Affinity DataKi: 2.94E+3nMAssay Description:Displacement of [3H]CHA from adenosine A1 receptor in rat brain cortical membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Institut FüR Biowissenschaften
Curated by ChEMBL
Institut FüR Biowissenschaften
Curated by ChEMBL
Affinity DataKi: 9.40E+3nMAssay Description:Displacement of [3H]CGS21680 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Institut FüR Biowissenschaften
Curated by ChEMBL
Institut FüR Biowissenschaften
Curated by ChEMBL
Affinity DataKi: 1.37E+4nMAssay Description:Displacement of [3H]CGS21680 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.70E+4nMAssay Description:Displacement of [3H]CHA from adenosine A1 receptor in rat brain cortical membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Institut FüR Biowissenschaften
Curated by ChEMBL
Institut FüR Biowissenschaften
Curated by ChEMBL
Affinity DataKi: 2.20E+4nMAssay Description:Displacement of [3H]CGS21680 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 2.60E+4nMAssay Description:Displacement of [3H]CHA from adenosine A1 receptor in rat brain cortical membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 13.7nMAssay Description:Inhibitory activity against Cathepsin B was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 21.6nMAssay Description:Inhibitory activity against Cathepsin B was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 60.9nMAssay Description:Inhibitory activity against Cathepsin B was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 344nMAssay Description:Inhibition of alpha-glucosidaseMore data for this Ligand-Target Pair
Affinity DataIC50: 488nMAssay Description:Inhibition of Clostridium perfringens neuraminidaseMore data for this Ligand-Target Pair
Affinity DataIC50: 531nMAssay Description:Inhibition of alpha-glucosidaseMore data for this Ligand-Target Pair
Affinity DataIC50: 6.79E+3nMAssay Description:Inhibition of bovine cathepsin B after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.80E+3nMAssay Description:Inhibition of bovine cathepsin B after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.82E+3nMAssay Description:Inhibition of alpha-glucosidaseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibitory activity against histone deacetylase (HDAC)More data for this Ligand-Target Pair
Affinity DataIC50: 2.51E+4nMAssay Description:Inhibition of truncated recombinant MT1-MMP expressed in Escherichia coli JM109 after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory activity against histone deacetylase (HDAC)More data for this Ligand-Target Pair
Affinity DataIC50: 3.12E+4nMAssay Description:Inhibition of truncated recombinant MT1-MMP expressed in Escherichia coli JM109 after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.10E+4nMAssay Description:Inhibitory activity against histone deacetylase (HDAC)More data for this Ligand-Target Pair
Affinity DataIC50: 8.00E+4nMAssay Description:Inhibitory activity against histone deacetylase (HDAC)More data for this Ligand-Target Pair