[2-(2-oxo-2,5-di...)
Affinity DataIC50:  1.70E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065352((1S,4aR,5S)-1,4a-Dimethyl-6-methylene-5-[2-(2-oxo-...)
Affinity DataIC50:  2.00E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065335((1S,4aS,5R,6S)-6-Hydroxy-1,4a-dimethyl-5-[2-(2-oxo...)
Affinity DataIC50:  2.00E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Rattus norvegicus)
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50133286(CHEMBL132091 | [3-(Biphenyl-4-yloxy)-propyl]-dimet...)
Affinity DataIC50:  2.50E+3nMAssay Description:Tested for Oxidosqualene-lanosterol cyclase inhibition in ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065342((1S,4aS,5R)-1,4a-Dimethyl-6-oxo-5-[2-(2-oxo-tetrah...)
Affinity DataIC50:  2.60E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065333(6-Hydroxymethyl-1,4a-dimethyl-5-[2-(2-oxo-2,5-dihy...)
Affinity DataIC50:  4.00E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065345((1S,4aR,5S)-1,4a,6-Trimethyl-5-[2-(2-oxo-tetrahydr...)
Affinity DataIC50:  4.80E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065346((1S,4aR,5S)-1,4a-Dimethyl-6-methylene-5-[2-(5-oxo-...)
Affinity DataIC50:  6.00E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065341((1R,6S,9aS)-6,9a-Dimethyl-3-oxo-1-[2-(5-oxo-2,5-di...)
Affinity DataIC50:  8.00E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065337((1S,4aR,5S)-5-((Z)-5-Hydroxy-3-hydroxymethyl-pent-...)
Affinity DataIC50:  1.20E+4nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50133286(CHEMBL132091 | [3-(Biphenyl-4-yloxy)-propyl]-dimet...)
Affinity DataIC50:  1.60E+4nMAssay Description:Tested for Oxidosqualene-lanosterol cyclase inhibition in P. cariniiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065351((Z)-2-[2-((1S,5S,8aR)-5-Hydroxymethyl-5,8a-dimethy...)
Affinity DataIC50:  2.10E+4nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065350((1S,4aR,5S)-1,4a-Dimethyl-6-methylene-5-[2-(2-oxo-...)
Affinity DataIC50:  2.30E+4nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065338(3-[2-((1S,5S,8aR)-5-Hydroxymethyl-5,8a-dimethyl-2-...)
Affinity DataIC50:  3.00E+4nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065349(4-[2-((1S,5S,8aR)-5-Hydroxymethyl-5,8a-dimethyl-2-...)
Affinity DataIC50:  1.10E+5nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065340((1S,4aR,5S)-5-(2-Furan-3-yl-ethyl)-1,4a-dimethyl-6...)
Affinity DataIC50: >1.00E+6nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065334((1S,4aS,5R,6R)-6-Hydroxy-6-hydroxymethyl-1,4a-dime...)
Affinity DataIC50: >1.00E+6nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed