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Found 265 with Last Name = 'utz' and Initial = 'w'
TargetAdenosine receptor A1(BOVINE)
Forschungszentrum JüLich

Curated by ChEMBL
LigandPNGBDBM50062858(8-Cyclopentyl-3-(2-fluoro-propyl)-1-propyl-3,7-dih...)
Affinity DataKi:  0.0940nMAssay Description:Displacement of [3H]-CPX from Adenosine A1 receptor of bovine brain cerebral cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Forschungszentrum JüLich

Curated by ChEMBL
LigandPNGBDBM21173(1,3-dipropyl-8-cyclopentylxanthine | 8-cyclopentyl...)
Affinity DataKi:  0.155nMAssay Description:Displacement of [3H]-CPX from Adenosine A1 receptor of bovine brain cerebral cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Forschungszentrum JüLich

Curated by ChEMBL
LigandPNGBDBM21173(1,3-dipropyl-8-cyclopentylxanthine | 8-cyclopentyl...)
Affinity DataKi:  0.155nMAssay Description:Displacement of [3H]-CPX from Adenosine A1 receptor of bovine brain cerebral cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Forschungszentrum JüLich

Curated by ChEMBL
LigandPNGBDBM50062852(8-Cyclopentyl-3-(3-fluoro-propyl)-1-propyl-3,7-dih...)
Affinity DataKi:  0.180nMAssay Description:In vitro binding affinity for Adenosine A1 receptor of bovine cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Forschungszentrum JüLich

Curated by ChEMBL
LigandPNGBDBM50062852(8-Cyclopentyl-3-(3-fluoro-propyl)-1-propyl-3,7-dih...)
Affinity DataKi:  0.183nMAssay Description:Displacement of [3H]-CPX from Adenosine A1 receptor of bovine brain cerebral cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Forschungszentrum JüLich

Curated by ChEMBL
LigandPNGBDBM50062853(8-Cyclopentyl-1-(3-fluoro-propyl)-3,7-dihydro-puri...)
Affinity DataKi:  0.216nMAssay Description:Displacement of [3H]-CPX from Adenosine A1 receptor of bovine brain cerebral cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Forschungszentrum JüLich

Curated by ChEMBL
LigandPNGBDBM50062856(8-Cyclopentyl-3-((E)-3-iodo-propenyl)-1-propyl-3,7...)
Affinity DataKi:  0.237nMAssay Description:Displacement of [3H]-CPX from Adenosine A1 receptor of bovine brain cerebral cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50203821(CHEMBL374749 | biphenyl-4-carboxylic acid {4-[4-(2...)
Affinity DataKi:  0.280nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 expressed in CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Forschungszentrum JüLich

Curated by ChEMBL
LigandPNGBDBM50062859(8-Cyclopentyl-1-ethoxymethyl-3-propyl-3,7-dihydro-...)
Affinity DataKi:  0.286nMAssay Description:Displacement of [3H]-CPX from Adenosine A1 receptor of bovine brain cerebral cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Forschungszentrum JüLich

Curated by ChEMBL
LigandPNGBDBM50011842(8-Cyclopentyl-3-methyl-1-propyl-3,7-dihydro-purine...)
Affinity DataKi:  0.310nMAssay Description:Displacement of [3H]-CPX from Adenosine A1 receptor of bovine brain cerebral cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50203819(4-(6-fluoropyridin-2-yl)-N-{4-[4-(2-methoxyphenyl)...)
Affinity DataKi:  0.370nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 expressed in CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50203820(4-(6-fluoropyridin-3-yl)-N-{4-[4-(2-methoxyphenyl)...)
Affinity DataKi:  0.450nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 expressed in CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Forschungszentrum JüLich

Curated by ChEMBL
LigandPNGBDBM50062855(8-Cyclopentyl-3-ethoxymethyl-1-propyl-3,7-dihydro-...)
Affinity DataKi:  0.493nMAssay Description:Displacement of [3H]-CPX from Adenosine A1 receptor of bovine brain cerebral cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Forschungszentrum JüLich

Curated by ChEMBL
LigandPNGBDBM50011824(8-Cyclopentyl-1-methyl-3-propyl-3,7-dihydro-purine...)
Affinity DataKi:  0.526nMAssay Description:Displacement of [3H]-CPX from Adenosine A1 receptor of bovine brain cerebral cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM85093(CAS_3853 | CHEMBL267014 | CHEMBL555670 | L 745,870...)
Affinity DataKi:  0.617nMAssay Description:Ability to displace [3H]spiperone from dopamine receptor D4.4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50116766((-)-Pramipexole | (6S)-N(6)-propyl-4,5,6,7-tetrahy...)
Affinity DataKi:  0.880nMAssay Description:High inhibition constant against [3H]-spiperone binding to human Dopamine receptor D3 expressed in CHO cellsMore data for this Ligand-Target Pair
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM55121(3-HYDROXYTYRAMINE HYDROCHLORIDE | 4-(2-aminoethyl)...)
Affinity DataKi:  1.20nMAssay Description:Binding Affinity was tested on the high affinity site of Dopamine receptor D4.4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAdenosine receptor A1(BOVINE)
Forschungszentrum JüLich

Curated by ChEMBL
LigandPNGBDBM50062857(8-Cyclopentyl-1-(2-fluoro-propyl)-3-propyl-3,7-dih...)
Affinity DataKi:  1.23nMAssay Description:Displacement of [3H]-CPX from Adenosine A1 receptor of bovine brain cerebral cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50109952(3-((4-(4-chlorophenyl)piperazin-1-yl)methyl)-7-eth...)
Affinity DataKi:  1.23nMAssay Description:Ability to displace [3H]spiperone from dopamine receptor D4.4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM84637(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
Affinity DataKi:  1.80nMAssay Description:High inhibition constant against [3H]-spiperone binding to human Dopamine receptor D4.4 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM55121(3-HYDROXYTYRAMINE HYDROCHLORIDE | 4-(2-aminoethyl)...)
Affinity DataKi:  1.80nMAssay Description:Binding Affinity on high Affinity Site of Bovine dopamine receptor D2. Tested for ability to displace the radioligand [3H]pramipexole was testedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide(RAT)
Georg-August-University

Curated by PDSP Ki Database
LigandPNGBDBM50250019(CHEMBL524658 | PACAP | PACAP(1-38) | PACAP-38 | PA...)
Affinity DataKi:  1.90nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50473574(CHEMBL609112)
Affinity DataKi:  1.91nMAssay Description:Ability to displace [3H]spiperone from dopamine receptor D4.4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50102712(2-((4-(4-chlorophenyl)piperazin-1-yl)methyl)-pyraz...)
Affinity DataKi:  2.19nMAssay Description:Ability to displace [3H]spiperone from dopamine receptor D4.4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50102712(2-((4-(4-chlorophenyl)piperazin-1-yl)methyl)-pyraz...)
Affinity DataKi:  2.20nMAssay Description:Binding affinity against human dopamine receptor D4.4 using radioligand [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50073805(3-((4-(4-chlorophenyl)piperazin-1-yl)methyl)H-pyra...)
Affinity DataKi:  2.29nMAssay Description:Ability to displace [3H]spiperone from dopamine receptor D4.4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50109941(3-((4-(4-chlorophenyl)piperazin-1-yl)methyl)-7-met...)
Affinity DataKi:  2.69nMAssay Description:Ability to displace [3H]spiperone from dopamine receptor D4.4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50073800(3-[4-(4-Iodo-phenyl)-piperazin-1-ylmethyl]-pyrazol...)
Affinity DataKi:  3.02nMAssay Description:Ability to displace [3H]spiperone from dopamine receptor D4.4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide(RAT)
Georg-August-University

Curated by PDSP Ki Database
LigandPNGBDBM81825(PACAP(1-23),VIP(24-28))
Affinity DataKi:  3.10nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50102717(6-[4-(4-Chloro-phenyl)-piperazin-1-ylmethyl]-pyraz...)
Affinity DataKi:  3.10nMAssay Description:Binding affinity against human dopamine receptor D4.4 using radioligand [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50073811(3-[4-(3-Chloro-phenyl)-piperazin-1-ylmethyl]-pyraz...)
Affinity DataKi:  3.89nMAssay Description:Ability to displace [3H]spiperone from dopamine receptor D4.4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50473581(CHEMBL611793)
Affinity DataKi:  4.37nMAssay Description:Ability to displace [3H]spiperone from dopamine receptor D4.4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide(RAT)
Georg-August-University

Curated by PDSP Ki Database
LigandPNGBDBM50250068(CHEMBL501240 | PACAP(1-27) | PACAP-27 | [Glu3]PACA...)
Affinity DataKi:  4.70nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50473578(CHEMBL218787)
Affinity DataKi:  5.01nMAssay Description:Ability to displace [3H]spiperone from dopamine receptor D4.4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50085331((4-Ethynyl-cyclohex-3-enyl)-dipropyl-amine | 4-eth...)
Affinity DataKi:  5.20nMAssay Description:Binding Affinity was tested on the high affinity site of Dopamine receptor D3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50105731((S)-7-Dipropylamino-5,6,7,8-tetrahydro-indolizine-...)
Affinity DataKi:  5.30nMAssay Description:High inhibition constant against [3H]-spiperone binding to human Dopamine receptor D3 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50473582(CHEMBL609116)
Affinity DataKi:  5.62nMAssay Description:Ability to displace [3H]spiperone from dopamine receptor D4.4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50079645(2-{4-[4-(4-Chloro-phenyl)-piperazin-1-ylmethyl]-1H...)
Affinity DataKi:  5.75nMAssay Description:Ability to displace [3H]spiperone from dopamine receptor D4.4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide(RAT)
Georg-August-University

Curated by PDSP Ki Database
LigandPNGBDBM81824(PACAP(1-33,Cys34))
Affinity DataKi:  6.40nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(BOVINE)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM55121(3-HYDROXYTYRAMINE HYDROCHLORIDE | 4-(2-aminoethyl)...)
Affinity DataKi:  7nMAssay Description:Binding Affinity was tested on High Affinity Site of Bovine Dopamine receptor D1. Tested for ability to displace the radioligand [3H]-SCH- 23390More data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50164427((S)-7-Dipropylamino-5,6,7,8-tetrahydro-indolizine-...)
Affinity DataKi:  7.20nMAssay Description:High inhibition constant against [3H]-spiperone binding to human Dopamine receptor D3 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50116766((-)-Pramipexole | (6S)-N(6)-propyl-4,5,6,7-tetrahy...)
Affinity DataKi:  8.10nMAssay Description:High inhibition constant against [3H]-spiperone binding to human Dopamine receptor D4.4 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50079646(2-{5-[4-(4-Chloro-phenyl)-piperazin-1-ylmethyl]-1H...)
Affinity DataKi:  9.55nMAssay Description:Ability to displace [3H]spiperone from dopamine receptor D4.4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM55121(3-HYDROXYTYRAMINE HYDROCHLORIDE | 4-(2-aminoethyl)...)
Affinity DataKi:  11nMAssay Description:Binding Affinity was tested on high Affinity Site of Bovine Dopamine D2 Receptor. Tested for ability to displace the radioligand [3H]spiperone was te...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50203820(4-(6-fluoropyridin-3-yl)-N-{4-[4-(2-methoxyphenyl)...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]spiperone from human dopamine D2(short) expressed in CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50085331((4-Ethynyl-cyclohex-3-enyl)-dipropyl-amine | 4-eth...)
Affinity DataKi:  15nMAssay Description:Binding Affinity was tested on high Affinity Site of Bovine dopamine receptor D2. Tested for ability to displace the radioligand [3H]pramipexoleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50203820(4-(6-fluoropyridin-3-yl)-N-{4-[4-(2-methoxyphenyl)...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]spiperone from human dopamine D2(long) expressed in CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)
Affinity DataKi:  15.8nMAssay Description:Ability to displace [3H]spiperone from dopamine receptor D4.4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)
Affinity DataKi:  16nMAssay Description:Binding affinity against human dopamine receptor D4.4 using radioligand [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50085333(CHEMBL163087 | Dipropyl-(4-trimethylsilanylethynyl...)
Affinity DataKi:  16nMAssay Description:Binding Affinity was tested on relative proportion of High Affinity Site of Dopamine receptor D2LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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